BRPI0917705A2 - composto, pró-droga, composição farmacêutica, método para tratar ou prevenir uma doença ou condição, e, uso do composto - Google Patents

composto, pró-droga, composição farmacêutica, método para tratar ou prevenir uma doença ou condição, e, uso do composto

Info

Publication number
BRPI0917705A2
BRPI0917705A2 BRPI0917705A BRPI0917705A BRPI0917705A2 BR PI0917705 A2 BRPI0917705 A2 BR PI0917705A2 BR PI0917705 A BRPI0917705 A BR PI0917705A BR PI0917705 A BRPI0917705 A BR PI0917705A BR PI0917705 A2 BRPI0917705 A2 BR PI0917705A2
Authority
BR
Brazil
Prior art keywords
compound
prodrug
disease
treating
preventing
Prior art date
Application number
BRPI0917705A
Other languages
English (en)
Portuguese (pt)
Inventor
Haruyuki Nishida
Ikuo Fujimori
Yasuyoshi Arikawa
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41508823&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0917705(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of BRPI0917705A2 publication Critical patent/BRPI0917705A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BRPI0917705A 2008-08-27 2009-08-26 composto, pró-droga, composição farmacêutica, método para tratar ou prevenir uma doença ou condição, e, uso do composto BRPI0917705A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2008218851 2008-08-27
JP2008269099 2008-10-17
PCT/JP2009/065279 WO2010024451A1 (en) 2008-08-27 2009-08-26 Pyrrole compounds

Publications (1)

Publication Number Publication Date
BRPI0917705A2 true BRPI0917705A2 (pt) 2016-02-16

Family

ID=41508823

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0917705A BRPI0917705A2 (pt) 2008-08-27 2009-08-26 composto, pró-droga, composição farmacêutica, método para tratar ou prevenir uma doença ou condição, e, uso do composto

Country Status (38)

Country Link
US (3) US8592597B2 (https=)
EP (1) EP2318390B1 (https=)
JP (1) JP5638515B2 (https=)
KR (1) KR101629181B1 (https=)
CN (1) CN102197033B (https=)
AR (1) AR073136A1 (https=)
AU (1) AU2009284867B2 (https=)
BR (1) BRPI0917705A2 (https=)
CA (1) CA2735162C (https=)
CL (1) CL2011000402A1 (https=)
CO (1) CO6321166A2 (https=)
CR (1) CR20110169A (https=)
CY (1) CY1114452T1 (https=)
DK (1) DK2318390T3 (https=)
DO (1) DOP2011000061A (https=)
EA (1) EA019741B1 (https=)
EC (1) ECSP11010912A (https=)
ES (1) ES2423289T3 (https=)
GE (1) GEP20135786B (https=)
HR (1) HRP20130653T1 (https=)
IL (1) IL211335A (https=)
JO (1) JO2871B1 (https=)
MA (1) MA32647B1 (https=)
ME (1) ME01598B (https=)
MX (1) MX2011001955A (https=)
MY (1) MY152008A (https=)
NZ (1) NZ591793A (https=)
PE (2) PE20110300A1 (https=)
PL (1) PL2318390T3 (https=)
PT (1) PT2318390E (https=)
RS (1) RS52872B (https=)
SI (1) SI2318390T1 (https=)
SM (1) SMT201300085B (https=)
TW (1) TWI473798B (https=)
UA (1) UA105185C2 (https=)
UY (1) UY32074A (https=)
WO (1) WO2010024451A1 (https=)
ZA (1) ZA201101774B (https=)

