YU26103A - Kombinacija jednog antagonista cbi receptora i sibutramina, farmaceutski oblici koji ih sadrže i njihova upotreba u lečenju gojaznosti - Google Patents

Kombinacija jednog antagonista cbi receptora i sibutramina, farmaceutski oblici koji ih sadrže i njihova upotreba u lečenju gojaznosti

Info

Publication number
YU26103A
YU26103A YU26103A YUP26103A YU26103A YU 26103 A YU26103 A YU 26103A YU 26103 A YU26103 A YU 26103A YU P26103 A YUP26103 A YU P26103A YU 26103 A YU26103 A YU 26103A
Authority
YU
Yugoslavia
Prior art keywords
sibutramin
association
pharmaceutical compositions
compositions containing
receptor antagonist
Prior art date
Application number
YU26103A
Other languages
English (en)
Inventor
Odile Piot-Grosjean
Philippe Picaut
Francois Petit
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8854974&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=YU26103(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of YU26103A publication Critical patent/YU26103A/sh

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Ovaj pronalazak se odnosi na kombinaciju jednog antagoniste CB1 receptora i sibutramina, farmaceutske oblike koji ih sadrže i njihovu upotrebu u lečenju gojaznosti.[The invention concerns the association of the CB1 receptor antagonist and a sibutramin, pharmaceutical compositions containing same and use thereof for treating obesity.
YU26103A 2000-10-04 2001-10-01 Kombinacija jednog antagonista cbi receptora i sibutramina, farmaceutski oblici koji ih sadrže i njihova upotreba u lečenju gojaznosti YU26103A (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0012646A FR2814678B1 (fr) 2000-10-04 2000-10-04 Association d'un antagoniste du recepteur cb1 et de sibutramine, les compositions pharmaceutiques les contenant et leur utilisation pour la traitement de l'obesite

Publications (1)

Publication Number Publication Date
YU26103A true YU26103A (sh) 2006-08-17

Family

ID=8854974

Family Applications (1)

Application Number Title Priority Date Filing Date
YU26103A YU26103A (sh) 2000-10-04 2001-10-01 Kombinacija jednog antagonista cbi receptora i sibutramina, farmaceutski oblici koji ih sadrže i njihova upotreba u lečenju gojaznosti

Country Status (29)

Country Link
EP (1) EP1328269B2 (sh)
JP (1) JP4221221B2 (sh)
KR (1) KR20030036885A (sh)
CN (1) CN100409845C (sh)
AT (1) ATE267595T1 (sh)
AU (2) AU2001293936B2 (sh)
BG (1) BG107739A (sh)
BR (1) BR0114410A (sh)
CA (1) CA2424934A1 (sh)
DE (1) DE60103556T3 (sh)
DK (1) DK1328269T5 (sh)
EA (1) EA005924B1 (sh)
EE (1) EE200300121A (sh)
ES (1) ES2217191T5 (sh)
FR (1) FR2814678B1 (sh)
HR (1) HRP20030249A2 (sh)
HU (1) HUP0302044A3 (sh)
IL (1) IL155236A0 (sh)
MX (1) MXPA03002845A (sh)
NO (1) NO20031521L (sh)
NZ (1) NZ524904A (sh)
PL (1) PL362833A1 (sh)
PT (1) PT1328269E (sh)
SI (1) SI1328269T2 (sh)
SK (1) SK4032003A3 (sh)
TR (1) TR200401264T4 (sh)
WO (1) WO2002028346A2 (sh)
YU (1) YU26103A (sh)
ZA (1) ZA200303015B (sh)

