AR117200A1 - Derivados de tiazol microbiocidas - Google Patents

Derivados de tiazol microbiocidas

Info

Publication number
AR117200A1
AR117200A1 ARP190103446A ARP190103446A AR117200A1 AR 117200 A1 AR117200 A1 AR 117200A1 AR P190103446 A ARP190103446 A AR P190103446A AR P190103446 A ARP190103446 A AR P190103446A AR 117200 A1 AR117200 A1 AR 117200A1
Authority
AR
Argentina
Prior art keywords
alkyl
cycloalkyl
haloalkyl
alkoxy
sulfur
Prior art date
Application number
ARP190103446A
Other languages
English (en)
Inventor
Mathias Blum
Andrew Edmunds
Clemens Lamberth
Stefano Rendine
Mattia Riccardo Monaco
David Burns
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR117200A1 publication Critical patent/AR117200A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D411/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/12Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/781,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Abstract

Compuestos de fórmula (1) en donde los sustituyentes son como se definen en la reivindicación 1, útiles como pesticidas y especialmente fungicidas. Reivindicación 1: Un compuesto de fórmula (1), donde, Y es C-F, C-H o N; R¹ es hidrógeno, halógeno, ciano, alquilo C₁₋₄, alcoxi C₁₋₄, haloalquilo C₁₋₄ o HC(O)NH-; R² es alquilo C₁₋₈, haloalquilo C₁₋₈, alcoxi C₁₋₈, cicloalquilo C₃₋₈, cicloalquil C₃₋₈-alquilo C₁₋₂, en donde los grupos cicloalquilo están opcionalmente sustituidos con 1 a 3 grupos representados por R³, fenilo, feniloalquilo C₁₋₂, en donde los anillos de fenilo están opcionalmente sustituidos con 1 a 3 grupos representados por R³, heteroarilo, heteroarilalquilo C₁₋₂, en donde el heteroarilo es un anillo monocíclico aromático de 5 ó 6 miembros que comprende 1, 2, 3 ó 4 heteroátomos seleccionados de manera individual de nitrógeno, oxígeno y azufre, heterociclilo, heterociclilalquilo C₁₋₂, en donde el heterociclilo es un anillo monocíclico no aromático de 4, 5 ó 6 miembros que comprende 1, 2 ó 3 heteroátomos seleccionados de manera individual de nitrógeno, oxígeno y azufre, o un sistema anular carbobiciclilo o carbotriciclilo anulado o espirocíclico no aromático de 5 a 12 miembros que comprende opcionalmente 1, 2, 3, 4 ó 5 heteroátomos seleccionados de manera individual de nitrógeno, oxígeno y azufre, y unidos opcionalmente al resto de la molécula a través de un conector alquileno C₁₋₂; R³ es halógeno, alquilo C₁₋₄, alcoxi C₁₋₄, haloalquilo C₁₋₄, cicloalquilo C₃₋₈ o cicloalquil C₃₋₈-alquilo C₁₋₂; X es N o C-H; o una sal o un N-óxido del mismo.
ARP190103446A 2018-11-30 2019-11-25 Derivados de tiazol microbiocidas AR117200A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP18209591 2018-11-30

Publications (1)

Publication Number Publication Date
AR117200A1 true AR117200A1 (es) 2021-07-21

Family

ID=64564711

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP190103446A AR117200A1 (es) 2018-11-30 2019-11-25 Derivados de tiazol microbiocidas

Country Status (27)

Country Link
US (1) US20220017501A1 (es)
EP (1) EP3887360B1 (es)
JP (1) JP2022509694A (es)
KR (1) KR20210098979A (es)
CN (1) CN113166082A (es)
AR (1) AR117200A1 (es)
AU (1) AU2019389778B2 (es)
BR (1) BR112021010367A2 (es)
CA (1) CA3120029A1 (es)
CL (1) CL2021001349A1 (es)
CO (1) CO2021007062A2 (es)
CR (1) CR20210282A (es)
DK (1) DK3887360T3 (es)
EA (1) EA202191456A1 (es)
ES (1) ES2941648T3 (es)
FI (1) FI3887360T3 (es)
GE (1) GEP20227439B (es)
HR (1) HRP20230310T1 (es)
HU (1) HUE061398T2 (es)
IL (1) IL283486A (es)
MX (1) MX2021006099A (es)
PL (1) PL3887360T3 (es)
PT (1) PT3887360T (es)
TW (1) TWI810412B (es)
UA (1) UA127364C2 (es)
UY (1) UY38492A (es)
WO (1) WO2020109509A1 (es)

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JP7044375B2 (ja) 2016-05-31 2022-03-30 ボード オブ リージェンツ,ザ ユニバーシティ オブ テキサス システム Ptpn11の複素環式阻害剤
MX2020011528A (es) 2018-05-02 2021-02-09 Navire Pharma Inc Inhibidores heterociclicos sustituidos de ptpn11.
WO2020033828A1 (en) 2018-08-10 2020-02-13 Board Of Regents, The University Of Texas System 6-(4-amino-3-methyl-2-oxa-8-azaspiro[4.5]decan-8-yl)-3-(2,3-dichlorophenyl)-2-methylpyrimidin-4(3h)-one derivatives and related compounds as ptpn11 (shp2) inhibitors for treating cancer
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AR127799A1 (es) 2021-12-02 2024-02-28 Syngenta Crop Protection Ag Composiciones fungicidas
WO2024068656A1 (en) 2022-09-28 2024-04-04 Syngenta Crop Protection Ag Fungicidal compositions
WO2024068655A1 (en) 2022-09-28 2024-04-04 Syngenta Crop Protection Ag Fungicidal compositions

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Also Published As

Publication number Publication date
TW202031130A (zh) 2020-09-01
JP2022509694A (ja) 2022-01-21
PT3887360T (pt) 2023-04-03
CL2021001349A1 (es) 2021-11-12
FI3887360T3 (fi) 2023-04-04
US20220017501A1 (en) 2022-01-20
ES2941648T3 (es) 2023-05-24
WO2020109509A1 (en) 2020-06-04
HUE061398T2 (hu) 2023-06-28
TWI810412B (zh) 2023-08-01
HRP20230310T1 (hr) 2023-05-12
AU2019389778B2 (en) 2024-03-14
EP3887360B1 (en) 2023-01-18
GEP20227439B (en) 2022-11-25
CN113166082A (zh) 2021-07-23
IL283486A (en) 2021-07-29
BR112021010367A2 (pt) 2021-08-24
DK3887360T3 (da) 2023-04-03
EA202191456A1 (ru) 2021-10-14
UY38492A (es) 2020-06-30
AU2019389778A1 (en) 2021-06-03
CA3120029A1 (en) 2020-06-04
CO2021007062A2 (es) 2021-06-10
PL3887360T3 (pl) 2023-05-08
EP3887360A1 (en) 2021-10-06
MX2021006099A (es) 2021-07-07
CR20210282A (es) 2021-06-30
UA127364C2 (uk) 2023-07-26
KR20210098979A (ko) 2021-08-11

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