DK0676409T3 - Erythromycinderivater, fremgangsmåde til deres fremstilling og deres anvendelse som lægemidler - Google Patents

Erythromycinderivater, fremgangsmåde til deres fremstilling og deres anvendelse som lægemidler

Info

Publication number
DK0676409T3
DK0676409T3 DK95400763T DK95400763T DK0676409T3 DK 0676409 T3 DK0676409 T3 DK 0676409T3 DK 95400763 T DK95400763 T DK 95400763T DK 95400763 T DK95400763 T DK 95400763T DK 0676409 T3 DK0676409 T3 DK 0676409T3
Authority
DK
Denmark
Prior art keywords
pharmaceuticals
processes
preparation
erythromycin derivatives
erythromycin
Prior art date
Application number
DK95400763T
Other languages
Danish (da)
English (en)
Inventor
Jean-Francois Chantot
Martret Odile Le
Constantin Agouridas
Alexis Denis
Yannick Benedetti
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of DK0676409T3 publication Critical patent/DK0676409T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
DK95400763T 1994-04-08 1995-04-06 Erythromycinderivater, fremgangsmåde til deres fremstilling og deres anvendelse som lægemidler DK0676409T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9404154A FR2718450B1 (fr) 1994-04-08 1994-04-08 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Publications (1)

Publication Number Publication Date
DK0676409T3 true DK0676409T3 (da) 2003-06-23

Family

ID=9461886

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95400763T DK0676409T3 (da) 1994-04-08 1995-04-06 Erythromycinderivater, fremgangsmåde til deres fremstilling og deres anvendelse som lægemidler

Country Status (49)

Country Link
US (2) US5656607A (oth)
EP (1) EP0676409B1 (oth)
JP (1) JP3000023B2 (oth)
KR (1) KR100317148B1 (oth)
CN (1) CN1059445C (oth)
AP (1) AP587A (oth)
AT (1) ATE234853T1 (oth)
AU (1) AU684939B2 (oth)
BG (1) BG61916B1 (oth)
BR (1) BR9506147A (oth)
CA (1) CA2164638C (oth)
CO (1) CO4370097A1 (oth)
CZ (1) CZ296005B6 (oth)
DE (1) DE69529934T2 (oth)
DK (1) DK0676409T3 (oth)
DZ (1) DZ1869A1 (oth)
EE (1) EE04498B1 (oth)
ES (1) ES2189820T3 (oth)
FI (1) FI111264B (oth)
FR (1) FR2718450B1 (oth)
GB (1) GB2288174A (oth)
GE (1) GEP19991836B (oth)
HR (1) HRP950217B1 (oth)
HU (1) HU215396B (oth)
IL (1) IL112954A (oth)
IS (1) IS1865B (oth)
JO (1) JO1850B1 (oth)
LV (1) LV11182B (oth)
MA (1) MA23501A1 (oth)
MD (1) MD663G2 (oth)
MY (1) MY114672A (oth)
NO (1) NO308361B1 (oth)
NZ (1) NZ284498A (oth)
OA (1) OA10200A (oth)
PE (1) PE2896A1 (oth)
PL (1) PL180837B1 (oth)
PT (1) PT676409E (oth)
RO (1) RO115634B1 (oth)
RU (1) RU2141965C1 (oth)
SA (1) SA97170757A (oth)
SI (1) SI0676409T1 (oth)
SK (1) SK284079B6 (oth)
SV (1) SV1995000018A (oth)
TN (1) TNSN95026A1 (oth)
TW (1) TW316908B (oth)
UA (1) UA44705C2 (oth)
WO (1) WO1995027720A1 (oth)
YU (1) YU49221B (oth)
ZA (1) ZA952059B (oth)

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FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2745289B1 (fr) * 1996-02-28 1998-05-29 Roussel Uclaf Nouveaux derives de l'acide 1(2h) quinoleine carboxylique, leur procede de preparation et leur application a la synthese de produits doues de proprietes antibiotiques
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FR2751656B1 (fr) * 1996-07-24 1998-10-16 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
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DE69733723T2 (de) * 1996-09-04 2006-04-20 Abbott Laboratories, Abbott Park 6-o-Substituierte Ketoliden mit antibakteriellen Wirkung
FR2757168B1 (fr) * 1996-12-12 1999-06-11 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
WO1998040392A1 (fr) * 1997-03-10 1998-09-17 Taisho Pharmaceutical Co., Ltd. Derives d'erythromycine a
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FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
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FR2786188B1 (fr) * 1998-11-24 2002-10-31 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments
EP1749832A3 (en) * 1998-12-10 2008-03-26 Pfizer Products Incorporated Carbamate and carbazate ketolide antibiotics
EP1298138B1 (en) * 1998-12-10 2006-11-02 Pfizer Products Inc. Carbamate and Carbazate Ketolide Antibiotics
TR200102129T2 (tr) 1998-12-10 2002-01-21 Pfizer Products Inc. Karbamat ve karbazat ketolid antibiyotikleri.
FR2789392B1 (fr) * 1999-02-04 2001-10-05 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity
ID30547A (id) * 1999-04-16 2001-12-20 Kosan Biosciences Inc Zat anti-infeksi makrolida
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
IL145976A0 (en) 1999-04-16 2002-07-25 Ortho Mcneil Pharm Inc Ketolide antibacterials
EA200100983A1 (ru) * 1999-05-24 2002-10-31 Пфайзер Продактс Инк. Производные 13-метилэритромицина
WO2003004509A2 (en) * 2001-07-03 2003-01-16 Chiron Corporation C12 modified erythromycin macrolides and ketolides having antibacterial activity
KR101035043B1 (ko) 2002-07-01 2011-05-19 아르키온 라이프 사이언씨즈 엘엘씨 글루코사민 및 ｎ-아세틸글루코사민의 제조를 위한 물질및 공정
ES2552682T3 (es) 2003-03-10 2015-12-01 Merck Sharp & Dohme Corp. Agentes antibacterianos novedosos
US7163924B2 (en) * 2003-04-25 2007-01-16 Chiron Corporation Ketolide derivatives
US7332476B2 (en) * 2003-04-25 2008-02-19 Novartis Ag Pyridyl substituted ketolide antibiotics
CN105732745A (zh) 2007-10-25 2016-07-06 森普拉制药公司 大环内酯类抗菌剂的制备方法
AU2009308182B2 (en) * 2008-10-24 2016-05-19 Cempra Pharmaceuticals, Inc. Biodefenses using triazole-containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
US9480679B2 (en) 2009-09-10 2016-11-01 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and MAC diseases
DK2550286T3 (en) 2010-03-22 2016-02-29 Cempra Pharmaceuticals Inc CRYSTALLINE FORMS OF A MACROLID AND APPLICATIONS THEREOF
CN105198944B (zh) 2010-05-20 2018-06-01 森普拉制药公司 制备大环内酯和酮内酯及其中间体的方法
EP2613630A4 (en) 2010-09-10 2014-01-15 Cempra Pharmaceuticals Inc HYDROGEN BOND FOR THE PREPARATION OF FLUOROCHETOLIDES FOR THE TREATMENT OF DISEASES
MX2014011537A (es) 2012-03-27 2015-02-10 Cempra Pharmaceuticals Inc Formulaciones parenterales para la administracion de antibioticos macrolidos.
HK1217665A1 (zh) 2013-03-14 2017-01-20 森普拉制药公司 用於治療呼吸道疾病的方法及其製劑
RU2015138797A (ru) 2013-03-15 2017-04-24 Семпра Фармасьютикалс, Инк. Конвергентные способы получения макролидных антибактериальных агентов
US9982005B2 (en) 2013-04-04 2018-05-29 President And Fellows Of Harvard College Macrolides and methods of their preparation and use
US10633407B2 (en) 2014-10-08 2020-04-28 President And Fellows Of Harvard College 14-membered ketolides and methods of their preparation and use
JP2018509452A (ja) 2015-03-25 2018-04-05 プレジデント アンド フェローズ オブ ハーバード カレッジ 修飾デソサミン糖をもつマクロライドおよびその使用
MD1222Z (ro) * 2017-05-31 2018-08-31 ИНСТИТУТ ЭЛЕКТРОННОЙ ИНЖЕНЕРИИ И НАНОТЕХНОЛОГИЙ "D. Ghitu" АНМ Procedeu de tratare a materialului săditor al florilor înainte de plantare
JP7199722B2 (ja) 2019-12-25 2023-01-06 旭精工株式会社 硬貨搬送振分機構及びそれを備えた硬貨識別搬送装置

