AU666750B2 - Novel processes for the production of 13-ether derivatives of milbemycins, and novel intermediates therefor - Google Patents

Novel processes for the production of 13-ether derivatives of milbemycins, and novel intermediates therefor Download PDF

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Publication number
AU666750B2
AU666750B2 AU44979/93A AU4497993A AU666750B2 AU 666750 B2 AU666750 B2 AU 666750B2 AU 44979/93 A AU44979/93 A AU 44979/93A AU 4497993 A AU4497993 A AU 4497993A AU 666750 B2 AU666750 B2 AU 666750B2
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formula
compound
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Ceased
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AU44979/93A
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AU4497993A (en
Inventor
Shunshi Kojima
Mitsugi Shibano
Mutsuo Suzuki
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Sankyo Co Ltd
Elanco Japan KK
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Sankyo Co Ltd
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Assigned to SANKYO COMPANY LIMITED, SANKYO LIFETECH COMPANY LIMITED reassignment SANKYO COMPANY LIMITED Alteration of Name(s) in Register under S187 Assignors: SANKYO COMPANY LIMITED
Assigned to NOVARTIS ANIMAL HEALTH K.K., SANKYO COMPANY LIMITED reassignment NOVARTIS ANIMAL HEALTH K.K. Alteration of Name(s) in Register under S187 Assignors: SANKYO COMPANY LIMITED, SANKYO LIFETECH COMPANY LIMITED
Anticipated expiration legal-status Critical
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU44979/93A 1992-09-01 1993-08-31 Novel processes for the production of 13-ether derivatives of milbemycins, and novel intermediates therefor Ceased AU666750B2 (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
JP4-233444 1992-09-01
JP23344492 1992-09-01
JP4-263660 1992-10-01
JP26366092 1992-10-01
JP4-322847 1992-12-02
JP32284792 1992-12-02

Publications (2)

Publication Number Publication Date
AU4497993A AU4497993A (en) 1994-03-10
AU666750B2 true AU666750B2 (en) 1996-02-22

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ID=27331997

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Application Number Title Priority Date Filing Date
AU44979/93A Ceased AU666750B2 (en) 1992-09-01 1993-08-31 Novel processes for the production of 13-ether derivatives of milbemycins, and novel intermediates therefor

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US (2) US5461168A (enExample)
EP (1) EP0594291B1 (enExample)
JP (1) JP2654337B2 (enExample)
KR (1) KR0161541B1 (enExample)
AT (1) ATE229960T1 (enExample)
AU (1) AU666750B2 (enExample)
CA (1) CA2105251C (enExample)
DE (1) DE69332577T2 (enExample)
DK (1) DK0594291T3 (enExample)
ES (1) ES2186672T3 (enExample)
NZ (1) NZ248559A (enExample)
PT (1) PT594291E (enExample)
TW (1) TW262474B (enExample)

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JP4499847B2 (ja) * 1998-05-25 2010-07-07 三井化学アグロ株式会社 ミルベマイシン類の１３−エステル誘導体の製造法
KR100612634B1 (ko) * 1998-05-25 2006-08-14 상꾜 아그로 가부시키가이샤 밀베마이신류의 13-에스테르 유도체의 제조법
JP2002121195A (ja) * 2000-10-12 2002-04-23 Sankyo Co Ltd １３位置換ミルベマイシン誘導体の製造法
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US7919522B2 (en) 2007-05-03 2011-04-05 Merial Limited Compositions comprising C-13 alkoxyether macrolide compounds and phenylpyrazole compounds
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US5461168A (en) 1995-10-24
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DE69332577T2 (de) 2003-11-20
EP0594291B1 (en) 2002-12-18
KR940007038A (ko) 1994-04-26
TW262474B (enExample) 1995-11-11
PT594291E (pt) 2003-03-31
CA2105251A1 (en) 1994-03-02
ES2186672T3 (es) 2003-05-16
NZ248559A (en) 1995-05-26
JPH06220068A (ja) 1994-08-09
AU4497993A (en) 1994-03-10
US5625078A (en) 1997-04-29
EP0594291A1 (en) 1994-04-27
ATE229960T1 (de) 2003-01-15
HK1010371A1 (en) 1999-06-17
CA2105251C (en) 2004-12-07
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DE69332577D1 (de) 2003-01-30

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