TR200402435T4 - 3-piridil-1-hidroksietiliden-1,1-bisfosfonik asit sodyumun hemipentahidrat veya monohidrat olarak seçici şekilde kristalleştirilmesi. - Google Patents
3-piridil-1-hidroksietiliden-1,1-bisfosfonik asit sodyumun hemipentahidrat veya monohidrat olarak seçici şekilde kristalleştirilmesi.Info
- Publication number
- TR200402435T4 TR200402435T4 TR2004/02435T TR200402435T TR200402435T4 TR 200402435 T4 TR200402435 T4 TR 200402435T4 TR 2004/02435 T TR2004/02435 T TR 2004/02435T TR 200402435 T TR200402435 T TR 200402435T TR 200402435 T4 TR200402435 T4 TR 200402435T4
- Authority
- TR
- Turkey
- Prior art keywords
- monohydrate
- hemipentahydrate
- hydroxyethylidene
- pyridyl
- acid sodium
- Prior art date
Links
- 150000004682 monohydrates Chemical class 0.000 title abstract 3
- DGAQECJNVWCQMB-PUAWFVPOSA-M Ilexoside XXIX Chemical compound C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)OS(=O)(=O)[O-])C)C)[C@@H]2[C@]1(C)O)C)C(=O)O[C@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O.[Na+] DGAQECJNVWCQMB-PUAWFVPOSA-M 0.000 title abstract 2
- 239000002253 acid Substances 0.000 title abstract 2
- 229910052708 sodium Inorganic materials 0.000 title abstract 2
- 239000011734 sodium Substances 0.000 title abstract 2
- 238000010956 selective crystallization Methods 0.000 title 1
- 238000002425 crystallisation Methods 0.000 abstract 1
- 230000008025 crystallization Effects 0.000 abstract 1
- 238000010899 nucleation Methods 0.000 abstract 1
- 230000006911 nucleation Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/58—Pyridine rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
- A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Physical Education & Sports Medicine (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Mevcut bulus,3-piridil-1-hidroksietiliden-1,1-bisfosfonik asit sodyum hemipentahidrat ve monohidrati, çekirdeklesme sicakliginin ve kristallesme hizinin kontrol edilmesini içeren hemipentahidrat veya monohidrat hazirlama yöntemlerini hidrat formlarindan birini veya her ikisini de içeren farmasötik bilesimleri tarif etmektedir.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US17950500P | 2000-02-01 | 2000-02-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200402435T4 true TR200402435T4 (tr) | 2004-12-21 |
Family
ID=22656866
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2004/02435T TR200402435T4 (tr) | 2000-02-01 | 2001-02-01 | 3-piridil-1-hidroksietiliden-1,1-bisfosfonik asit sodyumun hemipentahidrat veya monohidrat olarak seçici şekilde kristalleştirilmesi. |
Country Status (33)
Country | Link |
---|---|
US (1) | US6410520B2 (tr) |
EP (1) | EP1252170B2 (tr) |
JP (5) | JP2003521532A (tr) |
KR (1) | KR100549038B1 (tr) |
CN (1) | CN1183148C (tr) |
AR (1) | AR030187A1 (tr) |
AT (1) | ATE273984T1 (tr) |
AU (1) | AU784307B2 (tr) |
BR (1) | BRPI0107921B8 (tr) |
CA (1) | CA2399976C (tr) |
CO (1) | CO5271720A1 (tr) |
CZ (1) | CZ303400B6 (tr) |
DE (1) | DE60104978T3 (tr) |
DK (1) | DK1252170T4 (tr) |
ES (1) | ES2225481T5 (tr) |
HK (1) | HK1051046B (tr) |
HU (1) | HU230494B1 (tr) |
IL (2) | IL150511A0 (tr) |
MA (1) | MA25654A1 (tr) |
MX (1) | MXPA02007417A (tr) |
MY (1) | MY119968A (tr) |
NO (1) | NO329923B1 (tr) |
NZ (1) | NZ519966A (tr) |
PE (1) | PE20011061A1 (tr) |
PL (1) | PL207589B1 (tr) |
PT (1) | PT1252170E (tr) |
RU (1) | RU2236415C2 (tr) |
SA (1) | SA01220066B1 (tr) |
SK (1) | SK287884B6 (tr) |
TR (1) | TR200402435T4 (tr) |
TW (1) | TWI310769B (tr) |
WO (1) | WO2001056983A2 (tr) |
ZA (1) | ZA200205090B (tr) |
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CA2513543A1 (en) * | 2003-01-17 | 2004-08-05 | Teva Pharmaceutical Industries Ltd. | Risedronate sodium having a very low content of iron |
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ATE493423T1 (de) * | 2003-07-30 | 2011-01-15 | Warner Chilcott Co Llc | Verfahren zur steuerung der kristallstruktur von risedronat |
CZ298639B6 (cs) * | 2004-02-05 | 2007-12-05 | Zentiva, A. S. | Krystalická forma risedronátu monosodného |
WO2005082915A1 (en) * | 2004-02-26 | 2005-09-09 | Zentiva, A.S. | Amorphous forms of risedronate monosodium |
WO2005107714A2 (en) * | 2004-05-05 | 2005-11-17 | Alkermes Controlled Therapeutics, Inc. | Method of forming microparticles that include a bisphosphonate and a polymer |
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WO2006039721A2 (en) * | 2004-10-08 | 2006-04-13 | The Board Of Trustees Of The University Of Illinois | Bisphosphonate compounds and methods for bone resorption diseases, cancer, bone pain, immune disorders, and infectious diseases |
US8012949B2 (en) * | 2004-10-08 | 2011-09-06 | The Board Of Trustees Of The University Of Illinois | Bisphosphonate compounds and methods with enhanced potency for multiple targets including FPPS, GGPPS, and DPPS |
US7687482B2 (en) * | 2006-03-17 | 2010-03-30 | The Board Of Trustees Of The University Of Illinois | Bisphosphonate compounds and methods |
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PL199215B1 (pl) * | 2004-12-28 | 2008-08-29 | Politechnika Gdanska | Sposób wytwarzania kwasu [1-hydroksy-2-(3-pirydylo)etylidenobisfosfonowego] oraz jego soli monosodowej dwu i pół wodnej |
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EP1775302A1 (en) * | 2005-10-11 | 2007-04-18 | Sandoz A/S | Method for preparing crystalline sodium risedronate |
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JP5354858B2 (ja) * | 2006-05-09 | 2013-11-27 | 株式会社Adeka | スルホンアミド化合物の金属塩を含有するポリエステル樹脂組成物 |
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2001
- 2001-01-29 PE PE2001000096A patent/PE20011061A1/es active IP Right Grant
- 2001-01-29 US US09/771,825 patent/US6410520B2/en not_active Expired - Lifetime
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- 2001-02-01 DE DE60104978.0T patent/DE60104978T3/de not_active Expired - Lifetime
- 2001-02-01 JP JP2001556833A patent/JP2003521532A/ja active Pending
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2002
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