CN1229334C - α4介导的细胞粘附的抑制剂 - Google Patents

α4介导的细胞粘附的抑制剂 Download PDF

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Publication number
CN1229334C
CN1229334C CNB018149871A CN01814987A CN1229334C CN 1229334 C CN1229334 C CN 1229334C CN B018149871 A CNB018149871 A CN B018149871A CN 01814987 A CN01814987 A CN 01814987A CN 1229334 C CN1229334 C CN 1229334C
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compound
group
dimethoxy
phenylalanine
formula
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Expired - Fee Related
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CNB018149871A
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Chinese (zh)
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CN1449377A (zh
Inventor
筑本美喜子
野村纯宏
川口隆行
久米俊行
I·瑟卡
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Mitsubishi Tanabe Pharma Corp
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Tanabe Seiyaku Co Ltd
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    • C07ORGANIC CHEMISTRY
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    • C07C233/00Carboxylic acid amides
    • C07C233/64Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
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CNB018149871A 2000-08-31 2001-08-27 α4介导的细胞粘附的抑制剂 Expired - Fee Related CN1229334C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22912800P 2000-08-31 2000-08-31
US60/229,128 2000-08-31

Publications (2)

Publication Number Publication Date
CN1449377A CN1449377A (zh) 2003-10-15
CN1229334C true CN1229334C (zh) 2005-11-30

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US (6) US7026501B2 (enExample)
EP (1) EP1315694B1 (enExample)
JP (1) JP3899022B2 (enExample)
KR (1) KR100528049B1 (enExample)
CN (1) CN1229334C (enExample)
AR (1) AR034556A1 (enExample)
AT (1) ATE292615T1 (enExample)
AU (2) AU2001286778B2 (enExample)
BR (1) BR0113629A (enExample)
CA (1) CA2418054C (enExample)
CZ (1) CZ303460B6 (enExample)
DE (1) DE60109943T2 (enExample)
DK (1) DK1315694T3 (enExample)
ES (1) ES2240509T3 (enExample)
HK (1) HK1052684B (enExample)
HU (1) HUP0302693A3 (enExample)
IL (2) IL154305A0 (enExample)
MX (1) MXPA03001837A (enExample)
MY (1) MY129000A (enExample)
NO (1) NO327861B1 (enExample)
NZ (1) NZ524043A (enExample)
PL (1) PL206656B1 (enExample)
PT (1) PT1315694E (enExample)
RU (1) RU2250895C2 (enExample)
SI (1) SI1315694T1 (enExample)
TW (1) TWI224587B (enExample)
WO (1) WO2002018320A2 (enExample)
ZA (1) ZA200301039B (enExample)

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