AU2002350942A8 - Imidazolidineacetic acid derivatives - Google Patents

Imidazolidineacetic acid derivatives

Info

Publication number
AU2002350942A8
AU2002350942A8 AU2002350942A AU2002350942A AU2002350942A8 AU 2002350942 A8 AU2002350942 A8 AU 2002350942A8 AU 2002350942 A AU2002350942 A AU 2002350942A AU 2002350942 A AU2002350942 A AU 2002350942A AU 2002350942 A8 AU2002350942 A8 AU 2002350942A8
Authority
AU
Australia
Prior art keywords
acid derivatives
imidazolidineacetic acid
imidazolidineacetic
derivatives
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002350942A
Other versions
AU2002350942A1 (en
Inventor
Michael Bryan Roe
Andre Tartar
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ferring BV
Original Assignee
Ferring BV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferring BV filed Critical Ferring BV
Publication of AU2002350942A8 publication Critical patent/AU2002350942A8/en
Publication of AU2002350942A1 publication Critical patent/AU2002350942A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
AU2002350942A 2001-12-14 2002-12-12 Imidazolidineacetic acid derivatives Abandoned AU2002350942A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0129988A GB0129988D0 (en) 2001-12-14 2001-12-14 Imidazolidineacetic acid derivatives
GB0129988.2 2001-12-14
PCT/GB2002/005631 WO2003051848A2 (en) 2001-12-14 2002-12-12 Imidazolidineacetic acid derivatives

Publications (2)

Publication Number Publication Date
AU2002350942A8 true AU2002350942A8 (en) 2003-06-30
AU2002350942A1 AU2002350942A1 (en) 2003-06-30

Family

ID=9927662

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002350942A Abandoned AU2002350942A1 (en) 2001-12-14 2002-12-12 Imidazolidineacetic acid derivatives

Country Status (3)

Country Link
AU (1) AU2002350942A1 (en)
GB (1) GB0129988D0 (en)
WO (1) WO2003051848A2 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7842707B2 (en) 2004-07-23 2010-11-30 Nuada, Llc Peptidase inhibitors
EA015169B1 (en) 2005-09-14 2011-06-30 Такеда Фармасьютикал Компани Лимитед Use of dipeptidyl peptidase inhibitors
CN102675221A (en) 2005-09-16 2012-09-19 武田药品工业株式会社 Intermediate in method for preparing pyrimidinedione derivative
WO2007112347A1 (en) 2006-03-28 2007-10-04 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US8324383B2 (en) 2006-09-13 2012-12-04 Takeda Pharmaceutical Company Limited Methods of making polymorphs of benzoate salt of 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-benzonitrile
TW200838536A (en) 2006-11-29 2008-10-01 Takeda Pharmaceutical Polymorphs of succinate salt of 2-[6-(3-amino-piperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethy]-4-fluor-benzonitrile and methods of use therefor
US8093236B2 (en) 2007-03-13 2012-01-10 Takeda Pharmaceuticals Company Limited Weekly administration of dipeptidyl peptidase inhibitors
CZ2008512A3 (en) 2008-08-26 2010-03-10 Zentiva, A. S Process for preparing extremely pure vildagliptin
CN104262227B (en) * 2014-09-16 2018-09-18 东北制药集团股份有限公司 A method of preparing (S) -1- (2- chloracetyls) pyrrolidines -2- formonitrile HCNs

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW492957B (en) * 1996-11-07 2002-07-01 Novartis Ag N-substituted 2-cyanopyrrolidnes

Also Published As

Publication number Publication date
WO2003051848A3 (en) 2003-09-18
WO2003051848A2 (en) 2003-06-26
AU2002350942A1 (en) 2003-06-30
GB0129988D0 (en) 2002-02-06

Similar Documents

Publication Publication Date Title
ZA200309522B (en) Substituted cyclohexane-1-4diamine derivatives
IL160701A0 (en) 3-substituted-4-pyrimidone derivatives
AU2002358718A1 (en) 2-heteroarylcarboxylic acid amides
SI1671949T1 (en) Substituted Pyridinylamines
IL158388A0 (en) Novel arylheteroalkylamine derivatives
AU2002358700A8 (en) Urea derivatives as vr1- antagonists
IL158461A0 (en) Novel sulfonic acid derivatives
HUP0303449A3 (en) Substituted benzofuran-2-carboxamides derivatives
HK1068607A1 (en) Phenylalkyloxy-phenyl derivatives
AU2001280167A1 (en) Novel propenohydroxamic acid derivatives
PL362643A1 (en) Substituted fluoroalcoxyphenylsulfonylurea
HUP0303186A3 (en) 4-aminobenzopyran derivatives
HUP0401949A3 (en) 4-imidazolin-2-one derivatives
HUP0500026A3 (en) N-heteroarylnicotinamide derivatives
IL152759A0 (en) Quinolonecarboxylic acid derivatives
SI1406858T1 (en) Substituted 4-aminocyclohexanols
PL364901A1 (en) Oxalic acid derivatives
GB0129988D0 (en) Imidazolidineacetic acid derivatives
EP1364954A4 (en) Dicarba-closo-dodecarborane derivatives
PL358585A1 (en) N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
HUP0402101A3 (en) Butyric acid derivatives
ZA200402308B (en) NOVEL a-OXYGENATED OR a-THIOLATED CARBOXYLIC ACID PENETHYLAMIDE DERIVATIVES
PL364601A1 (en) Substituted benzo-nitro-heterocycles
PL357011A1 (en) Novel alpha-sulfin- and alpha-sulfonamino acid amide derivatives
GB0017435D0 (en) 3-arylsulfonyl-2-hydroxy-2-methylpropanoic acid derivatives

Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase