DE69332577T2 - Verfahren zur Herstellung von 13-Ether-Derivaten von Milbemycinen und Zwischenprodukte - Google Patents

Verfahren zur Herstellung von 13-Ether-Derivaten von Milbemycinen und Zwischenprodukte

Info

Publication number
DE69332577T2
DE69332577T2 DE69332577T DE69332577T DE69332577T2 DE 69332577 T2 DE69332577 T2 DE 69332577T2 DE 69332577 T DE69332577 T DE 69332577T DE 69332577 T DE69332577 T DE 69332577T DE 69332577 T2 DE69332577 T2 DE 69332577T2
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DE
Germany
Prior art keywords
groups
group
formula
defined above
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69332577T
Other languages
German (de)
English (en)
Other versions
DE69332577D1 (de
Inventor
Shunshi Kojima
Mitsugi Shibano
Mutsuo Suzuki
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mitsui Chemicals Agro Inc
Elanco Japan KK
Original Assignee
Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Sankyo Co Ltd filed Critical Sankyo Co Ltd
Application granted granted Critical
Publication of DE69332577D1 publication Critical patent/DE69332577D1/de
Publication of DE69332577T2 publication Critical patent/DE69332577T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
DE69332577T 1992-09-01 1993-09-01 Verfahren zur Herstellung von 13-Ether-Derivaten von Milbemycinen und Zwischenprodukte Expired - Fee Related DE69332577T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP23344492 1992-09-01
JP26366092 1992-10-01
JP32284792 1992-12-02

Publications (2)

Publication Number Publication Date
DE69332577D1 DE69332577D1 (de) 2003-01-30
DE69332577T2 true DE69332577T2 (de) 2003-11-20

Family

ID=27331997

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69332577T Expired - Fee Related DE69332577T2 (de) 1992-09-01 1993-09-01 Verfahren zur Herstellung von 13-Ether-Derivaten von Milbemycinen und Zwischenprodukte

Country Status (13)

Country Link
US (2) US5461168A (enExample)
EP (1) EP0594291B1 (enExample)
JP (1) JP2654337B2 (enExample)
KR (1) KR0161541B1 (enExample)
AT (1) ATE229960T1 (enExample)
AU (1) AU666750B2 (enExample)
CA (1) CA2105251C (enExample)
DE (1) DE69332577T2 (enExample)
DK (1) DK0594291T3 (enExample)
ES (1) ES2186672T3 (enExample)
NZ (1) NZ248559A (enExample)
PT (1) PT594291E (enExample)
TW (1) TW262474B (enExample)

Families Citing this family (165)

