DE69407978D1 - Androstenderivate - Google Patents

Androstenderivate

Info

Publication number
DE69407978D1
DE69407978D1 DE69407978T DE69407978T DE69407978D1 DE 69407978 D1 DE69407978 D1 DE 69407978D1 DE 69407978 T DE69407978 T DE 69407978T DE 69407978 T DE69407978 T DE 69407978T DE 69407978 D1 DE69407978 D1 DE 69407978D1
Authority
DE
Germany
Prior art keywords
androst
derivatives
androst derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69407978T
Other languages
English (en)
Other versions
DE69407978T2 (de
Inventor
Kenneth W Batchelor
Stephen V Frye
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
Glaxo Wellcome Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22407744&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE69407978(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Wellcome Inc filed Critical Glaxo Wellcome Inc
Publication of DE69407978D1 publication Critical patent/DE69407978D1/de
Application granted granted Critical
Publication of DE69407978T2 publication Critical patent/DE69407978T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/70—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/82—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/14—Benz[f]indenes; Hydrogenated benz[f]indenes
DE69407978T 1993-09-17 1994-09-16 Androstenderivate Expired - Lifetime DE69407978T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12328093A 1993-09-17 1993-09-17
PCT/US1994/010530 WO1995007927A1 (en) 1993-09-17 1994-09-16 Androstenone derivative

Publications (2)

Publication Number Publication Date
DE69407978D1 true DE69407978D1 (de) 1998-02-19
DE69407978T2 DE69407978T2 (de) 1998-05-07

Family

ID=22407744

Family Applications (2)

Application Number Title Priority Date Filing Date
DE69407978T Expired - Lifetime DE69407978T2 (de) 1993-09-17 1994-09-16 Androstenderivate
DE10399022C Active DE10399022I2 (de) 1993-09-17 1994-09-16 Androstenderivate

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE10399022C Active DE10399022I2 (de) 1993-09-17 1994-09-16 Androstenderivate

Country Status (41)

Country Link
US (2) US5565467A (de)
EP (1) EP0719278B1 (de)
JP (1) JP2904310B2 (de)
KR (1) KR100364953B1 (de)
CN (1) CN1057771C (de)
AP (1) AP494A (de)
AT (1) ATE162199T1 (de)
AU (1) AU690925B2 (de)
BG (1) BG62363B1 (de)
BR (1) BR1100329A (de)
CA (2) CA2170047C (de)
CY (2) CY2219B1 (de)
CZ (1) CZ286069B6 (de)
DE (2) DE69407978T2 (de)
DK (1) DK0719278T3 (de)
EE (1) EE03241B1 (de)
ES (1) ES2113127T3 (de)
FI (1) FI115216B (de)
GR (1) GR3026144T3 (de)
HK (1) HK1004334A1 (de)
HR (1) HRP940563B1 (de)
HU (1) HU220060B (de)
IL (1) IL110978A (de)
IS (1) IS1713B (de)
LU (1) LU91027I2 (de)
MY (1) MY119778A (de)
NL (1) NL300122I2 (de)
NO (2) NO306117B1 (de)
NZ (1) NZ274642A (de)
OA (1) OA10575A (de)
PE (1) PE15095A1 (de)
PL (1) PL180002B1 (de)
RO (1) RO117455B1 (de)
RU (1) RU2140926C1 (de)
SA (1) SA94150231B1 (de)
SG (1) SG52650A1 (de)
SI (1) SI0719278T1 (de)
SK (1) SK281869B6 (de)
TW (1) TW369521B (de)
WO (1) WO1995007927A1 (de)
ZA (2) ZA947118B (de)

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US5872126A (en) * 1996-09-06 1999-02-16 Merck & Co., Inc. Methods and compositions for treating preterm labor
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US5998427A (en) * 1998-05-14 1999-12-07 Glaxo Wellcome Inc. Androstenones
WO1999066915A2 (en) * 1998-06-23 1999-12-29 Southern Illinois University At Carbondale Therapeutic applications of estrogenic carboxylic acids
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EP1743656A3 (de) * 2002-04-24 2007-03-07 Boehringer Ingelheim Pharma GmbH & Co. KG pharmazeutische Kombination zur Behandlung von benigner Prostatahyperplasie oder zur Langzeitvorbeugung von akuter Harnretention
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