ZA947119B - Androstenones - Google Patents

Androstenones

Info

Publication number
ZA947119B
ZA947119B ZA947119A ZA947119A ZA947119B ZA 947119 B ZA947119 B ZA 947119B ZA 947119 A ZA947119 A ZA 947119A ZA 947119 A ZA947119 A ZA 947119A ZA 947119 B ZA947119 B ZA 947119B
Authority
ZA
South Africa
Prior art keywords
androstenones
Prior art date
Application number
ZA947119A
Other languages
English (en)
Inventor
Kenneth William Batchelor
Stephen Vernon Frye
Original Assignee
Glaxo Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22407744&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA947119(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Inc filed Critical Glaxo Inc
Publication of ZA947119B publication Critical patent/ZA947119B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/70—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/82—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/14—Benz[f]indenes; Hydrogenated benz[f]indenes
ZA947119A 1993-09-17 1994-09-15 Androstenones ZA947119B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12328093A 1993-09-17 1993-09-17

Publications (1)

Publication Number Publication Date
ZA947119B true ZA947119B (en) 1995-05-26

Family

ID=22407744

Family Applications (2)

Application Number Title Priority Date Filing Date
ZA947118A ZA947118B (en) 1993-09-17 1994-09-15 Androstenone derivative
ZA947119A ZA947119B (en) 1993-09-17 1994-09-15 Androstenones

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ZA947118A ZA947118B (en) 1993-09-17 1994-09-15 Androstenone derivative

Country Status (41)

Country Link
US (2) US5565467A (no)
EP (1) EP0719278B1 (no)
JP (1) JP2904310B2 (no)
KR (1) KR100364953B1 (no)
CN (1) CN1057771C (no)
AP (1) AP494A (no)
AT (1) ATE162199T1 (no)
AU (1) AU690925B2 (no)
BG (1) BG62363B1 (no)
BR (1) BR1100329A (no)
CA (2) CA2170047C (no)
CY (2) CY2219B1 (no)
CZ (1) CZ286069B6 (no)
DE (2) DE10399022I2 (no)
DK (1) DK0719278T3 (no)
EE (1) EE03241B1 (no)
ES (1) ES2113127T3 (no)
FI (1) FI115216B (no)
GR (1) GR3026144T3 (no)
HK (1) HK1004334A1 (no)
HR (1) HRP940563B1 (no)
HU (1) HU220060B (no)
IL (1) IL110978A (no)
IS (1) IS1713B (no)
LU (1) LU91027I2 (no)
MY (1) MY119778A (no)
NL (1) NL300122I2 (no)
NO (2) NO306117B1 (no)
NZ (1) NZ274642A (no)
OA (1) OA10575A (no)
PE (1) PE15095A1 (no)
PL (1) PL180002B1 (no)
RO (1) RO117455B1 (no)
RU (1) RU2140926C1 (no)
SA (1) SA94150231B1 (no)
SG (1) SG52650A1 (no)
SI (1) SI0719278T1 (no)
SK (1) SK281869B6 (no)
TW (1) TW369521B (no)
WO (1) WO1995007927A1 (no)
ZA (2) ZA947118B (no)

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US5547957A (en) * 1993-10-15 1996-08-20 Merck & Co., Inc. Method of treating androgenic alopecia with 5-α reductase inhibitors
ATE175420T1 (de) * 1993-10-21 1999-01-15 Merck & Co Inc 16-substituierte-4-aza-androstan-5-alpha- reduktase-isozym-i-inhibitoren
US5817818A (en) * 1994-09-16 1998-10-06 Glaxo Wellcome Inc. Androstenones
USRE39056E1 (en) * 1995-09-15 2006-04-04 Merck & Co, Inc. 4-Azasteroids for treatment of hyperandrogenic conditions
US5872126A (en) * 1996-09-06 1999-02-16 Merck & Co., Inc. Methods and compositions for treating preterm labor
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