PT1204659E - Benzofuranos serotoninergicos - Google Patents

Benzofuranos serotoninergicos

Info

Publication number
PT1204659E
PT1204659E PT00955245T PT00955245T PT1204659E PT 1204659 E PT1204659 E PT 1204659E PT 00955245 T PT00955245 T PT 00955245T PT 00955245 T PT00955245 T PT 00955245T PT 1204659 E PT1204659 E PT 1204659E
Authority
PT
Portugal
Prior art keywords
benzofuranos
serotoninergic
benzofurans
serotonergic
formula
Prior art date
Application number
PT00955245T
Other languages
English (en)
Inventor
Joseph Paul Burkhart
Yao-Chang Xu
Karin Briner
Timothy Paul Burkholder
Matthew Joseph Fisher
William Harlan Gritton
Shawn Christopher Miller
Jeffrey Thomas Mullaney
Leonard Larry Junio Winneroski
Yanping Xu
Brian Eugene Cunningham
Cynthia Darshini Jesudason
Matthew Robert Reinhard
Roger Ryan Rothhaar
Freddie Craig Stevens
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT1204659E publication Critical patent/PT1204659E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polyethers (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Polyurethanes Or Polyureas (AREA)
  • Dental Preparations (AREA)
  • Furan Compounds (AREA)
PT00955245T 1999-07-29 2000-07-21 Benzofuranos serotoninergicos PT1204659E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14618199P 1999-07-29 1999-07-29
US17260199P 1999-12-20 1999-12-20

Publications (1)

Publication Number Publication Date
PT1204659E true PT1204659E (pt) 2004-04-30

Family

ID=26843646

Family Applications (1)

Application Number Title Priority Date Filing Date
PT00955245T PT1204659E (pt) 1999-07-29 2000-07-21 Benzofuranos serotoninergicos

Country Status (13)

Country Link
EP (1) EP1204659B1 (pt)
JP (1) JP2003506369A (pt)
CN (1) CN1407982A (pt)
AT (1) ATE255105T1 (pt)
AU (1) AU768339B2 (pt)
BR (1) BR0012751A (pt)
CA (1) CA2380608A1 (pt)
DE (1) DE60006825T2 (pt)
DK (1) DK1204659T3 (pt)
ES (1) ES2209951T3 (pt)
MX (1) MXPA02000914A (pt)
PT (1) PT1204659E (pt)
WO (1) WO2001009122A2 (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0004245D0 (sv) 2000-11-20 2000-11-20 Pharmacia Ab Novel compounds and their use
PL360982A1 (en) 2000-11-20 2004-09-20 Biovitrum Ab Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor
CA2485537A1 (en) 2002-06-19 2003-12-31 Biovitrum Ab Novel compounds, their use and preparation
JP5173190B2 (ja) 2004-08-25 2013-03-27 武田薬品工業株式会社 腹圧性尿失禁の予防・治療剤及びそのスクリーニング方法
EP2018863B9 (en) 2006-05-16 2015-02-18 Takeda Pharmaceutical Company Limited Fused heterocyclic compound and use thereof
US20100266504A1 (en) 2007-11-15 2010-10-21 Takahiro Matsumoto Condensed pyridine derivative and use thereof
EP2510949A4 (en) 2009-12-11 2013-11-13 Astellas Pharma Inc THERAPEUTICS FOR FIBROMYALGIA
CN103601669B (zh) * 2013-05-20 2016-08-03 甘肃科瑞生物科技有限公司 一种1-叔丁氧羰基-2-甲基-4-哌啶酮的合成方法
WO2015066344A1 (en) 2013-11-01 2015-05-07 Arena Pharmaceuticals, Inc. 5-ht2c receptor agonists and compositions and methods of use
KR102037494B1 (ko) 2017-12-11 2019-10-28 씨제이헬스케어 주식회사 광학활성을 갖는 피페리딘 유도체의 중간체 및 이의 제조방법
US20210052600A1 (en) 2017-12-27 2021-02-25 Takeda Pharmaceutical Company Limited Therapeutic agents for stress urinary incontinence and incotinence of feces
CN110317129A (zh) * 2019-05-30 2019-10-11 杭州迈世腾药物科技有限公司 2-溴-5-甲氧基苯酚的合成方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0006524A1 (de) * 1978-06-22 1980-01-09 Ciba-Geigy Ag Neue Tetrahydropyridin- und Piperidinderivate und deren Säureadditionssalze, Verfahren zu deren Herstellung und solche enthaltende pharmazeutische Zusammensetzungen
DE3586794T2 (de) * 1984-12-21 1993-05-27 Duphar Int Res Arzneimittel mit psychotroper wirkung.
EP0398413A1 (en) * 1989-05-16 1990-11-22 Duphar International Research B.V "3,4-dehydropiperidine derivatives having psychotropic activity
JP2883995B2 (ja) * 1990-03-14 1999-04-19 第一製薬株式会社 ピペリジン誘導体及びその製造中間体
CA2335310A1 (en) * 1998-06-30 2000-01-06 Kenneth Lee Hauser Azepine derivatives having effects on serotonin related systems
ATE225345T1 (de) * 1998-06-30 2002-10-15 Lilly Co Eli Auf serotonin-verwandte systeme wirkende piperidin-derivate
JP2002519321A (ja) * 1998-06-30 2002-07-02 イーライ・リリー・アンド・カンパニー セロトニン関連系に効果を有するピロリジン、及び、ピロリン誘導体

Also Published As

Publication number Publication date
BR0012751A (pt) 2002-06-04
MXPA02000914A (es) 2002-07-30
ATE255105T1 (de) 2003-12-15
DE60006825T2 (de) 2004-08-12
AU6747400A (en) 2001-02-19
EP1204659B1 (en) 2003-11-26
JP2003506369A (ja) 2003-02-18
ES2209951T3 (es) 2004-07-01
WO2001009122A2 (en) 2001-02-08
EP1204659A2 (en) 2002-05-15
CN1407982A (zh) 2003-04-02
DE60006825D1 (de) 2004-01-08
CA2380608A1 (en) 2001-02-08
AU768339B2 (en) 2003-12-11
WO2001009122A3 (en) 2001-06-28
DK1204659T3 (da) 2004-04-05

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