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US10039813B2 (en) 2012-02-07 2018-08-07 Massachusetts Institute Of Technology Use of antagonists of ghrelin or ghrelin receptor to prevent or treat stress-sensitive psychiatric illness
AR091567A1 (es) 2012-06-27 2015-02-11 Takeda Pharmaceutical Preparacion liquida, metodo, kit de inyeccion
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WO2014144231A1 (en) 2013-03-15 2014-09-18 Massachusetts Institute Of Technology Use of antagonists of growth hormone or growth hormone receptor to prevent or treat stress-sensitive psychiatric illness
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CA2994604A1 (en) 2015-08-07 2017-02-16 Bayer Cropscience Aktiengesellschaft 2-(het)aryl-substituted condensed heterocyclic derivatives as pest control agents
CN106430006B (zh) * 2016-08-18 2018-06-12 国网湖南省电力公司带电作业中心 配电线路移动式绝缘登高作业装置及方法
CN108203430A (zh) * 2016-12-16 2018-06-26 天地人和生物科技有限公司 一种新型可逆性质子泵抑制剂及其制备方法和用途
BR112020000318A2 (pt) 2017-07-10 2020-07-14 Takeda Pharmaceutical Company Limited preparação
KR102126576B1 (ko) 2018-09-19 2020-06-24 주식회사 대웅제약 4-메톡시 피롤 유도체의 제조 방법
CN113527536B (zh) * 2020-04-21 2024-03-22 杭州德柯医疗科技有限公司 一种含氟多糖高分子化合物及其制备方法
MX2022016515A (es) * 2020-06-17 2023-01-30 Ildong Pharmaceutical Co Ltd Nuevo inhibidor de la secrecion de acido y uso del mismo.
EP4074317A1 (en) 2021-04-14 2022-10-19 Bayer AG Phosphorus derivatives as novel sos1 inhibitors
CN113620930B (zh) * 2021-07-12 2022-08-16 南京烁慧医药科技有限公司 一种含磺酰胺结构的化合物及其制备方法和应用、一种药物组合物及应用
KR20240119083A (ko) * 2021-12-15 2024-08-06 일동제약(주) 1-설포닐 피롤 유도체의 신규 염, 이의 제조 방법 및 이를 포함하는 약학 조성물
US20250084026A1 (en) * 2021-12-15 2025-03-13 Ildong Pharmaceutical Co., Ltd. Novel salt of 1-sulfonyl pyrrole derivative, preparation method thereof and pharmaceutical composition comprising thereof
KR20230102353A (ko) * 2021-12-30 2023-07-07 주식회사 대웅제약 삼중음성유방암의 예방 또는 치료용 약학적 조성물
WO2026029625A1 (ko) * 2024-08-02 2026-02-05 일양약품주식회사 4-사이클로프로필 피롤 유도체 및 이의 용도

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Also Published As

Publication number Publication date
PE20110300A1 (es) 2011-06-16
KR20110071067A (ko) 2011-06-28
DK2318390T3 (da) 2013-07-08
PT2318390E (pt) 2013-07-10
ECSP11010912A (es) 2011-04-29
JO2871B1 (en) 2015-03-15
CA2735162A1 (en) 2010-03-04
EA019741B1 (ru) 2014-05-30
HRP20130653T1 (en) 2013-08-31
US20140031393A1 (en) 2014-01-30
GEP20135786B (en) 2013-03-11
TW201010993A (en) 2010-03-16
DOP2011000061A (es) 2011-04-15
MY152008A (en) 2014-08-15
KR101629181B1 (ko) 2016-06-13
CO6321166A2 (es) 2011-09-20
CN102197033B (zh) 2014-07-16
JP5638515B2 (ja) 2014-12-10
IL211335A (en) 2013-12-31
MA32647B1 (fr) 2011-09-01
AU2009284867A2 (en) 2011-04-21
EA201170384A1 (ru) 2011-10-31
ZA201101774B (en) 2012-06-27
CY1114452T1 (el) 2016-10-05
TWI473798B (zh) 2015-02-21
EP2318390A1 (en) 2011-05-11
HK1157756A1 (en) 2012-07-06
CA2735162C (en) 2015-06-23
US8969387B2 (en) 2015-03-03
MX2011001955A (es) 2011-03-29
PE20141174A1 (es) 2014-09-19
ME01598B (me) 2014-09-20
US8592597B2 (en) 2013-11-26
CN102197033A (zh) 2011-09-21
US8993598B2 (en) 2015-03-31
AU2009284867A1 (en) 2010-03-04
ES2423289T3 (es) 2013-09-19
EP2318390B1 (en) 2013-05-01
NZ591793A (en) 2012-11-30
US20110172275A1 (en) 2011-07-14
SI2318390T1 (sl) 2013-08-30
SMT201300085B (it) 2013-09-06
UA105185C2 (uk) 2014-04-25
IL211335A0 (en) 2011-04-28
WO2010024451A1 (en) 2010-03-04
AU2009284867B2 (en) 2014-08-28
JP2012501296A (ja) 2012-01-19
RS52872B (sr) 2013-12-31
UY32074A (es) 2010-03-26
CL2011000402A1 (es) 2011-07-29
AR073136A1 (es) 2010-10-13
US20100056577A1 (en) 2010-03-04
CR20110169A (es) 2011-05-16
PL2318390T3 (pl) 2013-09-30

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