CN1229334C - α4介导的细胞粘附的抑制剂 - Google Patents

α4介导的细胞粘附的抑制剂 Download PDF

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Publication number
CN1229334C
CN1229334C CNB018149871A CN01814987A CN1229334C CN 1229334 C CN1229334 C CN 1229334C CN B018149871 A CNB018149871 A CN B018149871A CN 01814987 A CN01814987 A CN 01814987A CN 1229334 C CN1229334 C CN 1229334C
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compound
group
dimethoxy
phenylalanine
formula
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Expired - Fee Related
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CNB018149871A
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Chinese (zh)
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CN1449377A (zh
Inventor
筑本美喜子
野村纯宏
川口隆行
久米俊行
I·瑟卡
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Mitsubishi Tanabe Pharma Corp
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Tanabe Seiyaku Co Ltd
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    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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CNB018149871A 2000-08-31 2001-08-27 α4介导的细胞粘附的抑制剂 Expired - Fee Related CN1229334C (zh)

Applications Claiming Priority (2)

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US22912800P 2000-08-31 2000-08-31
US60/229,128 2000-08-31

Publications (2)

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CN1449377A CN1449377A (zh) 2003-10-15
CN1229334C true CN1229334C (zh) 2005-11-30

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US (6) US7026501B2 (enExample)
EP (1) EP1315694B1 (enExample)
JP (1) JP3899022B2 (enExample)
KR (1) KR100528049B1 (enExample)
CN (1) CN1229334C (enExample)
AR (1) AR034556A1 (enExample)
AT (1) ATE292615T1 (enExample)
AU (2) AU8677801A (enExample)
BR (1) BR0113629A (enExample)
CA (1) CA2418054C (enExample)
CZ (1) CZ303460B6 (enExample)
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IL (2) IL154305A0 (enExample)
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NO (1) NO327861B1 (enExample)
NZ (1) NZ524043A (enExample)
PL (1) PL206656B1 (enExample)
PT (1) PT1315694E (enExample)
RU (1) RU2250895C2 (enExample)
SI (1) SI1315694T1 (enExample)
TW (1) TWI224587B (enExample)
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CN114222730B (zh) 2019-08-14 2024-09-10 吉利德科学公司 用于抑制α4β7整合素的化合物

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CZ303460B6 (cs) 2012-09-26
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US20030176498A1 (en) 2003-09-18
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US20050282900A1 (en) 2005-12-22
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