ATE201399T1 - 3-pyrazelcarboxamidderivate mit cannabinoid- rezeptor-affinität - Google Patents

3-pyrazelcarboxamidderivate mit cannabinoid- rezeptor-affinität

Info

Publication number
ATE201399T1
ATE201399T1 AT94402890T AT94402890T ATE201399T1 AT E201399 T1 ATE201399 T1 AT E201399T1 AT 94402890 T AT94402890 T AT 94402890T AT 94402890 T AT94402890 T AT 94402890T AT E201399 T1 ATE201399 T1 AT E201399T1
Authority
AT
Austria
Prior art keywords
alkyl
derivatives
hydrogen
nr5r6
heterocyclic radical
Prior art date
Application number
AT94402890T
Other languages
English (en)
Inventor
Francis Barth
Pierre Casellas
Christian Congy
Serge Martinez
Murielle Rinaldi
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Application granted granted Critical
Publication of ATE201399T1 publication Critical patent/ATE201399T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Saccharide Compounds (AREA)
AT94402890T 1993-12-17 1994-12-15 3-pyrazelcarboxamidderivate mit cannabinoid- rezeptor-affinität ATE201399T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9315221A FR2714057B1 (fr) 1993-12-17 1993-12-17 Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant.

Publications (1)

Publication Number Publication Date
ATE201399T1 true ATE201399T1 (de) 2001-06-15

Family

ID=9454059

Family Applications (1)

Application Number Title Priority Date Filing Date
AT94402890T ATE201399T1 (de) 1993-12-17 1994-12-15 3-pyrazelcarboxamidderivate mit cannabinoid- rezeptor-affinität

Country Status (11)

Country Link
US (1) US5462960A (de)
EP (1) EP0658546B1 (de)
JP (1) JP3825062B2 (de)
AT (1) ATE201399T1 (de)
DE (1) DE69427269T2 (de)
DK (1) DK0658546T3 (de)
ES (1) ES2159549T3 (de)
FR (1) FR2714057B1 (de)
GR (1) GR3036378T3 (de)
PT (1) PT658546E (de)
SI (1) SI0658546T1 (de)

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* Cited by examiner, † Cited by third party
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DK0658546T3 (da) 2001-09-10
DE69427269D1 (de) 2001-06-28
JPH07324076A (ja) 1995-12-12
EP0658546B1 (de) 2001-05-23
FR2714057B1 (fr) 1996-03-08
FR2714057A1 (fr) 1995-06-23
GR3036378T3 (en) 2001-11-30
DE69427269T2 (de) 2002-03-14
SI0658546T1 (en) 2001-10-31
JP3825062B2 (ja) 2006-09-20
US5462960A (en) 1995-10-31
PT658546E (pt) 2001-11-30
EP0658546A1 (de) 1995-06-21
ES2159549T3 (es) 2001-10-16

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