DE69427269T2 - 3-Pyrazelcarboxamidderivate mit Cannabinoid-Rezeptor-Affinität - Google Patents

3-Pyrazelcarboxamidderivate mit Cannabinoid-Rezeptor-Affinität

Info

Publication number
DE69427269T2
DE69427269T2 DE69427269T DE69427269T DE69427269T2 DE 69427269 T2 DE69427269 T2 DE 69427269T2 DE 69427269 T DE69427269 T DE 69427269T DE 69427269 T DE69427269 T DE 69427269T DE 69427269 T2 DE69427269 T2 DE 69427269T2
Authority
DE
Germany
Prior art keywords
alkyl
derivatives
hydrogen
nr5r6
heterocyclic radical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69427269T
Other languages
English (en)
Other versions
DE69427269D1 (de
Inventor
Francis Barth
Pierre Casellas
Christian Congy
Serge Martinez
Murielle Rinaldi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo SA filed Critical Sanofi Synthelabo SA
Publication of DE69427269D1 publication Critical patent/DE69427269D1/de
Application granted granted Critical
Publication of DE69427269T2 publication Critical patent/DE69427269T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
DE69427269T 1993-12-17 1994-12-15 3-Pyrazelcarboxamidderivate mit Cannabinoid-Rezeptor-Affinität Expired - Lifetime DE69427269T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9315221A FR2714057B1 (fr) 1993-12-17 1993-12-17 Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant.

Publications (2)

Publication Number Publication Date
DE69427269D1 DE69427269D1 (de) 2001-06-28
DE69427269T2 true DE69427269T2 (de) 2002-03-14

Family

ID=9454059

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69427269T Expired - Lifetime DE69427269T2 (de) 1993-12-17 1994-12-15 3-Pyrazelcarboxamidderivate mit Cannabinoid-Rezeptor-Affinität

Country Status (11)

Country Link
US (1) US5462960A (de)
EP (1) EP0658546B1 (de)
JP (1) JP3825062B2 (de)
AT (1) ATE201399T1 (de)
DE (1) DE69427269T2 (de)
DK (1) DK0658546T3 (de)
ES (1) ES2159549T3 (de)
FR (1) FR2714057B1 (de)
GR (1) GR3036378T3 (de)
PT (1) PT658546E (de)
SI (1) SI0658546T1 (de)

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* Cited by examiner, † Cited by third party
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EP0658546A1 (de) 1995-06-21
JPH07324076A (ja) 1995-12-12
PT658546E (pt) 2001-11-30
DK0658546T3 (da) 2001-09-10
SI0658546T1 (en) 2001-10-31
FR2714057B1 (fr) 1996-03-08
EP0658546B1 (de) 2001-05-23
FR2714057A1 (fr) 1995-06-23
US5462960A (en) 1995-10-31
ES2159549T3 (es) 2001-10-16
GR3036378T3 (en) 2001-11-30
ATE201399T1 (de) 2001-06-15
JP3825062B2 (ja) 2006-09-20
DE69427269D1 (de) 2001-06-28

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