DK1204654T3 - Benzofurylpiperaziner og benzofurylhomopiperaziner: Serotonin agonister - Google Patents

Benzofurylpiperaziner og benzofurylhomopiperaziner: Serotonin agonister

Info

Publication number
DK1204654T3
DK1204654T3 DK00948745T DK00948745T DK1204654T3 DK 1204654 T3 DK1204654 T3 DK 1204654T3 DK 00948745 T DK00948745 T DK 00948745T DK 00948745 T DK00948745 T DK 00948745T DK 1204654 T3 DK1204654 T3 DK 1204654T3
Authority
DK
Denmark
Prior art keywords
sup
benzofurylpiperazines
benzofurylhomopiperazines
serotonin agonists
formula
Prior art date
Application number
DK00948745T
Other languages
English (en)
Inventor
Karin Briner
Joseph Paul Burkhart
Timothy Paul Burkholder
Brian Eugene Cunningham
Matthew Joseph Fisher
William Harlan Gritton
Shawn Christopher Miller
Jeffrey Thomas Mullaney
Matthew Robert Reinhard
Dennis Charles Thompson
Leonard Larry Junio Winneroski
Yanping Xu
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of DK1204654T3 publication Critical patent/DK1204654T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
DK00948745T 1999-07-29 2000-07-21 Benzofurylpiperaziner og benzofurylhomopiperaziner: Serotonin agonister DK1204654T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14627099P 1999-07-29 1999-07-29
PCT/US2000/019543 WO2001009111A1 (en) 1999-07-29 2000-07-21 Benzofurylpiperazines and benzofurylhomopiperazines: serotonin agonists

Publications (1)

Publication Number Publication Date
DK1204654T3 true DK1204654T3 (da) 2003-11-17

Family

ID=22516599

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00948745T DK1204654T3 (da) 1999-07-29 2000-07-21 Benzofurylpiperaziner og benzofurylhomopiperaziner: Serotonin agonister

Country Status (14)

Country Link
US (1) US6967201B1 (da)
EP (1) EP1204654B1 (da)
JP (1) JP2003506365A (da)
CN (1) CN1365359A (da)
AT (1) ATE245636T1 (da)
AU (1) AU768310B2 (da)
BR (1) BR0012752A (da)
CA (1) CA2378878A1 (da)
DE (1) DE60004066T2 (da)
DK (1) DK1204654T3 (da)
ES (1) ES2203498T3 (da)
MX (1) MXPA02000973A (da)
PT (1) PT1204654E (da)
WO (1) WO2001009111A1 (da)

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Also Published As

Publication number Publication date
CA2378878A1 (en) 2001-02-08
AU6220200A (en) 2001-02-19
MXPA02000973A (es) 2002-07-30
EP1204654B1 (en) 2003-07-23
EP1204654A1 (en) 2002-05-15
CN1365359A (zh) 2002-08-21
US6967201B1 (en) 2005-11-22
ATE245636T1 (de) 2003-08-15
WO2001009111A1 (en) 2001-02-08
AU768310B2 (en) 2003-12-04
DE60004066T2 (de) 2004-04-15
DE60004066D1 (de) 2003-08-28
PT1204654E (pt) 2003-11-28
ES2203498T3 (es) 2004-04-16
JP2003506365A (ja) 2003-02-18
BR0012752A (pt) 2002-04-02

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