BR112014011351A2 - inibidores de acc e usos dos mesmos - Google Patents

inibidores de acc e usos dos mesmos

Info

Publication number
BR112014011351A2
BR112014011351A2 BR112014011351A BR112014011351A BR112014011351A2 BR 112014011351 A2 BR112014011351 A2 BR 112014011351A2 BR 112014011351 A BR112014011351 A BR 112014011351A BR 112014011351 A BR112014011351 A BR 112014011351A BR 112014011351 A2 BR112014011351 A2 BR 112014011351A2
Authority
BR
Brazil
Prior art keywords
acc
inhibitors
acc inhibitors
compositions
methods
Prior art date
Application number
BR112014011351A
Other languages
English (en)
Other versions
BR112014011351B1 (pt
Inventor
E Masse Craig
Harriman Geraldine
Harwood James
robert greenwood Jeremy
Bhat Sathesh
Original Assignee
Nimbus Apollo Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nimbus Apollo Inc filed Critical Nimbus Apollo Inc
Priority to BR122019026836-3A priority Critical patent/BR122019026836B1/pt
Publication of BR112014011351A2 publication Critical patent/BR112014011351A2/pt
Publication of BR112014011351B1 publication Critical patent/BR112014011351B1/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Abstract

abstract the present invention provides compounds useful as inhibitors of acetyl coa carboxylase (acc), compositions thereof, and methods of using the same. 5540217v3 tradução do resumo resumo patente de invenção: "inibidores de acc e usos dos mesmos". a presente invenção proporciona compostos úteis como inibidores de carboxilase de acetil-coa (acetyl coa carboxylase - acc), composições dos mesmos e métodos de uso dos mesmos.
BR112014011351-3A 2011-11-11 2012-11-09 inibidores de acc e usos dos mesmos BR112014011351B1 (pt)

Priority Applications (1)

Application Number Priority Date Filing Date Title
BR122019026836-3A BR122019026836B1 (pt) 2011-11-11 2012-11-09 composto, e, métodos de inibição de acc em uma amostra biológica e em uma planta

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US201161559023P 2011-11-11 2011-11-11
US61/559,023 2011-11-11
US201261615092P 2012-03-23 2012-03-23
US61/615,092 2012-03-23
US201261651878P 2012-05-25 2012-05-25
US61/651,878 2012-05-25
US201261675513P 2012-07-25 2012-07-25
US61/675,513 2012-07-25
PCT/US2012/064528 WO2013071169A1 (en) 2011-11-11 2012-11-09 Acc inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
BR112014011351A2 true BR112014011351A2 (pt) 2017-06-06
BR112014011351B1 BR112014011351B1 (pt) 2021-02-17

Family

ID=48281206

Family Applications (2)

Application Number Title Priority Date Filing Date
BR112014011351-3A BR112014011351B1 (pt) 2011-11-11 2012-11-09 inibidores de acc e usos dos mesmos
BR122019026836-3A BR122019026836B1 (pt) 2011-11-11 2012-11-09 composto, e, métodos de inibição de acc em uma amostra biológica e em uma planta

Family Applications After (1)

Application Number Title Priority Date Filing Date
BR122019026836-3A BR122019026836B1 (pt) 2011-11-11 2012-11-09 composto, e, métodos de inibição de acc em uma amostra biológica e em uma planta

Country Status (26)

Country Link
US (5) US8969557B2 (pt)
EP (3) EP3628320B1 (pt)
JP (4) JP6114297B2 (pt)
KR (3) KR102172902B1 (pt)
CN (3) CN109970760B (pt)
AU (3) AU2012335088B2 (pt)
BR (2) BR112014011351B1 (pt)
CA (1) CA2855372C (pt)
CL (1) CL2014001241A1 (pt)
CY (2) CY1120224T1 (pt)
DK (2) DK2776038T3 (pt)
EA (2) EA030264B1 (pt)
ES (3) ES2767956T3 (pt)
HK (1) HK1201207A1 (pt)
HR (2) HRP20180534T1 (pt)
HU (2) HUE047049T2 (pt)
LT (2) LT3329919T (pt)
MX (3) MX344490B (pt)
PL (3) PL2776038T3 (pt)
PT (2) PT3329919T (pt)
RS (1) RS57157B1 (pt)
SI (2) SI3329919T1 (pt)
TW (4) TWI582095B (pt)
UA (2) UA123760C2 (pt)
WO (1) WO2013071169A1 (pt)
ZA (3) ZA201403633B (pt)

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DK2776038T3 (en) 2018-04-23
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PL2776038T3 (pl) 2018-06-29
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KR102060290B1 (ko) 2019-12-27
AU2017265088B2 (en) 2019-08-08
ZA201704173B (en) 2021-08-25
CN104105485A (zh) 2014-10-15
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TW201350489A (zh) 2013-12-16
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US9944655B2 (en) 2018-04-17
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JP6543358B2 (ja) 2019-07-10
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CL2014001241A1 (es) 2014-11-28
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US20150203510A1 (en) 2015-07-23
RS57157B1 (sr) 2018-07-31
HUE047049T2 (hu) 2020-04-28
PT2776038T (pt) 2018-04-18
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ZA201403633B (en) 2021-10-27

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