ZA200205090B - Selective crystallization of 3-pyridyl-1-hydroxyethylidene-1,1-bisphosphonic acid sodium as the hemipentahydrate or monohydrate. - Google Patents

Selective crystallization of 3-pyridyl-1-hydroxyethylidene-1,1-bisphosphonic acid sodium as the hemipentahydrate or monohydrate.

Info

Publication number
ZA200205090B
ZA200205090B ZA200205090A ZA200205090A ZA200205090B ZA 200205090 B ZA200205090 B ZA 200205090B ZA 200205090 A ZA200205090 A ZA 200205090A ZA 200205090 A ZA200205090 A ZA 200205090A ZA 200205090 B ZA200205090 B ZA 200205090B
Authority
ZA
South Africa
Prior art keywords
hemipentahydrate
hydroxyethylidene
monohydrate
pyridyl
acid sodium
Prior art date
Application number
ZA200205090A
Other languages
English (en)
Inventor
Cazer Fredrick Dana
Perry Gregory Eugene
Billings Dennis Michael
Redman-Furey Nancy Lee
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22656866&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200205090(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of ZA200205090B publication Critical patent/ZA200205090B/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/58—Pyridine rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
ZA200205090A 2000-02-01 2002-06-25 Selective crystallization of 3-pyridyl-1-hydroxyethylidene-1,1-bisphosphonic acid sodium as the hemipentahydrate or monohydrate. ZA200205090B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17950500P 2000-02-01 2000-02-01

Publications (1)

Publication Number Publication Date
ZA200205090B true ZA200205090B (en) 2003-04-30

Family

ID=22656866

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200205090A ZA200205090B (en) 2000-02-01 2002-06-25 Selective crystallization of 3-pyridyl-1-hydroxyethylidene-1,1-bisphosphonic acid sodium as the hemipentahydrate or monohydrate.

Country Status (33)

Country Link
US (1) US6410520B2 (xx)
EP (1) EP1252170B2 (xx)
JP (5) JP2003521532A (xx)
KR (1) KR100549038B1 (xx)
CN (1) CN1183148C (xx)
AR (1) AR030187A1 (xx)
AT (1) ATE273984T1 (xx)
AU (1) AU784307B2 (xx)
BR (1) BRPI0107921B8 (xx)
CA (1) CA2399976C (xx)
CO (1) CO5271720A1 (xx)
CZ (1) CZ303400B6 (xx)
DE (1) DE60104978T3 (xx)
DK (1) DK1252170T4 (xx)
ES (1) ES2225481T5 (xx)
HK (1) HK1051046B (xx)
HU (1) HU230494B1 (xx)
IL (2) IL150511A0 (xx)
MA (1) MA25654A1 (xx)
MX (1) MXPA02007417A (xx)
MY (1) MY119968A (xx)
NO (1) NO329923B1 (xx)
NZ (1) NZ519966A (xx)
PE (1) PE20011061A1 (xx)
PL (1) PL207589B1 (xx)
PT (1) PT1252170E (xx)
RU (1) RU2236415C2 (xx)
SA (1) SA01220066B1 (xx)
SK (1) SK287884B6 (xx)
TR (1) TR200402435T4 (xx)
TW (1) TWI310769B (xx)
WO (1) WO2001056983A2 (xx)
ZA (1) ZA200205090B (xx)

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US7687482B2 (en) * 2006-03-17 2010-03-30 The Board Of Trustees Of The University Of Illinois Bisphosphonate compounds and methods
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KR100798855B1 (ko) * 2007-02-14 2008-01-28 주식회사 엔지켐 리세드론산 나트륨 헤미펜타하이드레이트의 제조방법
KR100812528B1 (ko) * 2007-04-12 2008-03-12 보령제약 주식회사 리세드로네이트 나트륨염의 헤미펜타히드레이트의 선택적결정화방법
US20100317859A1 (en) * 2007-05-16 2010-12-16 Actavis Group Ptc Ehf Process for the Preparation of Risedronate Sodium
WO2009050731A2 (en) * 2007-06-20 2009-04-23 Alkem Laboratories Ltd Novel process for preparing risedronic acid
DE102007030370A1 (de) 2007-06-29 2009-01-02 Ratiopharm Gmbh Essigsäure-Solvate von Risedronat, Polymorph hiervon, deren Herstellung und Verwendung sowie pharmazeutische Zusammensetzung, enthaltend diese
KR100925835B1 (ko) * 2007-12-07 2009-11-06 동우신테크 주식회사 리세드로네이트 나트륨 무수물 및 수화물의 제조방법
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Also Published As

Publication number Publication date
JP2016028083A (ja) 2016-02-25
HK1051046B (zh) 2005-04-29
DK1252170T4 (da) 2014-01-20
BR0107921A (pt) 2002-10-22
RU2236415C2 (ru) 2004-09-20
IL150511A (en) 2006-12-10
KR100549038B1 (ko) 2006-02-02
CO5271720A1 (es) 2003-04-30
EP1252170A2 (en) 2002-10-30
EP1252170B1 (en) 2004-08-18
WO2001056983A3 (en) 2002-03-07
JP2012255013A (ja) 2012-12-27
CN1183148C (zh) 2005-01-05
ES2225481T3 (es) 2005-03-16
TR200402435T4 (tr) 2004-12-21
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