BG51452A3 - Метод за получаване на производни на аминокиселини - Google Patents

Метод за получаване на производни на аминокиселини Download PDF

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Publication number
BG51452A3
BG51452A3 BG093425A BG9342590A BG51452A3 BG 51452 A3 BG51452 A3 BG 51452A3 BG 093425 A BG093425 A BG 093425A BG 9342590 A BG9342590 A BG 9342590A BG 51452 A3 BG51452 A3 BG 51452A3
Authority
BG
Bulgaria
Prior art keywords
amino acid
compound
acid derivatives
benzyloxycarbonyl
pharmaceutically acceptable
Prior art date
Application number
BG093425A
Other languages
Bulgarian (bg)
English (en)
Inventor
Joseph Martin
Sally Redshaw
Original Assignee
F. Hoffmann - La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F. Hoffmann - La Roche Ag filed Critical F. Hoffmann - La Roche Ag
Publication of BG51452A3 publication Critical patent/BG51452A3/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/021—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)n-C(=0)-, n being 5 or 6; for n > 6, classification in C07K5/06 - C07K5/10, according to the moiety having normal peptide bonds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Communicable Diseases (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Confectionery (AREA)
  • Cleaning Or Clearing Of The Surface Of Open Water (AREA)
  • Measurement Of Force In General (AREA)
BG093425A 1989-12-11 1990-12-10 Метод за получаване на производни на аминокиселини BG51452A3 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB898927913A GB8927913D0 (en) 1989-12-11 1989-12-11 Amino acid derivatives
SG120493A SG120493G (en) 1989-12-11 1993-11-02 N-tert-Butyl-decahydro-2(3-amino-2-hydroxy-4-phenyl-butyl) isoquinoline-3-carboxamide and asparaginyl derivatives thereof

Publications (1)

Publication Number Publication Date
BG51452A3 true BG51452A3 (bg) 1993-05-14

Family

ID=26296345

Family Applications (1)

Application Number Title Priority Date Filing Date
BG093425A BG51452A3 (bg) 1989-12-11 1990-12-10 Метод за получаване на производни на аминокиселини

Country Status (48)

Country Link
US (1) US5196438A (cs)
EP (1) EP0432695B1 (cs)
JP (1) JP2807093B2 (cs)
KR (1) KR970005912B1 (cs)
CN (2) CN1066329C (cs)
AT (1) ATE122661T1 (cs)
AU (1) AU634319B2 (cs)
BG (1) BG51452A3 (cs)
BR (1) BR9006264A (cs)
CA (1) CA2030433C (cs)
CU (1) CU22305A3 (cs)
CZ (1) CZ280558B6 (cs)
DE (2) DE19675051I2 (cs)
DK (1) DK0432695T3 (cs)
DZ (1) DZ1467A1 (cs)
EG (1) EG19722A (cs)
ES (1) ES2072959T3 (cs)
FI (2) FI973895A0 (cs)
GB (2) GB8927913D0 (cs)
GR (1) GR3017114T3 (cs)
HK (1) HK129093A (cs)
HR (1) HRP930341B1 (cs)
HU (2) HU207298B (cs)
ID (1) ID1018B (cs)
IE (1) IE67523B1 (cs)
IL (1) IL96550A (cs)
IN (1) IN172553B (cs)
IS (1) IS1803B (cs)
LT (1) LT3682B (cs)
LU (1) LU90014I2 (cs)
LV (1) LV5738B4 (cs)
MA (1) MA22014A1 (cs)
MC (1) MC2195A1 (cs)
MT (1) MTP1075B (cs)
MW (1) MW8890A1 (cs)
MX (1) MX173630B (cs)
NL (1) NL970013I2 (cs)
NO (1) NO176566C (cs)
OA (1) OA09334A (cs)
PL (1) PL165225B1 (cs)
PT (1) PT96145B (cs)
RO (1) RO107942B1 (cs)
RU (1) RU2071470C1 (cs)
SG (1) SG120493G (cs)
SI (1) SI9012315B (cs)
SK (1) SK576590A3 (cs)
ZA (1) ZA909743B (cs)
ZW (1) ZW17490A1 (cs)

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ZA909743B (en) 1991-08-28
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OA09334A (fr) 1992-09-15
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HUT56073A (en) 1991-07-29
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LTIP862A (en) 1995-03-27
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