FI85376C - Foerfarande foer framstaellning av terapeutiskt aktiva 6-(substituerad metylen) penicillanderivat. - Google Patents

Foerfarande foer framstaellning av terapeutiskt aktiva 6-(substituerad metylen) penicillanderivat. Download PDF

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Publication number
FI85376C
FI85376C FI850375A FI850375A FI85376C FI 85376 C FI85376 C FI 85376C FI 850375 A FI850375 A FI 850375A FI 850375 A FI850375 A FI 850375A FI 85376 C FI85376 C FI 85376C
Authority
FI
Finland
Prior art keywords
formula
compound
mixture
give
nmr
Prior art date
Application number
FI850375A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI850375A0 (fi
FI85376B (fi
FI850375L (fi
Inventor
Yuhpyng Liang Chen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI850375A0 publication Critical patent/FI850375A0/fi
Publication of FI850375L publication Critical patent/FI850375L/fi
Priority to FI902112A priority Critical patent/FI902112A0/fi
Priority to FI902113A priority patent/FI902113A0/fi
Priority to FI902114A priority patent/FI902114A0/fi
Publication of FI85376B publication Critical patent/FI85376B/fi
Application granted granted Critical
Publication of FI85376C publication Critical patent/FI85376C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI850375A 1984-01-30 1985-01-29 Foerfarande foer framstaellning av terapeutiskt aktiva 6-(substituerad metylen) penicillanderivat. FI85376C (fi)

Priority Applications (3)

Application Number Priority Date Filing Date Title
FI902112A FI902112A0 (fi) 1984-01-30 1990-04-26 Foerfarande foer framstaellning av b-laktamas inhiberande 6-hydroximetylpenicillansyraderivat.
FI902113A FI902113A0 (fi) 1984-01-30 1990-04-26 6-metylenpenicillansyraderivat.
FI902114A FI902114A0 (fi) 1984-01-30 1990-04-26 6-hydroximetylpenicillansyraderivat.

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US57535484A 1984-01-30 1984-01-30
US57535484 1984-01-30

Publications (4)

Publication Number Publication Date
FI850375A0 FI850375A0 (fi) 1985-01-29
FI850375L FI850375L (fi) 1985-07-31
FI85376B FI85376B (fi) 1991-12-31
FI85376C true FI85376C (fi) 1992-04-10

Family

ID=24299979

Family Applications (1)

Application Number Title Priority Date Filing Date
FI850375A FI85376C (fi) 1984-01-30 1985-01-29 Foerfarande foer framstaellning av terapeutiskt aktiva 6-(substituerad metylen) penicillanderivat.

Country Status (15)

Country Link
JP (1) JPS61109791A (xx)
KR (1) KR880001029B1 (xx)
CS (5) CS248733B2 (xx)
DD (3) DD247677A5 (xx)
EG (1) EG16904A (xx)
ES (5) ES8604972A1 (xx)
FI (1) FI85376C (xx)
HU (2) HU194891B (xx)
IL (1) IL74190A (xx)
NO (1) NO165594C (xx)
PL (5) PL145130B1 (xx)
PT (1) PT79893B (xx)
SU (4) SU1395144A3 (xx)
YU (5) YU44770B (xx)
ZA (1) ZA85682B (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0276942B1 (en) * 1987-01-27 1992-04-01 Pfizer Inc. 6-beta(substituted)-(s)-hydroxymethylpenicillanic acids and derivatives thereof
US6156745A (en) 1997-12-29 2000-12-05 Research Corporation Technologies, Inc. 2β-substituted-6-alkylidene penicillanic acid derivatives as β-lactamase inhibitors
US6407091B1 (en) 1999-04-15 2002-06-18 Research Corporation Technologies, Inc. β-lactamase inhibiting compounds
ES2272795T3 (es) 2001-07-24 2007-05-01 Southern Methodist University Foundation For Research 7-alquildieno-3-sustituidos-3-cefem-4-carboxilatos como inhibidores de beta-lactamasa.
JP2005525399A (ja) 2002-04-04 2005-08-25 アラムクス エルエルシー セリンおよびメタロ−β−ラクタマーゼの阻害剤
GB0711776D0 (en) * 2007-06-18 2007-07-25 Syngenta Participations Ag Substituted aromatic heterocyclic compounds as fungicides
JP6183053B2 (ja) * 2012-08-22 2017-08-23 宇部興産株式会社 テトラヒドロピラニルピリミジン化合物の製造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors

Also Published As

Publication number Publication date
NO165594B (no) 1990-11-26
YU119787A (en) 1988-04-30
FI850375A0 (fi) 1985-01-29
PL149242B1 (en) 1990-01-31
ZA85682B (en) 1986-09-24
PT79893A (en) 1985-02-01
CS248733B2 (en) 1987-02-12
YU44636B (en) 1990-10-31
SU1503683A3 (ru) 1989-08-23
YU119487A (en) 1988-02-29
PT79893B (en) 1987-02-03
YU119687A (en) 1988-04-30
ES8704952A1 (es) 1987-04-16
SU1395144A3 (ru) 1988-05-07
ES548427A0 (es) 1987-05-01
ES548426A0 (es) 1986-11-16
CS248749B2 (en) 1987-02-12
ES8700860A1 (es) 1986-11-16
PL251750A1 (en) 1985-12-17
ES548428A0 (es) 1987-01-16
YU119587A (en) 1988-02-29
HUT40443A (en) 1986-12-28
IL74190A0 (en) 1985-04-30
PL256014A1 (en) 1986-12-02
YU44770B (en) 1991-02-28
FI85376B (fi) 1991-12-31
JPS61109791A (ja) 1986-05-28
ES8702916A1 (es) 1987-01-16
CS248746B2 (en) 1987-02-12
ES548429A0 (es) 1987-04-16
PL145130B1 (en) 1988-08-31
ES8604972A1 (es) 1986-02-16
SU1508961A3 (ru) 1989-09-15
DD247677A5 (de) 1987-07-15
YU44805B (en) 1991-02-28
PL256016A1 (en) 1986-12-02
NO165594C (no) 1991-03-06
DD234015A5 (de) 1986-03-19
CS248748B2 (en) 1987-02-12
DD247678A5 (de) 1987-07-15
ES8705451A1 (es) 1987-05-01
SU1396969A3 (ru) 1988-05-15
NO850350L (no) 1985-07-31
HU194891B (en) 1988-03-28
PL145990B1 (en) 1988-12-31
HUT37799A (en) 1986-02-28
YU44635B (en) 1990-10-31
HU194567B (en) 1988-02-29
YU14085A (en) 1987-12-31
CS248747B2 (en) 1987-02-12
PL256015A1 (en) 1986-11-18
KR850005445A (ko) 1985-08-26
IL74190A (en) 1989-09-28
EG16904A (en) 1992-06-30
FI850375L (fi) 1985-07-31
YU44634B (en) 1990-10-31
KR880001029B1 (ko) 1988-06-15
ES539890A0 (es) 1986-02-16
PL256013A1 (en) 1986-10-21
PL149797B1 (en) 1990-03-31
PL147514B1 (en) 1989-06-30

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Owner name: PFIZER INC.