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AT342770B (de) * 1975-04-07 1978-04-25 Thomae Gmbh Dr K Verfahren zur herstellung neuer erythromycinderivate
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Also Published As

Publication number Publication date
HUT73772A (en) 1996-09-30
FI955913A7 (fi) 1995-12-08
CZ322395A3 (en) 1996-08-14
BG100150A (bg) 1996-06-28
CZ296005B6 (cs) 2005-12-14
HRP950217B1 (en) 2004-06-30
HU9503505D0 (en) 1996-02-28
SI0676409T1 (en) 2003-06-30
NZ284498A (en) 1997-07-27
DZ1869A1 (fr) 2002-02-17
LV11182A (lv) 1996-04-20
HU215396B (hu) 1998-12-28
AU2310795A (en) 1995-10-30
ATE234853T1 (de) 2003-04-15
AP587A (en) 1997-04-29
UA44705C2 (uk) 2002-03-15
SV1995000018A (es) 1997-10-24
WO1995027720A1 (fr) 1995-10-19
CA2164638C (fr) 2003-12-30
PL311871A1 (en) 1996-03-18
JP3000023B2 (ja) 2000-01-17
FR2718450A1 (fr) 1995-10-13
GB9506856D0 (en) 1995-05-24
EP0676409B1 (fr) 2003-03-19
JO1850B1 (en) 1995-12-27
MA23501A1 (fr) 1995-12-31
IS4309A (is) 1995-11-17
BR9506147A (pt) 1996-04-16
JPH07278177A (ja) 1995-10-24
LV11182B (en) 1997-04-20
FI955913A0 (fi) 1995-12-08
ES2189820T3 (es) 2003-07-16
YU49221B (sh) 2004-11-25
CA2164638A1 (fr) 1995-10-19
PL180837B1 (pl) 2001-04-30
BG61916B1 (bg) 1998-09-30
HRP950217A2 (en) 1997-08-31
US5760233A (en) 1998-06-02
RO115634B1 (ro) 2000-04-28
AU684939B2 (en) 1998-01-08
IL112954A0 (en) 1995-06-29
SK154695A3 (en) 1996-10-02
AP9500743A0 (en) 1995-07-31
GEP19991836B (en) 1999-11-05
NO954942L (no) 1996-02-07
CN1126997A (zh) 1996-07-17
MD663G2 (ro) 1997-07-31
SA97170757A (ar) 2005-12-03
YU21695A (sh) 1997-12-05
MD663F1 (ro) 1997-01-31
IS1865B (is) 2003-05-02
NO954942D0 (no) 1995-12-06
PT676409E (pt) 2003-08-29
OA10200A (fr) 1996-12-18
TW316908B (oth) 1997-10-01
MY114672A (en) 2002-12-31
CO4370097A1 (es) 1996-10-07
FR2718450B1 (fr) 1997-01-10
EE04498B1 (et) 2005-06-15
ZA952059B (en) 1996-03-13
RU2141965C1 (ru) 1999-11-27
NO308361B1 (no) 2000-09-04
EP0676409A1 (fr) 1995-10-11
US5656607A (en) 1997-08-12
EE9500080A (et) 1996-12-16
TNSN95026A1 (fr) 1996-02-06
KR100317148B1 (ko) 2002-06-22
SK284079B6 (sk) 2004-09-08
DE69529934D1 (de) 2003-04-24
DE69529934T2 (de) 2003-09-04
CN1059445C (zh) 2000-12-13
PE2896A1 (es) 1996-02-12
IL112954A (en) 2000-07-16
GB2288174A (en) 1995-10-11
FI111264B (fi) 2003-06-30

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