EE200000610A - p38 heterotsüklilised inhibiitorid - Google Patents

p38 heterotsüklilised inhibiitorid

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Publication number
EE200000610A
EE200000610A EEP200000610A EEP200000610A EE200000610A EE 200000610 A EE200000610 A EE 200000610A EE P200000610 A EEP200000610 A EE P200000610A EE P200000610 A EEP200000610 A EE P200000610A EE 200000610 A EE200000610 A EE 200000610A
Authority
EE
Estonia
Prior art keywords
heterocyclic inhibitors
heterocyclic
inhibitors
Prior art date
Application number
EEP200000610A
Other languages
English (en)
Estonian (et)
Inventor
Gerald Salituro Francesco
P. Galullo Vincent
Bellon Steven
W. Bemis Guy
E. Cochran John
Original Assignee
Vertex Pharmaceuticals Incorporated
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharmaceuticals Incorporated filed Critical Vertex Pharmaceuticals Incorporated
Publication of EE200000610A publication Critical patent/EE200000610A/xx

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
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