CA1235415A - Camptothecin derivatives and process for preparing same - Google Patents

Camptothecin derivatives and process for preparing same

Info

Publication number
CA1235415A
CA1235415A CA000458228A CA458228A CA1235415A CA 1235415 A CA1235415 A CA 1235415A CA 000458228 A CA000458228 A CA 000458228A CA 458228 A CA458228 A CA 458228A CA 1235415 A CA1235415 A CA 1235415A
Authority
CA
Canada
Prior art keywords
group
camptothecin
formula
starting material
carbonyloxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000458228A
Other languages
English (en)
French (fr)
Inventor
Tadashi Miyasaka
Seigo Sawada
Kenichiro Nokata
Eiichi Sugino
Masahiko Mutai
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Yakult Honsha Co Ltd
Original Assignee
Yakult Honsha Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yakult Honsha Co Ltd filed Critical Yakult Honsha Co Ltd
Application granted granted Critical
Publication of CA1235415A publication Critical patent/CA1235415A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
CA000458228A 1983-07-14 1984-07-05 Camptothecin derivatives and process for preparing same Expired CA1235415A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP58126946A JPS6019790A (ja) 1983-07-14 1983-07-14 新規なカンプトテシン誘導体
JP126946/58 1983-07-14

Publications (1)

Publication Number Publication Date
CA1235415A true CA1235415A (en) 1988-04-19

Family

ID=14947803

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000458228A Expired CA1235415A (en) 1983-07-14 1984-07-05 Camptothecin derivatives and process for preparing same

Country Status (8)

Country Link
US (1) US4604463A (enExample)
EP (1) EP0137145B1 (enExample)
JP (1) JPS6019790A (enExample)
AT (1) ATE33839T1 (enExample)
CA (1) CA1235415A (enExample)
DE (2) DE137145T1 (enExample)
LU (1) LU90074I2 (enExample)
NL (1) NL980026I2 (enExample)

Families Citing this family (171)

* Cited by examiner, † Cited by third party
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NL980026I2 (nl) 1999-02-01
ATE33839T1 (de) 1988-05-15
JPS6019790A (ja) 1985-01-31
DE137145T1 (de) 1985-11-21
DE3470744D1 (en) 1988-06-01
JPH034077B2 (enExample) 1991-01-22
US4604463A (en) 1986-08-05
LU90074I2 (fr) 1997-08-21
EP0137145A1 (en) 1985-04-17
NL980026I1 (nl) 1998-11-02
EP0137145B1 (en) 1988-04-27

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