ATE280169T1 - Serotonerge benzothiophene - Google Patents

Serotonerge benzothiophene

Info

Publication number
ATE280169T1
ATE280169T1 AT00950264T AT00950264T ATE280169T1 AT E280169 T1 ATE280169 T1 AT E280169T1 AT 00950264 T AT00950264 T AT 00950264T AT 00950264 T AT00950264 T AT 00950264T AT E280169 T1 ATE280169 T1 AT E280169T1
Authority
AT
Austria
Prior art keywords
benzothiophenes
serotonergic
formula
provides
present
Prior art date
Application number
AT00950264T
Other languages
English (en)
Inventor
Karin Briner
Timothy Paul Burkholder
Richard Gerard Conway
Brian Eugene Cunningham
Don Richard Finley
Lawrence Joseph Heinz
Cynthia Darshini Jesudason
Daniel Timothy Kohlman
Sidney Xi Liang
Yao-Chang Xu
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of ATE280169T1 publication Critical patent/ATE280169T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
AT00950264T 1999-07-29 2000-07-21 Serotonerge benzothiophene ATE280169T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14618599P 1999-07-29 1999-07-29
US17278499P 1999-12-20 1999-12-20
PCT/US2000/017864 WO2001009126A1 (en) 1999-07-29 2000-07-21 Serotonergic benzothiophenes

Publications (1)

Publication Number Publication Date
ATE280169T1 true ATE280169T1 (de) 2004-11-15

Family

ID=26843654

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00950264T ATE280169T1 (de) 1999-07-29 2000-07-21 Serotonerge benzothiophene

Country Status (8)

Country Link
EP (1) EP1204660B1 (de)
JP (1) JP2003506371A (de)
AT (1) ATE280169T1 (de)
AU (1) AU6339000A (de)
CA (1) CA2378879A1 (de)
DE (1) DE60015146T2 (de)
ES (1) ES2231229T3 (de)
WO (1) WO2001009126A1 (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001046147A1 (en) * 1999-12-20 2001-06-28 Eli Lilly And Company A process for preparing 4-substituted piperidines
SE0004245D0 (sv) 2000-11-20 2000-11-20 Pharmacia Ab Novel compounds and their use
ATE433962T1 (de) 2000-11-20 2009-07-15 Biovitrum Ab Publ Piperazinylpyrazinverbindungen als antagonisten des serotonin-5-ht2-rezeptors
AU2003243089B2 (en) 2002-06-19 2010-01-07 Biovitrum Ab (Publ) Novel compounds, their use and preparation
WO2006022420A1 (ja) 2004-08-25 2006-03-02 Takeda Pharmaceutical Company Limited 腹圧性尿失禁の予防・治療剤及びそのスクリーニング方法
TWI320783B (en) 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
JP5528699B2 (ja) 2006-05-16 2014-06-25 武田薬品工業株式会社 縮合複素環化合物およびその用途
JP5520051B2 (ja) 2007-11-15 2014-06-11 武田薬品工業株式会社 縮合ピリジン誘導体およびその用途
EP2510949A4 (de) 2009-12-11 2013-11-13 Astellas Pharma Inc Therapeutikum für fibromyalgie
WO2015066344A1 (en) 2013-11-01 2015-05-07 Arena Pharmaceuticals, Inc. 5-ht2c receptor agonists and compositions and methods of use
EP3733204A4 (de) 2017-12-27 2021-09-15 Takeda Pharmaceutical Company Limited Therapeutikum für belastungsinkontinenz und stuhlinkontinenz
WO2020220020A1 (en) * 2019-04-26 2020-10-29 The Regents Of The University Of California Silicon-fluoride heteroaromatic systems for applications in positron emission tomography (pet) molecular imaging

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0398413A1 (de) * 1989-05-16 1990-11-22 Duphar International Research B.V 3,4-Dehydropiperidin-Derivate mit psychotroper Wirkung
JP2883995B2 (ja) * 1990-03-14 1999-04-19 第一製薬株式会社 ピペリジン誘導体及びその製造中間体
TW222631B (de) * 1991-07-15 1994-04-21 Duphar Int Res
US5436246A (en) * 1992-09-17 1995-07-25 Merrell Dow Pharmaceuticals Inc. Serotonin receptor agents
US6021791A (en) * 1998-06-29 2000-02-08 Speedfam-Ipec Corporation Method and apparatus for immersion cleaning of semiconductor devices
WO2000000198A1 (en) * 1998-06-30 2000-01-06 Eli Lilly And Company Piperidine derivatives having effects on serotonin related systems
EP1100501A4 (de) * 1998-06-30 2002-12-04 Lilly Co Eli Pyrrolidine und pyrroliinederivate mit einer wirkung auf serotonin-relatierte systeme

Also Published As

Publication number Publication date
EP1204660A1 (de) 2002-05-15
DE60015146D1 (en) 2004-11-25
CA2378879A1 (en) 2001-02-08
WO2001009126A1 (en) 2001-02-08
JP2003506371A (ja) 2003-02-18
DE60015146T2 (de) 2006-02-16
EP1204660B1 (de) 2004-10-20
AU6339000A (en) 2001-02-19
ES2231229T3 (es) 2005-05-16

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties