DE102007054497B3 - Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung - Google Patents

Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung Download PDF

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Publication number
DE102007054497B3
DE102007054497B3 DE102007054497A DE102007054497A DE102007054497B3 DE 102007054497 B3 DE102007054497 B3 DE 102007054497B3 DE 102007054497 A DE102007054497 A DE 102007054497A DE 102007054497 A DE102007054497 A DE 102007054497A DE 102007054497 B3 DE102007054497 B3 DE 102007054497B3
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DE
Germany
Prior art keywords
formula
crystalline
crystalline hydrate
theta
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE102007054497A
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German (de)
English (en)
Inventor
Theodor Andreas Dr. Wollmann
Regina Duffy
Frank Dr. Cullmann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis Deutschland GmbH
Original Assignee
Sanofi Aventis Deutschland GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40386121&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE102007054497(B3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis Deutschland GmbH filed Critical Sanofi Aventis Deutschland GmbH
Priority to DE102007063671A priority Critical patent/DE102007063671A1/de
Priority to DE102007054497A priority patent/DE102007054497B3/de
Priority to PCT/EP2008/009323 priority patent/WO2009062619A1/de
Priority to EP08850642A priority patent/EP2220040B1/de
Priority to JP2010533467A priority patent/JP5401463B2/ja
Priority to TW097143436A priority patent/TW200936566A/zh
Priority to CL2008003358A priority patent/CL2008003358A1/es
Priority to PE2008001909A priority patent/PE20091165A1/es
Priority to PA20088803701A priority patent/PA8803701A1/es
Priority to US12/269,802 priority patent/US8003636B2/en
Priority to ARP080104951A priority patent/AR069305A1/es
Priority to UY31469A priority patent/UY31469A1/es
Publication of DE102007054497B3 publication Critical patent/DE102007054497B3/de
Application granted granted Critical
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE102007054497A 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung Expired - Fee Related DE102007054497B3 (de)

Priority Applications (12)

Application Number Priority Date Filing Date Title
DE102007063671A DE102007063671A1 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
DE102007054497A DE102007054497B3 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung
PCT/EP2008/009323 WO2009062619A1 (de) 2007-11-13 2008-11-06 Neue kristalline diphenylazetidinonhydrate, diese verbindungen enthaltende arzneimittel und deren verwendung
EP08850642A EP2220040B1 (de) 2007-11-13 2008-11-06 Neue kristalline diphenylazetidinonhydrate, diese verbindungen enthaltende arzneimittel und deren verwendung
JP2010533467A JP5401463B2 (ja) 2007-11-13 2008-11-06 新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用
CL2008003358A CL2008003358A1 (es) 2007-11-13 2008-11-11 Hidratos cristalinos de n-(4((2s,3r)-3-((s)-3-(4-fluorofenil)-3-hidroxipropil)-2-(4-metoxifenil)4-oxoazetidin-1-il)bencil)-n-((2s,3r,4r,5r)-2,3,4,5,6-pentahidroxihexil)dodecandiamida; procedimiento de preparacion de dicho compuesto; composiicon farmaceutica que lo comprende; y uso para tratar trastornos del metabolismo de lipidos.
TW097143436A TW200936566A (en) 2007-11-13 2008-11-11 Novel crystalline diphenylazetidinone hydrates, medicaments comprising these compounds and use thereof
PE2008001909A PE20091165A1 (es) 2007-11-13 2008-11-11 Hidratos de difenilazetidinona cristalinos y composiciones que comprenden a estos compuestos
PA20088803701A PA8803701A1 (es) 2007-11-13 2008-11-12 Nuevos hidratos de difenilazetidinona cristalinos, medicamentos que comprenden a estos compuestos y uso de los mismos
US12/269,802 US8003636B2 (en) 2007-11-13 2008-11-12 Certain crystalline diphenylazetidinone hydrates, pharmaceutical compositions thereof and methods for their use
ARP080104951A AR069305A1 (es) 2007-11-13 2008-11-13 Nuevos hidratos de difenilazetidinona cristalinos, medicamento que comprenden a estos compuestos y uso de los mismos
UY31469A UY31469A1 (es) 2007-11-13 2008-11-13 Nuevos hidratos de difenilazetidinona cristalinos, medicamentos que comprenden a estos compuestos y uso de los mismos

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007063671A DE102007063671A1 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
DE102007054497A DE102007054497B3 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung

Publications (1)

Publication Number Publication Date
DE102007054497B3 true DE102007054497B3 (de) 2009-07-23

Family

ID=40386121

Family Applications (2)

Application Number Title Priority Date Filing Date
DE102007054497A Expired - Fee Related DE102007054497B3 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung
DE102007063671A Withdrawn DE102007063671A1 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate, diese Verbindungen enthaltende Arzneimittel und deren Verwendung

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE102007063671A Withdrawn DE102007063671A1 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate, diese Verbindungen enthaltende Arzneimittel und deren Verwendung

Country Status (11)

Country Link
US (1) US8003636B2 (enExample)
EP (1) EP2220040B1 (enExample)
JP (1) JP5401463B2 (enExample)
AR (1) AR069305A1 (enExample)
CL (1) CL2008003358A1 (enExample)
DE (2) DE102007054497B3 (enExample)
PA (1) PA8803701A1 (enExample)
PE (1) PE20091165A1 (enExample)
TW (1) TW200936566A (enExample)
UY (1) UY31469A1 (enExample)
WO (1) WO2009062619A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
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US8486926B2 (en) * 2006-11-17 2013-07-16 Harbor Therapeutics, Inc. Steroid tetrol solid state forms
US20080319221A1 (en) * 2007-06-22 2008-12-25 Bernd Junker Esters of Pentahydroxyhexylcarbamoyl Alkanoic Acids
CN101939009B (zh) * 2008-02-05 2013-07-17 哈博生物科学公司 药学固体形式
DK2273994T3 (en) 2008-04-03 2016-02-01 Neurmedix Inc PHARMACEUTICAL FORMS OF A MEDICINE
AU2013362400B2 (en) * 2012-12-22 2016-07-28 Novo Nordisk A/S Crystal form of compound used as mineralocorticoid receptor antagonist and preparation method therefor
US10080759B2 (en) 2014-01-22 2018-09-25 Duke University Methods of treating pruritus
WO2015112588A1 (en) 2014-01-22 2015-07-30 Biomimetix Jv, Llc Methods of treating skin disorders

Citations (1)

* Cited by examiner, † Cited by third party
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AR069305A1 (es) 2010-01-13
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