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EP1749002B1 (en) 2004-05-10 2009-05-27 F.Hoffmann-La Roche Ag Pyrrole or imidazole amides for treating obesity
US20060025448A1 (en) 2004-07-22 2006-02-02 Cadila Healthcare Limited Hair growth stimulators
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FR2876689B1 (fr) * 2004-10-14 2008-02-22 Aventis Pharma Sa Nouveau procede et intermediaires de preparation de derives de n-(1-benzhydryl-azetidin-3-yl)-n-phenyl-methylsulfonamide
JP2008517976A (ja) 2004-10-25 2008-05-29 ゾルファイ ファーマスーティカルズ ゲゼルシャフト ミット ベシュレンクテル ハフツング Cb1カンナビノイド受容体拮抗薬及びカリウムチャンネルオープナーから成る、真性糖尿病1型、肥満及び関連症状の治療用の医薬組成物
RU2394027C2 (ru) 2004-10-27 2010-07-10 Ф. Хоффманн-Ля Рош Аг Новые индольные или бензимидазольные производные
WO2006050842A1 (en) 2004-11-09 2006-05-18 F. Hoffmann-La Roche Ag Dibenzosuberone derivatives
RU2404164C2 (ru) 2005-04-06 2010-11-20 Ф.Хоффманн-Ля Рош Аг Производные пиридин-3-карбоксамида в качестве обратных агонистов св1
US7906652B2 (en) 2005-11-28 2011-03-15 Merck Sharp & Dohme Corp. Heterocycle-substituted 3-alkyl azetidine derivatives
WO2007102999A2 (en) * 2006-02-21 2007-09-13 Ampla Pharmaceuticals Inc. Cb1 antagonists and inverse agonists
WO2007110449A1 (en) * 2006-03-29 2007-10-04 Euro-Celtique S.A. Benzenesulfonamide compounds and their use
WO2007118854A1 (en) 2006-04-13 2007-10-25 Euro-Celtique S.A. Benzenesulfonamide compounds and the use thereof
WO2007118853A1 (en) 2006-04-13 2007-10-25 Euro-Celtique S.A. Benzenesulfonamide compounds and their use as blockers of calcium channels
US7629346B2 (en) 2006-06-19 2009-12-08 Hoffmann-La Roche Inc. Pyrazinecarboxamide derivatives as CB1 antagonists
WO2008038143A2 (en) * 2006-06-22 2008-04-03 Medichem, S.A. Novel solid forms of rimonabant and synthetic processes for their preparation
EP2057144A4 (en) * 2006-09-01 2010-06-02 Hetero Drugs Ltd NEW POLYMORPHIC FROM RIMONABANT
US7781593B2 (en) 2006-09-14 2010-08-24 Hoffmann-La Roche Inc. 5-phenyl-nicotinamide derivatives
KR20090069318A (ko) * 2006-09-25 2009-06-30 베링거 인겔하임 인터내셔날 게엠베하 Cb2 수용체를 조절하는 화합물
DE102007002260A1 (de) 2007-01-16 2008-07-31 Sanofi-Aventis Verwendung von substituierten Pyranonsäurederivaten zur Herstellung von Medikamenten zur Behandlung des Metabolischen Syndroms
EP1953144A1 (en) * 2007-01-30 2008-08-06 Sandoz AG Novel polymorphic forms of N-piperidino-5-(4-chlorophenyl)-1-(2, 4-dichlorphenyl)-4-methyl-3-pyrazolecarboxamide
WO2008124118A1 (en) 2007-04-09 2008-10-16 Purdue Pharma L.P. Benzenesulfonyl compounds and the use therof
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Also Published As

Publication number Publication date
EA200300441A1 (ru) 2003-08-28
AU9393601A (en) 2002-04-15
IL155236A0 (en) 2003-11-23
HUP0302044A2 (hu) 2003-11-28
EP1328269B2 (fr) 2008-07-30
JP4221221B2 (ja) 2009-02-12
MXPA03002845A (es) 2004-09-10
NZ524904A (en) 2004-11-26
ES2217191T5 (es) 2009-02-16
DK1328269T4 (da) 2008-11-24
ES2217191T3 (es) 2004-11-01
FR2814678A1 (fr) 2002-04-05
DE60103556T2 (de) 2005-06-30
ZA200303015B (en) 2004-02-26
PL362833A1 (en) 2004-11-02
SI1328269T2 (sl) 2008-12-31
DK1328269T5 (da) 2009-03-16
HRP20030249A2 (en) 2005-02-28
EA005924B1 (ru) 2005-08-25
CN100409845C (zh) 2008-08-13
AU2001293936B2 (en) 2007-01-25
NO20031521D0 (no) 2003-04-03
SI1328269T1 (en) 2004-10-31
CA2424934A1 (fr) 2002-04-11
EE200300121A (et) 2005-04-15
HUP0302044A3 (en) 2005-05-30
WO2002028346A3 (fr) 2002-08-29
DK1328269T3 (da) 2004-09-20
BR0114410A (pt) 2004-02-17
NO20031521L (no) 2003-04-24
PT1328269E (pt) 2004-08-31
DE60103556T3 (de) 2009-04-09
CN1473040A (zh) 2004-02-04
FR2814678B1 (fr) 2002-12-20
KR20030036885A (ko) 2003-05-09
EP1328269A2 (fr) 2003-07-23
ATE267595T1 (de) 2004-06-15
BG107739A (bg) 2004-01-30
SK4032003A3 (en) 2003-09-11
DE60103556D1 (de) 2004-07-01
EP1328269B1 (fr) 2004-05-26
JP2004512279A (ja) 2004-04-22
WO2002028346A2 (fr) 2002-04-11
TR200401264T4 (tr) 2004-07-21

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