CO5180579A1 - Composicion oral solida que comprende levidopa, carbidopa y entacapone - Google Patents

Composicion oral solida que comprende levidopa, carbidopa y entacapone

Info

Publication number
CO5180579A1
CO5180579A1 CO00048944A CO00048944A CO5180579A1 CO 5180579 A1 CO5180579 A1 CO 5180579A1 CO 00048944 A CO00048944 A CO 00048944A CO 00048944 A CO00048944 A CO 00048944A CO 5180579 A1 CO5180579 A1 CO 5180579A1
Authority
CO
Colombia
Prior art keywords
entacapone
carbidopa
solid oral
oral composition
levidopa
Prior art date
Application number
CO00048944A
Other languages
English (en)
Inventor
Matti Virkki
Vakervou Kari
Ritalia Marja
Partanen Marja
Niskanen Mervi
Lintulaakso Jarmo
Laaksonen Marja
Kervinen Lasse
Kallioinen Sari
Original Assignee
Orion Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8554988&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO5180579(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Orion Corp filed Critical Orion Corp
Publication of CO5180579A1 publication Critical patent/CO5180579A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid, pantothenic acid
    • A61K31/198Alpha-aminoacids, e.g. alanine, edetic acids [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Abstract

La presente invención se relaciona con una composición farmacéutica, en especial con una composición sólida oral, que comprende cantidades farmacéuticamente efectivas de entacapone, levodopa y carbidopa o de sus sales o hidratos farmacéuticamente aceptables y un excipiente farmacéuticamente aceptable, en donde el excipiente es un alcohol de azúcar o almidón o un alcohol de azúcar y almidón. El entacapone, la levodopa y la carbidopa son útiles para tratar el mal de Parkinson.
CO00048944A 1999-06-30 2000-06-29 Composicion oral solida que comprende levidopa, carbidopa y entacapone CO5180579A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FI991485A FI109453B (fi) 1999-06-30 1999-06-30 Farmaseuttinen koostumus

Publications (1)

Publication Number Publication Date
CO5180579A1 true CO5180579A1 (es) 2002-07-30

Family

ID=8554988

Family Applications (1)

Application Number Title Priority Date Filing Date
CO00048944A CO5180579A1 (es) 1999-06-30 2000-06-29 Composicion oral solida que comprende levidopa, carbidopa y entacapone

Country Status (42)

Country Link
US (2) US6500867B1 (es)
EP (1) EP1189608B1 (es)
JP (2) JP4204783B2 (es)
KR (1) KR100905428B1 (es)
CN (1) CN1168440C (es)
AR (1) AR033796A1 (es)
AT (1) ATE245417T1 (es)
AU (1) AU765932B2 (es)
BG (1) BG65364B1 (es)
BR (2) BR0011867A (es)
CA (1) CA2378469C (es)
CO (1) CO5180579A1 (es)
CZ (2) CZ304416B6 (es)
DE (1) DE60004052T2 (es)
DK (1) DK1189608T3 (es)
EA (1) EA004503B1 (es)
EE (1) EE05473B1 (es)
ES (1) ES2203495T3 (es)
FI (1) FI109453B (es)
FR (1) FR2797587A1 (es)
GE (1) GEP20043314B (es)
HK (1) HK1047040B (es)
HR (1) HRP20020088B1 (es)
HU (1) HU230395B1 (es)
IL (1) IL146807A (es)
IT (1) ITMI20001450A1 (es)
ME (1) ME00520B (es)
MX (1) MXPA01013167A (es)
MY (1) MY127685A (es)
NO (2) NO330260B1 (es)
NZ (1) NZ515780A (es)
PE (1) PE20010399A1 (es)
PL (1) PL197818B1 (es)
PT (1) PT1189608E (es)
RS (1) RS50368B (es)
SI (1) SI1189608T1 (es)
SK (1) SK286451B6 (es)
TR (1) TR200103763T2 (es)
TW (1) TWI241187B (es)
UA (1) UA75047C2 (es)
WO (1) WO2001001984A1 (es)
ZA (1) ZA200109868B (es)

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Also Published As

Publication number Publication date
ZA200109868B (en) 2003-05-28
DK1189608T3 (da) 2003-11-10
MXPA01013167A (es) 2002-07-02
HRP20020088B1 (en) 2007-05-31
CZ304416B6 (cs) 2014-04-23
IL146807A (en) 2006-10-05
BR0011867A (pt) 2002-03-05
DE60004052T2 (de) 2004-04-15
ITMI20001450A0 (it) 2000-06-28
YU92501A (sh) 2004-09-03
AR033796A1 (es) 2004-01-07
EE05473B1 (et) 2011-10-17
JP2008156373A (ja) 2008-07-10
NO330260B1 (no) 2011-03-14
CA2378469C (en) 2009-10-06
AU765932B2 (en) 2003-10-02
HK1047040A1 (en) 2003-02-07
PE20010399A1 (es) 2001-04-10
WO2001001984A1 (en) 2001-01-11
GEP20043314B (en) 2004-02-10
SI1189608T1 (en) 2004-04-30
JP4204783B2 (ja) 2009-01-07
SK286451B6 (sk) 2008-10-07
PL352775A1 (en) 2003-09-08
US6797732B2 (en) 2004-09-28
DE60004052D1 (de) 2003-08-28
EP1189608A1 (en) 2002-03-27
CN1168440C (zh) 2004-09-29
HUP0202273A3 (en) 2002-11-28
CA2378469A1 (en) 2001-01-11
HK1047040B (zh) 2005-04-29
PT1189608E (pt) 2003-12-31
BG65364B1 (bg) 2008-04-30
NZ515780A (en) 2004-06-25
RS50368B (sr) 2009-11-10
EP1189608B1 (en) 2003-07-23
ITMI20001450A1 (it) 2001-12-28
US6500867B1 (en) 2002-12-31
EA200200106A1 (ru) 2002-06-27
NO20016203L (no) 2002-02-25
SK19232001A3 (sk) 2002-06-04
NO20110090L (no) 2002-02-25
ME00520B (me) 2011-10-10
FI991485A (fi) 2000-12-31
EE200100716A (et) 2003-02-17
KR100905428B1 (ko) 2009-06-30
MY127685A (en) 2006-12-29
HRP20020088A2 (en) 2005-10-31
BRPI0011867B8 (pt) 2021-05-25
TR200103763T2 (tr) 2002-04-22
ES2203495T3 (es) 2004-04-16
ATE245417T1 (de) 2003-08-15
CN1358090A (zh) 2002-07-10
BRPI0011867B1 (pt) 2019-01-08
FR2797587A1 (fr) 2001-02-23
BG106251A (en) 2002-08-30
KR20020010155A (ko) 2002-02-02
TWI241187B (en) 2005-10-11
JP2003503454A (ja) 2003-01-28
EA004503B1 (ru) 2004-04-29
NO20016203D0 (no) 2001-12-18
HUP0202273A2 (en) 2002-10-28
CZ303010B6 (cs) 2012-02-29
UA75047C2 (en) 2006-03-15
PL197818B1 (pl) 2008-04-30
AU5830600A (en) 2001-01-22
FI991485A0 (fi) 1999-06-30
HU230395B1 (hu) 2016-04-28
CZ20014636A3 (cs) 2002-05-15
JP4885896B2 (ja) 2012-02-29
US20030017201A1 (en) 2003-01-23
FI109453B (fi) 2002-08-15

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