JP5401463B2 - 新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用 - Google Patents

新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用 Download PDF

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JP5401463B2
JP5401463B2 JP2010533467A JP2010533467A JP5401463B2 JP 5401463 B2 JP5401463 B2 JP 5401463B2 JP 2010533467 A JP2010533467 A JP 2010533467A JP 2010533467 A JP2010533467 A JP 2010533467A JP 5401463 B2 JP5401463 B2 JP 5401463B2
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formula
compound
administered
combination
crystalline hydrate
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JP2011503127A5 (enExample
JP2011503127A (ja
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テーオドール・アンドレーアス・ヴォルマン
レジーナ・デューフィー
フランク・クルマン
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サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2010533467A 2007-11-13 2008-11-06 新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用 Expired - Fee Related JP5401463B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DE102007054497A DE102007054497B3 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung
DE102007054497.0 2007-11-13
US99025507P 2007-11-26 2007-11-26
US60/990,255 2007-11-26
PCT/EP2008/009323 WO2009062619A1 (de) 2007-11-13 2008-11-06 Neue kristalline diphenylazetidinonhydrate, diese verbindungen enthaltende arzneimittel und deren verwendung

Publications (3)

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JP2011503127A JP2011503127A (ja) 2011-01-27
JP2011503127A5 JP2011503127A5 (enExample) 2011-12-22
JP5401463B2 true JP5401463B2 (ja) 2014-01-29

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JP2010533467A Expired - Fee Related JP5401463B2 (ja) 2007-11-13 2008-11-06 新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用

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US (1) US8003636B2 (enExample)
EP (1) EP2220040B1 (enExample)
JP (1) JP5401463B2 (enExample)
AR (1) AR069305A1 (enExample)
CL (1) CL2008003358A1 (enExample)
DE (2) DE102007054497B3 (enExample)
PA (1) PA8803701A1 (enExample)
PE (1) PE20091165A1 (enExample)
TW (1) TW200936566A (enExample)
UY (1) UY31469A1 (enExample)
WO (1) WO2009062619A1 (enExample)

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CN101939009B (zh) * 2008-02-05 2013-07-17 哈博生物科学公司 药学固体形式
DK2273994T3 (en) 2008-04-03 2016-02-01 Neurmedix Inc PHARMACEUTICAL FORMS OF A MEDICINE
AU2013362400B2 (en) * 2012-12-22 2016-07-28 Novo Nordisk A/S Crystal form of compound used as mineralocorticoid receptor antagonist and preparation method therefor
US10080759B2 (en) 2014-01-22 2018-09-25 Duke University Methods of treating pruritus
WO2015112588A1 (en) 2014-01-22 2015-07-30 Biomimetix Jv, Llc Methods of treating skin disorders

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US8003636B2 (en) 2011-08-23
JP2011503127A (ja) 2011-01-27
PE20091165A1 (es) 2009-08-31
AR069305A1 (es) 2010-01-13
DE102007063671A1 (de) 2009-06-25
EP2220040A1 (de) 2010-08-25
TW200936566A (en) 2009-09-01
WO2009062619A1 (de) 2009-05-22
PA8803701A1 (es) 2009-06-23
UY31469A1 (es) 2009-07-17
CL2008003358A1 (es) 2009-06-26
EP2220040B1 (de) 2013-01-16
US20090203578A1 (en) 2009-08-13

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