BG107739A - Комбинация от антагонист на св1 рецептор и сибутрамин, фармацевтични състави, които ги съдържат, и използването им за лечение на затлъстяване - Google Patents

Комбинация от антагонист на св1 рецептор и сибутрамин, фармацевтични състави, които ги съдържат, и използването им за лечение на затлъстяване Download PDF

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Publication number
BG107739A
BG107739A BG107739A BG10773903A BG107739A BG 107739 A BG107739 A BG 107739A BG 107739 A BG107739 A BG 107739A BG 10773903 A BG10773903 A BG 10773903A BG 107739 A BG107739 A BG 107739A
Authority
BG
Bulgaria
Prior art keywords
methyl
chlorophenyl
methylsulfonyl
bis
azetidine
Prior art date
Application number
BG107739A
Other languages
Bulgarian (bg)
English (en)
Inventor
Odile Piot-Grosjean
Philippe Picaut
Francois Petitet
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8854974&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG107739(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of BG107739A publication Critical patent/BG107739A/bg

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Plural Heterocyclic Compounds (AREA)
BG107739A 2000-10-04 2003-04-17 Комбинация от антагонист на св1 рецептор и сибутрамин, фармацевтични състави, които ги съдържат, и използването им за лечение на затлъстяване BG107739A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0012646A FR2814678B1 (fr) 2000-10-04 2000-10-04 Association d'un antagoniste du recepteur cb1 et de sibutramine, les compositions pharmaceutiques les contenant et leur utilisation pour la traitement de l'obesite
PCT/FR2001/003022 WO2002028346A2 (fr) 2000-10-04 2001-10-01 Association d'un antagoniste du recepteur cb1 et de sibutramine, pour le traitement de l'obesite

Publications (1)

Publication Number Publication Date
BG107739A true BG107739A (bg) 2004-01-30

Family

ID=8854974

Family Applications (1)

Application Number Title Priority Date Filing Date
BG107739A BG107739A (bg) 2000-10-04 2003-04-17 Комбинация от антагонист на св1 рецептор и сибутрамин, фармацевтични състави, които ги съдържат, и използването им за лечение на затлъстяване

Country Status (29)

Country Link
EP (1) EP1328269B2 (da)
JP (1) JP4221221B2 (da)
KR (1) KR20030036885A (da)
CN (1) CN100409845C (da)
AT (1) ATE267595T1 (da)
AU (2) AU2001293936B2 (da)
BG (1) BG107739A (da)
BR (1) BR0114410A (da)
CA (1) CA2424934A1 (da)
DE (1) DE60103556T3 (da)
DK (1) DK1328269T5 (da)
EA (1) EA005924B1 (da)
EE (1) EE200300121A (da)
ES (1) ES2217191T5 (da)
FR (1) FR2814678B1 (da)
HR (1) HRP20030249A2 (da)
HU (1) HUP0302044A3 (da)
IL (1) IL155236A0 (da)
MX (1) MXPA03002845A (da)
NO (1) NO20031521L (da)
NZ (1) NZ524904A (da)
PL (1) PL362833A1 (da)
PT (1) PT1328269E (da)
SI (1) SI1328269T2 (da)
SK (1) SK4032003A3 (da)
TR (1) TR200401264T4 (da)
WO (1) WO2002028346A2 (da)
YU (1) YU26103A (da)
ZA (1) ZA200303015B (da)

