DE69407978D1 - Androstenderivate - Google Patents

Androstenderivate

Info

Publication number
DE69407978D1
DE69407978D1 DE69407978A DE69407978A DE69407978D1 DE 69407978 D1 DE69407978 D1 DE 69407978D1 DE 69407978 A DE69407978 A DE 69407978A DE 69407978 A DE69407978 A DE 69407978A DE 69407978 D1 DE69407978 D1 DE 69407978D1
Authority
DE
Germany
Prior art keywords
androstene
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69407978A
Other languages
English (en)
Other versions
DE69407978T2 (de
Inventor
Kenneth W Batchelor
Stephen V Frye
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Wellcome Inc
Original Assignee
Glaxo Wellcome Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
Priority to US12328093A priority Critical
Application filed by Glaxo Wellcome Inc filed Critical Glaxo Wellcome Inc
Priority to PCT/US1994/010530 priority patent/WO1995007927A1/en
Application granted granted Critical
Publication of DE69407978D1 publication Critical patent/DE69407978D1/de
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22407744&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE69407978(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Anticipated expiration legal-status Critical
Application status is Expired - Lifetime legal-status Critical

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J3/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/70Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/82Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J73/00Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/02Ortho- or ortho- and peri-condensed systems
    • C07C2603/04Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/14Benz[f]indenes; Hydrogenated benz[f]indenes
DE69407978A 1993-09-17 1994-09-16 Androstenderivate Expired - Lifetime DE69407978D1 (de)

Priority Applications (2)

Application Number Priority Date Filing Date Title
US12328093A true 1993-09-17 1993-09-17
PCT/US1994/010530 WO1995007927A1 (en) 1993-09-17 1994-09-16 Androstenone derivative

Publications (1)

Publication Number Publication Date
DE69407978D1 true DE69407978D1 (de) 1998-02-19

Family

ID=22407744

Family Applications (3)

Application Number Title Priority Date Filing Date
DE10399022C Active DE10399022I2 (de) 1993-09-17 1994-09-16 Androstenderivate
DE69407978A Expired - Lifetime DE69407978D1 (de) 1993-09-17 1994-09-16 Androstenderivate
DE69407978T Expired - Lifetime DE69407978T2 (de) 1993-09-17 1994-09-16 Androstenderivate

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE10399022C Active DE10399022I2 (de) 1993-09-17 1994-09-16 Androstenderivate

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE69407978T Expired - Lifetime DE69407978T2 (de) 1993-09-17 1994-09-16 Androstenderivate

Country Status (41)

Country Link
US (2) US5565467A (de)
EP (1) EP0719278B1 (de)
JP (1) JP2904310B2 (de)
KR (1) KR100364953B1 (de)
CN (1) CN1057771C (de)
AP (1) AP494A (de)
AT (1) AT162199T (de)
AU (1) AU690925B2 (de)
BG (1) BG62363B1 (de)
BR (1) BR1100329A (de)
CA (2) CA2170047C (de)
CY (1) CY2219B1 (de)
CZ (1) CZ286069B6 (de)
DE (3) DE10399022I2 (de)
DK (1) DK0719278T3 (de)
EE (1) EE03241B1 (de)
ES (1) ES2113127T3 (de)
FI (1) FI115216B (de)
GR (1) GR3026144T3 (de)
HK (1) HK1004334A1 (de)
HR (1) HRP940563B1 (de)
HU (1) HU220060B (de)
IL (1) IL110978A (de)
IS (1) IS1713B (de)
LU (1) LU91027I2 (de)
MY (1) MY119778A (de)
NL (1) NL300122I2 (de)
NO (2) NO306117B1 (de)
NZ (1) NZ274642A (de)
OA (1) OA10575A (de)
PE (1) PE15095A1 (de)
PL (1) PL180002B1 (de)
RO (1) RO117455B1 (de)
RU (1) RU2140926C1 (de)
SA (1) SA312B1 (de)
SG (1) SG52650A1 (de)
SI (1) SI0719278T1 (de)
SK (1) SK281869B6 (de)
TW (1) TW369521B (de)
WO (1) WO1995007927A1 (de)
ZA (2) ZA9407118B (de)

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US5872126A (en) * 1996-09-06 1999-02-16 Merck & Co., Inc. Methods and compositions for treating preterm labor
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RU2000125533A (ru) * 1998-03-11 2002-10-20 Эндорешерш, Инк. (Ca) Ингибиторы 17-бета-гидроксистероиддегидрогеназ 5 и 3 типа и способы их применения
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EA008377B1 (ru) * 2002-04-24 2007-04-27 Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг Фармацевтическая комбинация для лечения доброкачественной гиперплазии простаты или для долговременной профилактики острой ишурии
AU2003223754B2 (en) * 2002-04-30 2007-08-16 Merck Sharp & Dohme Corp. 4-azasteroid derivatives as androgen receptor modulators
US7326717B2 (en) * 2003-05-06 2008-02-05 L'oreal Pyrimidine n-oxide compounds for stimulating the growth of keratin fibers and/or reducing loss thereof
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HU220060B (hu) 2001-10-28
CN1057771C (zh) 2000-10-25
CZ74596A3 (en) 1996-09-11
FI115216B (fi) 2005-03-31
EE03241B1 (et) 1999-12-15
HUT73850A (en) 1996-09-30
PE15095A1 (es) 1995-06-04
FI961231A0 (fi) 1996-03-15
CA2462061A1 (en) 1995-03-23
PL180002B1 (en) 2000-11-30
ZA9407119B (en) 1995-05-26
NO306117B1 (no) 1999-09-20
WO1995007927A1 (en) 1995-03-23
NL300122I2 (nl) 2003-09-01
CZ286069B6 (cs) 2000-01-12
NL300122I1 (nl) 2003-06-02
LU91027I2 (fr) 2004-04-28
IS4205A (is) 1995-03-18
AP494A (en) 1996-05-15
JP2904310B2 (ja) 1999-06-14
US5846976A (en) 1998-12-08
HU9600656D0 (en) 1996-05-28
MY119778A (en) 2005-07-29
IL110978A (en) 1999-01-26
DK719278T3 (de)
AU690925B2 (en) 1998-05-07
US5565467A (en) 1996-10-15
BG100410A (bg) 1996-09-30
CN1131424A (zh) 1996-09-18
HRP940563A2 (en) 1997-02-28
HK1004334A1 (en) 1998-11-20
EP0719278A1 (de) 1996-07-03
DE69407978T2 (de) 1998-05-07
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CA2170047A1 (en) 1995-03-23
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RO117455B1 (ro) 2002-03-29
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GR3026144T3 (en) 1998-05-29
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NZ274642A (en) 1997-11-24
RU2140926C1 (ru) 1999-11-10
DE10399022I2 (de) 2012-09-13
BR1100329A (pt) 2000-06-13
FI115216B1 (de)
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