AR026605A1 - Un derivado de 6-mercapto-ciclodextrina, su uso, una composicion farmaceutica que lo comprende, un kit para proporcionar bloqueo neuromuscular y sureversion, y un metodo para la reversion del bloqueo neuromuscular inducido por farmacos - Google Patents
Un derivado de 6-mercapto-ciclodextrina, su uso, una composicion farmaceutica que lo comprende, un kit para proporcionar bloqueo neuromuscular y sureversion, y un metodo para la reversion del bloqueo neuromuscular inducido por farmacosInfo
- Publication number
- AR026605A1 AR026605A1 ARP000106216A ARP000106216A AR026605A1 AR 026605 A1 AR026605 A1 AR 026605A1 AR P000106216 A ARP000106216 A AR P000106216A AR P000106216 A ARP000106216 A AR P000106216A AR 026605 A1 AR026605 A1 AR 026605A1
- Authority
- AR
- Argentina
- Prior art keywords
- neuromuscular
- mercapto
- derivative
- sureversion
- pharmacos
- Prior art date
Links
- 206010029315 Neuromuscular blockade Diseases 0.000 title abstract 2
- 229920000858 Cyclodextrin Polymers 0.000 title 1
- 230000002232 neuromuscular Effects 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 1
- 125000003161 (C1-C6) alkylene group Chemical group 0.000 abstract 1
- -1 carboxyphenyl Chemical group 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000000896 monocarboxylic acid group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000004299 tetrazol-5-yl group Chemical group [H]N1N=NC(*)=N1 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08B—POLYSACCHARIDES; DERIVATIVES THEREOF
- C08B37/00—Preparation of polysaccharides not provided for in groups C08B1/00 - C08B35/00; Derivatives thereof
- C08B37/0006—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid
- C08B37/0009—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid alpha-D-Glucans, e.g. polydextrose, alternan, glycogen; (alpha-1,4)(alpha-1,6)-D-Glucans; (alpha-1,3)(alpha-1,4)-D-Glucans, e.g. isolichenan or nigeran; (alpha-1,4)-D-Glucans; (alpha-1,3)-D-Glucans, e.g. pseudonigeran; Derivatives thereof
- C08B37/0012—Cyclodextrin [CD], e.g. cycle with 6 units (alpha), with 7 units (beta) and with 8 units (gamma), large-ring cyclodextrin or cycloamylose with 9 units or more; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
- A61K31/716—Glucans
- A61K31/724—Cyclodextrins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Polymers & Plastics (AREA)
- Biochemistry (AREA)
- Materials Engineering (AREA)
- Neurology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP99309558 | 1999-11-29 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR026605A1 true AR026605A1 (es) | 2003-02-19 |
Family
ID=8241767
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP000106216A AR026605A1 (es) | 1999-11-29 | 2000-11-27 | Un derivado de 6-mercapto-ciclodextrina, su uso, una composicion farmaceutica que lo comprende, un kit para proporcionar bloqueo neuromuscular y sureversion, y un metodo para la reversion del bloqueo neuromuscular inducido por farmacos |
Country Status (33)
Country | Link |
---|---|
US (3) | USRE44733E1 (OSRAM) |
EP (1) | EP1259550B1 (OSRAM) |
JP (2) | JP3880041B2 (OSRAM) |
KR (1) | KR100716524B1 (OSRAM) |
CN (1) | CN1188428C (OSRAM) |
AR (1) | AR026605A1 (OSRAM) |
AT (1) | ATE288450T1 (OSRAM) |
AU (1) | AU776536B2 (OSRAM) |
BE (1) | BE2008C047I2 (OSRAM) |
BR (1) | BRPI0015947B8 (OSRAM) |
CA (1) | CA2390463C (OSRAM) |
CO (1) | CO5251450A1 (OSRAM) |
CY (1) | CY2008018I1 (OSRAM) |
CZ (1) | CZ298206B6 (OSRAM) |
DE (2) | DE122008000068I2 (OSRAM) |
DK (1) | DK1259550T3 (OSRAM) |
ES (1) | ES2237496T3 (OSRAM) |
FR (1) | FR08C0052I2 (OSRAM) |
HU (1) | HU227451B1 (OSRAM) |
IL (1) | IL149423A0 (OSRAM) |
LU (1) | LU91501I2 (OSRAM) |
MX (1) | MXPA02004940A (OSRAM) |
NL (1) | NL300356I2 (OSRAM) |
NO (2) | NO328790B1 (OSRAM) |
NZ (1) | NZ518752A (OSRAM) |
PE (1) | PE20010902A1 (OSRAM) |
PL (1) | PL203012B1 (OSRAM) |
PT (1) | PT1259550E (OSRAM) |
RU (1) | RU2260013C2 (OSRAM) |
SK (1) | SK286282B6 (OSRAM) |
TW (1) | TWI242015B (OSRAM) |
WO (1) | WO2001040316A1 (OSRAM) |
ZA (1) | ZA200203538B (OSRAM) |
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US7737132B2 (en) | 2005-01-28 | 2010-06-15 | Pinnacle Pharmaceuticals | β-cyclodextrin derivatives as antibacterial agents |
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US5180716A (en) * | 1990-08-01 | 1993-01-19 | The Regents Of The University Of California | Cyclodextrin complexes for neuraxial administration of drugs |
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TWI242015B (en) | 1999-11-29 | 2005-10-21 | Akzo Nobel Nv | 6-mercapto-cyclodextrin derivatives: reversal agents for drug-induced neuromuscular block |
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WO2002064635A1 (en) | 2001-02-14 | 2002-08-22 | Akzo Nobel N.V. | 2-alkylated-cyclodextrin derivatives: reversal agents for drug-induced neuromuscular block |
TW200402417A (en) | 2002-06-21 | 2004-02-16 | Akzo Nobel Nv | 1-[(Indol-3-yl)carbonyl]piperazine derivatives |
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