DK1077943T3 - Heterocykliske inhibitorer af p38 - Google Patents
Heterocykliske inhibitorer af p38Info
- Publication number
- DK1077943T3 DK1077943T3 DK99920427T DK99920427T DK1077943T3 DK 1077943 T3 DK1077943 T3 DK 1077943T3 DK 99920427 T DK99920427 T DK 99920427T DK 99920427 T DK99920427 T DK 99920427T DK 1077943 T3 DK1077943 T3 DK 1077943T3
- Authority
- DK
- Denmark
- Prior art keywords
- heterocyclic inhibitors
- heterocyclic
- inhibitors
- Prior art date
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
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- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/06—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals
- C07D295/073—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals with the ring nitrogen atoms and the substituents separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
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- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
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US8505398P | 1998-05-11 | 1998-05-11 | |
US12762699P | 1999-04-01 | 1999-04-01 | |
US12909999P | 1999-04-13 | 1999-04-13 | |
PCT/US1999/010291 WO1999058502A1 (en) | 1998-05-11 | 1999-05-11 | Heterocyclic inhibitors of p38 |
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DK1077943T3 true DK1077943T3 (da) | 2009-03-16 |
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Application Number | Title | Priority Date | Filing Date |
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DK99920427T DK1077943T3 (da) | 1998-05-11 | 1999-05-11 | Heterocykliske inhibitorer af p38 |
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EP (3) | EP2062879A1 (da) |
JP (2) | JP4704560B2 (da) |
KR (1) | KR100696219B1 (da) |
CN (1) | CN1306512A (da) |
AP (1) | AP2000001996A0 (da) |
AT (1) | ATE417828T1 (da) |
AU (1) | AU764047B2 (da) |
BG (1) | BG65025B1 (da) |
BR (1) | BR9911786A (da) |
CA (1) | CA2331460C (da) |
CZ (1) | CZ300702B6 (da) |
DE (1) | DE69940115D1 (da) |
DK (1) | DK1077943T3 (da) |
EA (1) | EA200001176A1 (da) |
EE (1) | EE200000610A (da) |
ES (1) | ES2318893T3 (da) |
GE (1) | GEP20032954B (da) |
HK (1) | HK1034907A1 (da) |
HU (1) | HUP0105174A3 (da) |
IL (2) | IL139479A0 (da) |
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NO (1) | NO319755B1 (da) |
NZ (1) | NZ508653A (da) |
PL (1) | PL198352B1 (da) |
PT (1) | PT1077943E (da) |
SK (1) | SK286689B6 (da) |
TW (1) | TWI249527B (da) |
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1999
- 1999-05-10 MY MYPI99001841A patent/MY132496A/en unknown
- 1999-05-11 EP EP08021820A patent/EP2062879A1/en not_active Withdrawn
- 1999-05-11 EE EEP200000610A patent/EE200000610A/xx unknown
- 1999-05-11 TW TW088107631A patent/TWI249527B/zh not_active IP Right Cessation
- 1999-05-11 AT AT99920427T patent/ATE417828T1/de active
- 1999-05-11 JP JP2000548306A patent/JP4704560B2/ja not_active Expired - Fee Related
- 1999-05-11 IL IL13947999A patent/IL139479A0/xx unknown
- 1999-05-11 EP EP10177856A patent/EP2336111A1/en not_active Withdrawn
- 1999-05-11 AP APAP/P/2000/001996A patent/AP2000001996A0/en unknown
- 1999-05-11 KR KR1020007012601A patent/KR100696219B1/ko not_active IP Right Cessation
- 1999-05-11 GE GEAP19995666A patent/GEP20032954B/en unknown
- 1999-05-11 CN CN99807647A patent/CN1306512A/zh active Pending
- 1999-05-11 CA CA2331460A patent/CA2331460C/en not_active Expired - Fee Related
- 1999-05-11 AU AU37923/99A patent/AU764047B2/en not_active Ceased
- 1999-05-11 NZ NZ508653A patent/NZ508653A/en not_active IP Right Cessation
- 1999-05-11 PL PL344046A patent/PL198352B1/pl not_active IP Right Cessation
- 1999-05-11 CZ CZ20004172A patent/CZ300702B6/cs not_active IP Right Cessation
- 1999-05-11 BR BR9911786-0A patent/BR9911786A/pt not_active Application Discontinuation
- 1999-05-11 SK SK1688-2000A patent/SK286689B6/sk not_active IP Right Cessation
- 1999-05-11 UA UA2000127087A patent/UA74325C2/uk unknown
- 1999-05-11 DK DK99920427T patent/DK1077943T3/da active
- 1999-05-11 ES ES99920427T patent/ES2318893T3/es not_active Expired - Lifetime
- 1999-05-11 HU HU0105174A patent/HUP0105174A3/hu unknown
- 1999-05-11 EA EA200001176A patent/EA200001176A1/ru unknown
- 1999-05-11 PT PT99920427T patent/PT1077943E/pt unknown
- 1999-05-11 EP EP99920427A patent/EP1077943B1/en not_active Expired - Lifetime
- 1999-05-11 DE DE69940115T patent/DE69940115D1/de not_active Expired - Lifetime
- 1999-05-11 WO PCT/US1999/010291 patent/WO1999058502A1/en not_active Application Discontinuation
-
2000
- 2000-11-05 IL IL139479A patent/IL139479A/en not_active IP Right Cessation
- 2000-11-10 NO NO20005673A patent/NO319755B1/no not_active IP Right Cessation
- 2000-11-10 IS IS5711A patent/IS5711A/is unknown
- 2000-12-07 BG BG105031A patent/BG65025B1/bg unknown
- 2000-12-21 US US09/746,722 patent/US6632945B2/en not_active Expired - Fee Related
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2001
- 2001-08-13 HK HK01105642.0A patent/HK1034907A1/xx not_active IP Right Cessation
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2003
- 2003-08-08 US US10/638,126 patent/US7115637B2/en not_active Expired - Fee Related
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2006
- 2006-05-08 US US11/430,512 patent/US7423049B2/en not_active Expired - Fee Related
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2008
- 2008-08-01 US US12/184,996 patent/US20090075981A1/en not_active Abandoned
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2010
- 2010-03-12 JP JP2010056785A patent/JP2010150282A/ja not_active Withdrawn
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