TWI701253B - Ａｃｃ抑制劑及彼等之用途 - Google Patents
Ａｃｃ抑制劑及彼等之用途 Download PDFInfo
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- TWI701253B TWI701253B TW107147492A TW107147492A TWI701253B TW I701253 B TWI701253 B TW I701253B TW 107147492 A TW107147492 A TW 107147492A TW 107147492 A TW107147492 A TW 107147492A TW I701253 B TWI701253 B TW I701253B
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- Prior art keywords
- compound
- nitrogen
- pharmaceutically acceptable
- independently selected
- ring
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Classifications
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- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A—HUMAN NECESSITIES
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Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161559023P | 2011-11-11 | 2011-11-11 | |
| US61/559,023 | 2011-11-11 | ||
| US201261615092P | 2012-03-23 | 2012-03-23 | |
| US61/615,092 | 2012-03-23 | ||
| US201261651878P | 2012-05-25 | 2012-05-25 | |
| US61/651,878 | 2012-05-25 | ||
| US201261675513P | 2012-07-25 | 2012-07-25 | |
| US61/675,513 | 2012-07-25 |
Publications (2)
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| US20080287465A1 (en) * | 2004-07-21 | 2008-11-20 | Athersys, Inc. | Cyclic N-Hydroxy Imides as Inhibitors of Flap Endonuclease and Uses Thereof |
| US20070208040A1 (en) * | 2006-03-02 | 2007-09-06 | Elfatih Elzein | A2a adenosine receptor antagonists |
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