BR112016006319A2 - inibidores de irak e usos dos mesmos - Google Patents

inibidores de irak e usos dos mesmos

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Publication number
BR112016006319A2
BR112016006319A2 BR112016006319A BR112016006319A BR112016006319A2 BR 112016006319 A2 BR112016006319 A2 BR 112016006319A2 BR 112016006319 A BR112016006319 A BR 112016006319A BR 112016006319 A BR112016006319 A BR 112016006319A BR 112016006319 A2 BR112016006319 A2 BR 112016006319A2
Authority
BR
Brazil
Prior art keywords
irak inhibitors
irak
inhibitors
compositions
methods
Prior art date
Application number
BR112016006319A
Other languages
English (en)
Inventor
E Masse Craig
L Romero Donna
C Harriman Geraldine
robert greenwood Jeremy
Robinson Shaughnessy
Original Assignee
Nimbus Iris Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nimbus Iris Inc filed Critical Nimbus Iris Inc
Publication of BR112016006319A2 publication Critical patent/BR112016006319A2/pt

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    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
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Abstract

a presente invenção fornece compostos, composições dos mesmos e métodos de uso das mesmas.
BR112016006319A 2013-09-27 2014-09-25 inibidores de irak e usos dos mesmos BR112016006319A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361883497P 2013-09-27 2013-09-27
PCT/US2014/057444 WO2015048281A1 (en) 2013-09-27 2014-09-25 Irak inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
BR112016006319A2 true BR112016006319A2 (pt) 2017-08-01

Family

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Family Applications (1)

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BR112016006319A BR112016006319A2 (pt) 2013-09-27 2014-09-25 inibidores de irak e usos dos mesmos

Country Status (11)

Country Link
US (2) US9518065B2 (pt)
EP (1) EP3049086A4 (pt)
JP (1) JP2016531870A (pt)
KR (1) KR20160092991A (pt)
CN (1) CN106232122A (pt)
BR (1) BR112016006319A2 (pt)
CA (1) CA2925211A1 (pt)
MX (1) MX2016003843A (pt)
RU (1) RU2016110852A (pt)
TW (1) TW201522349A (pt)
WO (1) WO2015048281A1 (pt)

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WO2017024589A1 (zh) * 2015-08-13 2017-02-16 北京韩美药品有限公司 Irak4抑制剂及其应用
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