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WO2005049615A1 (en) * 2003-11-21 2005-06-02 Pfizer Products Inc. Pyrazolo`1,5-a!`1,3,5! triazin -4-one derivatives as cb1 receptor antagonists
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EP1716132B1 (en) 2004-01-28 2010-08-25 F. Hoffmann-La Roche AG Spiro-benzodioxoles and their use as cb1 antagonists
JP2007536298A (ja) 2004-05-10 2007-12-13 エフ．ホフマン−ラ　ロシュ　アーゲー 肥満を処置するためのピロールまたはイミダゾールアミド
US20060025448A1 (en) 2004-07-22 2006-02-02 Cadila Healthcare Limited Hair growth stimulators
WO2006039334A1 (en) * 2004-09-29 2006-04-13 Schering Corporation Combinations of substituted azetidonones and cb1 antagonists
FR2876689B1 (fr) * 2004-10-14 2008-02-22 Aventis Pharma Sa Nouveau procede et intermediaires de preparation de derives de n-(1-benzhydryl-azetidin-3-yl)-n-phenyl-methylsulfonamide
CA2585175A1 (en) 2004-10-25 2006-05-04 Solvay Pharmaceuticals Gmbh Pharmaceutical compositions comprising cb1 cannabinoid receptor antagonists and potassium channel openers for the treatment of diabetes mellitus type i, obesity and related conditions
ES2309812T3 (es) 2004-10-27 2008-12-16 F. Hoffmann-La Roche Ag Nuevos derivados de indol o benzimidazol.
EP1812418B1 (en) 2004-11-09 2010-10-27 F. Hoffmann-La Roche AG Dibenzosuberone derivatives
DE602006007563D1 (de) 2005-04-06 2009-08-13 Hoffmann La Roche Agonisten
US7906652B2 (en) 2005-11-28 2011-03-15 Merck Sharp & Dohme Corp. Heterocycle-substituted 3-alkyl azetidine derivatives
US20080027087A1 (en) * 2006-02-21 2008-01-31 Ampla Pharmaceuticals, Inc. CB1 antagonists and inverse agonists
WO2007110449A1 (en) * 2006-03-29 2007-10-04 Euro-Celtique S.A. Benzenesulfonamide compounds and their use
WO2007118854A1 (en) 2006-04-13 2007-10-25 Euro-Celtique S.A. Benzenesulfonamide compounds and the use thereof
US8791264B2 (en) 2006-04-13 2014-07-29 Purdue Pharma L.P. Benzenesulfonamide compounds and their use as blockers of calcium channels
US7629346B2 (en) 2006-06-19 2009-12-08 Hoffmann-La Roche Inc. Pyrazinecarboxamide derivatives as CB1 antagonists
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Also Published As

Publication number Publication date
MXPA03002845A (es) 2004-09-10
AU9393601A (en) 2002-04-15
ES2217191T5 (es) 2009-02-16
CN100409845C (zh) 2008-08-13
HUP0302044A2 (hu) 2003-11-28
EP1328269B2 (fr) 2008-07-30
ATE267595T1 (de) 2004-06-15
CN1473040A (zh) 2004-02-04
FR2814678B1 (fr) 2002-12-20
ZA200303015B (en) 2004-02-26
PT1328269E (pt) 2004-08-31
CA2424934A1 (fr) 2002-04-11
DE60103556T2 (de) 2005-06-30
WO2002028346A2 (fr) 2002-04-11
WO2002028346A3 (fr) 2002-08-29
ES2217191T3 (es) 2004-11-01
AU2001293936B2 (en) 2007-01-25
EA200300441A1 (ru) 2003-08-28
NO20031521D0 (no) 2003-04-03
SI1328269T1 (en) 2004-10-31
KR20030036885A (ko) 2003-05-09
BR0114410A (pt) 2004-02-17
DK1328269T3 (da) 2004-09-20
FR2814678A1 (fr) 2002-04-05
PL362833A1 (en) 2004-11-02
EA005924B1 (ru) 2005-08-25
DK1328269T5 (da) 2009-03-16
HRP20030249A2 (en) 2005-02-28
EP1328269A2 (fr) 2003-07-23
YU26103A (sh) 2006-08-17
NZ524904A (en) 2004-11-26
DK1328269T4 (da) 2008-11-24
IL155236A0 (en) 2003-11-23
NO20031521L (no) 2003-04-24
SI1328269T2 (sl) 2008-12-31
EP1328269B1 (fr) 2004-05-26
HUP0302044A3 (en) 2005-05-30
TR200401264T4 (tr) 2004-07-21
SK4032003A3 (en) 2003-09-11
JP2004512279A (ja) 2004-04-22
DE60103556D1 (de) 2004-07-01
EE200300121A (et) 2005-04-15
DE60103556T3 (de) 2009-04-09
JP4221221B2 (ja) 2009-02-12

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