* Cited by examiner, † Cited by third party
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WO1999061447A1 (en) * 1998-05-25 1999-12-02 Sankyo Company, Limited Process for producing 13-ester derivatives of milbemycins
JP4499847B2 (ja) * 1998-05-25 2010-07-07 三井化学アグロ株式会社 ミルベマイシン類の１３−エステル誘導体の製造法
JP2002121195A (ja) * 2000-10-12 2002-04-23 Sankyo Co Ltd １３位置換ミルベマイシン誘導体の製造法
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TWI487486B (zh) 2009-12-01 2015-06-11 Syngenta Participations Ag 以異唑啉衍生物為主之殺蟲化合物
ES2543747T3 (es) 2010-02-17 2015-08-21 Syngenta Participations Ag Derivados de isoxazolina como insecticidas
AU2011217466B2 (en) 2010-02-22 2015-02-26 Syngenta Participations Ag Dihydrofuran derivatives as insecticidal compounds
EA201201179A1 (ru) 2010-02-25 2013-04-30 Зингента Партисипейшнс Аг Способ получения изоксазолиновых производных
BR112013008063A2 (pt) 2010-10-05 2016-06-14 Syngenta Participations Ag pirrolidin-il-aril-carboxamidas inseticidas
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CN103221395A (zh) 2010-11-23 2013-07-24 先正达参股股份有限公司 杀虫化合物
CN103261188A (zh) 2010-12-17 2013-08-21 先正达参股股份有限公司 杀虫化合物
AR085318A1 (es) 2011-02-09 2013-09-25 Syngenta Participations Ag Derivados de triazol que tienen actividad insecticida
US20140005235A1 (en) 2011-03-22 2014-01-02 Syngenta Participations Ag Insecticidal compounds
KR20140034798A (ko) 2011-05-18 2014-03-20 신젠타 파티서페이션즈 아게 아릴티오아세트아미드 유도체에 기반한 살곤충 화합물
US9339505B2 (en) 2011-05-31 2016-05-17 Syngenta Participations Ag Pesticidal mixtures including isoxazoline derivatives
TW201311677A (zh) 2011-05-31 2013-03-16 Syngenta Participations Ag 殺蟲化合物
WO2012175474A1 (en) 2011-06-20 2012-12-27 Syngenta Participations Ag 1,2,3 triazole pesticides
US20140343049A1 (en) 2011-08-22 2014-11-20 Syngenta Participations Ag Dihydrofuran derivatives as insecticidal compounds
CN103732567A (zh) 2011-08-22 2014-04-16 先正达参股股份有限公司 作为杀虫化合物的二氢呋喃衍生物
CN103764644A (zh) 2011-08-25 2014-04-30 先正达参股股份有限公司 作为杀虫化合物的异噁唑啉衍生物
WO2013026930A1 (en) 2011-08-25 2013-02-28 Syngenta Participations Ag Process for the preparation of thietane derivatives
WO2013026933A1 (en) 2011-08-25 2013-02-28 Syngenta Participations Ag Isoxazoline derivatives as insecticidal compounds
WO2013026929A1 (en) 2011-08-25 2013-02-28 Syngenta Participations Ag Dihydropyrrole derivatives as insecticidal compounds
WO2013026695A1 (en) 2011-08-25 2013-02-28 Syngenta Participations Ag Isoxazoline derivatives as insecticidal compounds
CN103842358A (zh) 2011-09-13 2014-06-04 先正达参股股份有限公司 作为杀虫化合物的异噻唑啉衍生物
WO2013050261A1 (en) 2011-10-03 2013-04-11 Syngenta Participations Ag Insecticidal 2-methoxybenzamide derivatives
JP2014534182A (ja) 2011-10-03 2014-12-18 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト 殺虫化合物としてのイソオキサゾリン誘導体
WO2013135674A1 (en) 2012-03-12 2013-09-19 Syngenta Participations Ag Insecticidal 2-aryl-acetamide compounds
WO2014001120A1 (en) 2012-06-25 2014-01-03 Syngenta Participations Ag Isothiazole derivatives as insecticidal compounds
WO2014001121A1 (en) 2012-06-25 2014-01-03 Syngenta Participations Ag Isothiazole derivatives as insecticidal compounds
CN104755457A (zh) 2012-10-31 2015-07-01 先正达参股股份有限公司 杀虫化合物
WO2014079935A1 (en) 2012-11-21 2014-05-30 Syngenta Participations Ag Insecticidal compounds based on arylthioacetamide derivatives
US9402395B2 (en) 2013-04-02 2016-08-02 Syngenta Participations Ag Insecticidal compounds
US9635853B2 (en) 2013-04-02 2017-05-02 Syngenta Participations Ag Insecticidal compounds
WO2015007451A1 (en) 2013-07-15 2015-01-22 Syngenta Participations Ag Microbiocidal heterobicyclic derivatives
EP3556744B1 (en) 2013-12-23 2022-06-01 Syngenta Participations AG Insecticidal compounds
FI3206486T3 (fi) 2014-10-14 2023-03-19 ICB Pharma Fysikaalisen vaikutustavan omaavia pestisidiformulaatioita
WO2016087593A1 (en) 2014-12-05 2016-06-09 Syngenta Participations Ag Novel fungicidal quinolinylamidines
ES2935981T3 (es) 2015-03-27 2023-03-13 Syngenta Participations Ag Intermedios para la preparación de derivados heterobicíclicos microbicidas
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US20180319753A1 (en) 2015-10-28 2018-11-08 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
BR112018008947A8 (pt) 2015-11-04 2019-02-26 Syngenta Participations Ag derivados de anilida microbiocidas
US10640497B2 (en) 2015-12-02 2020-05-05 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
CN108368099B (zh) 2015-12-17 2021-11-12 先正达参股股份有限公司 杀微生物的噁二唑衍生物
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WO2017162868A1 (en) 2016-03-24 2017-09-28 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
BR112018070568B1 (pt) 2016-04-08 2022-03-08 Syngenta Participations Ag Compostos derivados de oxadiazol microbiocidas, composição agroquímica, método de controle ou prevenção da infestação de plantas úteis por microrganismos fitopatogênicos e uso do referido composto
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AR108745A1 (es) 2016-06-21 2018-09-19 Syngenta Participations Ag Derivados de oxadiazol microbiocidas
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WO2019011926A1 (en) 2017-07-11 2019-01-17 Syngenta Participations Ag MICROBIOCIDE OXADIAZOLE DERIVATIVES
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WO2019011928A1 (en) 2017-07-11 2019-01-17 Syngenta Participations Ag MICROBIOCIDE OXADIAZOLE DERIVATIVES
BR112020000414A2 (pt) 2017-07-12 2020-07-21 Syngenta Participations Ag derivados de oxadiazol microbicidas
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US5461168A (en) 1995-10-24
AU4497993A (en) 1994-03-10
JPH06220068A (ja) 1994-08-09
CA2105251C (en) 2004-12-07
US5625078A (en) 1997-04-29
KR940007038A (ko) 1994-04-26
TW262474B (enExample) 1995-11-11
NZ248559A (en) 1995-05-26
EP0594291A1 (en) 1994-04-27
DK0594291T3 (da) 2003-01-27
ES2186672T3 (es) 2003-05-16
PT594291E (pt) 2003-03-31
CA2105251A1 (en) 1994-03-02
ATE229960T1 (de) 2003-01-15
DE69332577D1 (de) 2003-01-30
EP0594291B1 (en) 2002-12-18
JP2654337B2 (ja) 1997-09-17
HK1010371A1 (en) 1999-06-17
AU666750B2 (en) 1996-02-22

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