RU2250895C2 - ИНГИБИТОРЫ КЛЕТОЧНОЙ АДГЕЗИИ, ОПОСРЕДОВАННОЙ α4-ИНТЕГРИНАМИ - Google Patents

ИНГИБИТОРЫ КЛЕТОЧНОЙ АДГЕЗИИ, ОПОСРЕДОВАННОЙ α4-ИНТЕГРИНАМИ Download PDF

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RU2250895C2
RU2250895C2 RU2003105885/04A RU2003105885A RU2250895C2 RU 2250895 C2 RU2250895 C2 RU 2250895C2 RU 2003105885/04 A RU2003105885/04 A RU 2003105885/04A RU 2003105885 A RU2003105885 A RU 2003105885A RU 2250895 C2 RU2250895 C2 RU 2250895C2
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Russia
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group
compound
pharmaceutically acceptable
phenylalanine
acceptable salt
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RU2003105885/04A
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English (en)
Russian (ru)
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RU2003105885A (ru
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Такаюки КАВАГУТИ (JP)
Такаюки КАВАГУТИ
Сумихиро НОМУРА (JP)
Сумихиро Номура
Микико ЦУКИМОТО (JP)
Микико ЦУКИМОТО
Тошиюки КУМЕ (JP)
Тошиюки КУМЕ
Ила СИРКАР (US)
Ила СИРКАР
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Танабе Сейяку Ко., Лтд.
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
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RU2003105885/04A 2000-08-31 2001-08-27 ИНГИБИТОРЫ КЛЕТОЧНОЙ АДГЕЗИИ, ОПОСРЕДОВАННОЙ α4-ИНТЕГРИНАМИ RU2250895C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22912800P 2000-08-31 2000-08-31
US60/229,128 2000-08-31

Publications (2)

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RU2003105885A RU2003105885A (ru) 2004-08-10
RU2250895C2 true RU2250895C2 (ru) 2005-04-27

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US (6) US7026501B2 (enExample)
EP (1) EP1315694B1 (enExample)
JP (1) JP3899022B2 (enExample)
KR (1) KR100528049B1 (enExample)
CN (1) CN1229334C (enExample)
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