AR095276A1 - Péptidos para el rejuvenecimiento de la piel y métodos para utilizarlos - Google Patents

Péptidos para el rejuvenecimiento de la piel y métodos para utilizarlos

Info

Publication number
AR095276A1
AR095276A1 ARP140100889A ARP140100889A AR095276A1 AR 095276 A1 AR095276 A1 AR 095276A1 AR P140100889 A ARP140100889 A AR P140100889A AR P140100889 A ARP140100889 A AR P140100889A AR 095276 A1 AR095276 A1 AR 095276A1
Authority
AR
Argentina
Prior art keywords
collagen
composition
compositions
carnosine
acid derivative
Prior art date
Application number
ARP140100889A
Other languages
English (en)
Inventor
Dreher Frank
Original Assignee
Neocutis S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neocutis S A filed Critical Neocutis S A
Publication of AR095276A1 publication Critical patent/AR095276A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/4172Imidazole-alkanecarboxylic acids, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05Dipeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06Tripeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/07Tetrapeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/494Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
    • A61K8/4946Imidazoles or their condensed derivatives, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/64Proteins; Peptides; Derivatives or degradation products thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/18Antioxidants, e.g. antiradicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/08Anti-ageing preparations
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Birds (AREA)
  • Gerontology & Geriatric Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cosmetics (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Composiciones para estimular la formación de uno o más componentes de matriz extracelular que contienen un derivado lipoaminoácido del dipéptido carnosina. Composiciones que contienen N-Octanoil carnosina en combinación con los tripéptidos y/o tetrapéptidos seleccionados así como también, composiciones farmacéuticas y/o cosméticas que contienen dichas composiciones. Métodos para utilizar las composiciones y composiciones de la presente para tratar, aliviar y/o mejorar un síntoma, condición, trastorno o enfermedad de la piel o mucosa donde el síntoma, condición, trastorno o enfermedad está asociado con cambios en los componentes de la matriz extracelular. Reivindicación 2: La composición de la reivindicación 1, caracterizada porque el derivado lipoaminoácido del dipéptido carnosina es N-Octanoil Carnosina. Reivindicación 3: La composición de la reivindicación 2, caracterizada porque la composición además comprende uno o más vehículos o excipientes adecuados para la administración tópica o subcutánea. Reivindicación 4: La composición de la reivindicación 3, caracterizada porque el, uno o más componentes de matriz extracelular se seleccionan del grupo formado por colágeno I, colágeno III, colágeno V, colágeno VI, colágeno VII, colágeno XVI, elastina, laminina, ácido hialurónico, fibrilina, sulfato de heparán proteoglicano 2, y combinaciones de los mismos. Reivindicación 9: La composición de la reivindicación 8, caracterizada porque la composición comprende Octanoil Carnosina, el derivado lipoaminoácido del tripéptido GHK (N-Palmitoil-GHK), y el tetrapéptido GEKG (Nº ID DE SEC: 1).
ARP140100889A 2013-03-13 2014-03-12 Péptidos para el rejuvenecimiento de la piel y métodos para utilizarlos AR095276A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361779601P 2013-03-13 2013-03-13

Publications (1)

Publication Number Publication Date
AR095276A1 true AR095276A1 (es) 2015-09-30

Family

ID=51263427

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140100889A AR095276A1 (es) 2013-03-13 2014-03-12 Péptidos para el rejuvenecimiento de la piel y métodos para utilizarlos

Country Status (14)

Country Link
US (3) US9375398B2 (es)
EP (1) EP2970382B1 (es)
JP (1) JP6326601B2 (es)
KR (1) KR102276326B1 (es)
CN (1) CN105189531B (es)
AR (1) AR095276A1 (es)
AU (1) AU2014229557B2 (es)
CA (1) CA2902938C (es)
HK (1) HK1212363A1 (es)
MX (1) MX360649B (es)
RU (1) RU2666533C2 (es)
SG (1) SG11201506069RA (es)
TW (1) TWI652066B (es)
WO (1) WO2014140890A2 (es)

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