ZA914423B - Cyclic amide derivatives - Google Patents

Cyclic amide derivatives

Info

Publication number
ZA914423B
ZA914423B ZA914423A ZA914423A ZA914423B ZA 914423 B ZA914423 B ZA 914423B ZA 914423 A ZA914423 A ZA 914423A ZA 914423 A ZA914423 A ZA 914423A ZA 914423 B ZA914423 B ZA 914423B
Authority
ZA
South Africa
Prior art keywords
cyclic amide
aryl
integer
amide compound
substituted
Prior art date
Application number
ZA914423A
Other languages
English (en)
Inventor
Hachiro Sugimoto
Sugimoto Hachiro
Masahiro Yonaga
Yonaga Masahiro
Norio Karibe
Karibe Norio
Youichi Limura
Limura Youichi
Satoshi Nagato
Nagato Satoshi
Atsushi Sasaki
Sasaki Atsushi
Yoshiharu Yamanishi
Yamanishi Yoshiharu
Hiroo Ogura
Ogura Hiroo
Takashi Kosasa
Kosasa Takashi
Kumi Uchikoshi
Uchikoshi Kumi
Kiyomi Yamatsu
Yamatsu Kiyomi
Original Assignee
Esai Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Esai Co Ltd filed Critical Esai Co Ltd
Publication of ZA914423B publication Critical patent/ZA914423B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrrole Compounds (AREA)
ZA914423A 1990-06-15 1991-06-10 Cyclic amide derivatives ZA914423B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP15713490 1990-06-15

Publications (1)

Publication Number Publication Date
ZA914423B true ZA914423B (en) 1992-03-25

Family

ID=15642948

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA914423A ZA914423B (en) 1990-06-15 1991-06-10 Cyclic amide derivatives

Country Status (17)

Country Link
US (6) US5292735A (fr)
EP (3) EP0468187B1 (fr)
JP (2) JP2807577B2 (fr)
KR (1) KR940004391B1 (fr)
CN (1) CN1045206C (fr)
AT (3) ATE170517T1 (fr)
AU (2) AU653938B2 (fr)
CA (2) CA2175502C (fr)
DE (3) DE69129090T2 (fr)
DK (2) DK0677516T3 (fr)
ES (2) ES2123858T3 (fr)
FI (1) FI114797B (fr)
HU (2) HU216188B (fr)
NO (1) NO180540B1 (fr)
NZ (2) NZ238534A (fr)
PT (1) PT97993B (fr)
ZA (1) ZA914423B (fr)

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NZ722077A (en) 2013-12-20 2021-12-24 Agenebio Inc Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
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WO1991006297A1 (fr) * 1989-10-27 1991-05-16 The Du Pont Merck Pharmaceutical Company (n-phthalimidoalkyle)piperidines
TW197442B (fr) * 1990-02-08 1993-01-01 Pfizer
DK37790A (da) * 1990-02-13 1991-08-14 Novo Nordisk As Indolderivater, deres fremstilling og anvendelse
FR2660657B1 (fr) * 1990-04-09 1993-05-07 Adir Nouveaux derives du 3-aminochromane, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
JP2807577B2 (ja) * 1990-06-15 1998-10-08 エーザイ株式会社 環状アミド誘導体
EP0626373B1 (fr) * 1993-05-26 1998-12-23 Sumitomo Pharmaceuticals Company, Limited Dérivés de guinazolinone

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Publication number Publication date
DE69129090T2 (de) 1998-08-06
EP0742216B1 (fr) 2001-11-21
PT97993A (pt) 1992-03-31
EP0742216A2 (fr) 1996-11-13
DE69129090D1 (de) 1998-04-23
EP0677516B1 (fr) 1998-09-02
US5504088A (en) 1996-04-02
HU211895A9 (en) 1995-12-28
US5654308A (en) 1997-08-05
HU216188B (hu) 1999-05-28
CN1057262A (zh) 1991-12-25
NO180540B1 (no) 1997-05-26
ATE170517T1 (de) 1998-09-15
PT97993B (pt) 1998-11-30
JPH0899974A (ja) 1996-04-16
AU653938B2 (en) 1994-10-20
KR920000754A (ko) 1992-01-29
DE69130120T2 (de) 1999-02-18
HUT61742A (en) 1993-03-01
CA2044515C (fr) 1997-05-20
EP0742216A3 (fr) 1997-05-28
EP0468187A2 (fr) 1992-01-29
EP0677516A1 (fr) 1995-10-18
ES2123858T3 (es) 1999-01-16
US5292735A (en) 1994-03-08
US5620976A (en) 1997-04-15
ATE209198T1 (de) 2001-12-15
US5919778A (en) 1999-07-06
KR940004391B1 (en) 1994-05-25
EP0468187B1 (fr) 1998-03-18
US5521182A (en) 1996-05-28
FI114797B (fi) 2004-12-31
ES2113355T3 (es) 1998-05-01
NO912252A (no) 1991-12-16
CN1045206C (zh) 1999-09-22
NO180540C (no) 1997-05-07
NZ238534A (en) 1995-07-26
HU911986D0 (en) 1991-12-30
AU680704B2 (en) 1997-08-07
JPH04235161A (ja) 1992-08-24
CA2175502C (fr) 2001-07-10
AU1024695A (en) 1995-03-30
JP2807577B2 (ja) 1998-10-08
NZ272015A (en) 1999-07-29
EP0468187A3 (en) 1992-04-15
DE69130120D1 (de) 1998-10-08
FI912851A (fi) 1991-12-16
DE69132827T2 (de) 2002-06-27
AU7813691A (en) 1991-12-19
DE69132827D1 (de) 2002-01-03
DK0468187T3 (da) 1999-01-11
CA2175502A1 (fr) 1991-12-16
DK0677516T3 (da) 1999-06-07
CA2044515A1 (fr) 1991-12-16
NO912252D0 (no) 1991-06-12
NO180540B (no) 1997-01-27
FI912851A0 (fi) 1991-06-13
JP3224187B2 (ja) 2001-10-29
ATE164156T1 (de) 1998-04-15

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