PE20091165A1 - Hidratos de difenilazetidinona cristalinos y composiciones que comprenden a estos compuestos - Google Patents

Hidratos de difenilazetidinona cristalinos y composiciones que comprenden a estos compuestos

Info

Publication number
PE20091165A1
PE20091165A1 PE2008001909A PE2008001909A PE20091165A1 PE 20091165 A1 PE20091165 A1 PE 20091165A1 PE 2008001909 A PE2008001909 A PE 2008001909A PE 2008001909 A PE2008001909 A PE 2008001909A PE 20091165 A1 PE20091165 A1 PE 20091165A1
Authority
PE
Peru
Prior art keywords
formula
crystalline
diphenylazethydinone
hydrates
compounds
Prior art date
Application number
PE2008001909A
Other languages
English (en)
Inventor
Theodor Andreas Wollmann
Regina Duffy
Frank Cullmann
Original Assignee
Sanofi Aventis Deutschland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40386121&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20091165(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis Deutschland filed Critical Sanofi Aventis Deutschland
Publication of PE20091165A1 publication Critical patent/PE20091165A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics

Abstract

REFERIDA A UN HIDRATO DE DIFENILAZETIDINONA CRISTALINO DE FORMULA (I), DONDE n TIENE UN VALOR DE 0,5 A 1,8. DICHO HIDRATO CRISTALINO TIENE UN PICO PRINCIPAL DE 20,83 GRADOS 2 TETA ± 0,2 GRADOS 2 TETA EN EL XRPD MEDIDO CON RADIACION CuKALFA. TAMBIEN ESTA REFERIDA A UN PROCEDIMIENTO DE PREPARACION QUE COMPRENDE DISOLVER EL COMPUESTO AMORFO DE FORMULA (II) EN UN DISOLVENTE ORGANICO TAL COMO ETANOL O UNA MEZCLA DE ETANOL/AGUA, Y ANADIR ESTA SOLUCION A UNA SUSPENSION DE CRISTALES DE SIEMBRA DEL COMPUESTO DE FORMULA (I)
PE2008001909A 2007-11-13 2008-11-11 Hidratos de difenilazetidinona cristalinos y composiciones que comprenden a estos compuestos PE20091165A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102007054497A DE102007054497B3 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung

Publications (1)

Publication Number Publication Date
PE20091165A1 true PE20091165A1 (es) 2009-08-31

Family

ID=40386121

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2008001909A PE20091165A1 (es) 2007-11-13 2008-11-11 Hidratos de difenilazetidinona cristalinos y composiciones que comprenden a estos compuestos

Country Status (11)

Country Link
US (1) US8003636B2 (es)
EP (1) EP2220040B1 (es)
JP (1) JP5401463B2 (es)
AR (1) AR069305A1 (es)
CL (1) CL2008003358A1 (es)
DE (2) DE102007054497B3 (es)
PA (1) PA8803701A1 (es)
PE (1) PE20091165A1 (es)
TW (1) TW200936566A (es)
UY (1) UY31469A1 (es)
WO (1) WO2009062619A1 (es)

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JP2011511011A (ja) * 2008-02-05 2011-04-07 ハーバー バイオサイエンシーズ，インコーポレイテッド 医薬的固体状態形態
PT2273994E (pt) 2008-04-03 2016-03-15 Neurmedix Inc Formas de estado sólido de um produto farmacêutico
BR112015014839B1 (pt) * 2012-12-22 2022-09-06 Kbp Biosciences Co., Ltd Forma cristalina do composto utilizado como antagonista do receptor de mineralocorticoide, seus usos, seu processo de preparação e composição farmacêutica
US10064871B2 (en) 2014-01-22 2018-09-04 Biomimetix Jv, Llc Methods of treating skin disorders
US10080759B2 (en) 2014-01-22 2018-09-25 Duke University Methods of treating pruritus

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UY31469A1 (es) 2009-07-17
US8003636B2 (en) 2011-08-23
EP2220040A1 (de) 2010-08-25
TW200936566A (en) 2009-09-01
PA8803701A1 (es) 2009-06-23
EP2220040B1 (de) 2013-01-16
JP2011503127A (ja) 2011-01-27
CL2008003358A1 (es) 2009-06-26
AR069305A1 (es) 2010-01-13
DE102007054497B3 (de) 2009-07-23
JP5401463B2 (ja) 2014-01-29
DE102007063671A1 (de) 2009-06-25
US20090203578A1 (en) 2009-08-13

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