BR112014017021A2 - inibidores de irak e usos dos mesmos - Google Patents
inibidores de irak e usos dos mesmosInfo
- Publication number
- BR112014017021A2 BR112014017021A2 BR112014017021A BR112014017021A BR112014017021A2 BR 112014017021 A2 BR112014017021 A2 BR 112014017021A2 BR 112014017021 A BR112014017021 A BR 112014017021A BR 112014017021 A BR112014017021 A BR 112014017021A BR 112014017021 A2 BR112014017021 A2 BR 112014017021A2
- Authority
- BR
- Brazil
- Prior art keywords
- irak inhibitors
- compositions
- methods
- irak
- inhibitors
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
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- A61K31/33—Heterocyclic compounds
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Abstract
abstract the present invention provides compounds, compositions thereof, and methods of using the same. **************************** tradução do resumo resumo patente de invenção: "inibidores de irak e usos dos mesmos". a presente invenção fornece compostos, composições dos mesmos, e métodos de usar os mesmos. 21769624v1 1/1 21769624v1
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261585194P | 2012-01-10 | 2012-01-10 | |
US201261663227P | 2012-06-22 | 2012-06-22 | |
US201261682637P | 2012-08-13 | 2012-08-13 | |
US201261724695P | 2012-11-09 | 2012-11-09 | |
US201261734133P | 2012-12-06 | 2012-12-06 | |
PCT/US2013/020981 WO2013106535A1 (en) | 2012-01-10 | 2013-01-10 | Irak inhibitors and uses thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
BR112014017021A2 true BR112014017021A2 (pt) | 2017-06-13 |
BR112014017021A8 BR112014017021A8 (pt) | 2017-07-04 |
Family
ID=48781892
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112014017021A BR112014017021A8 (pt) | 2012-01-10 | 2013-01-10 | inibidores de irak e usos dos mesmos |
Country Status (10)
Country | Link |
---|---|
US (2) | US9212190B2 (pt) |
EP (1) | EP2802330A4 (pt) |
JP (2) | JP6126131B2 (pt) |
CN (1) | CN104582705A (pt) |
AU (2) | AU2013207972B2 (pt) |
BR (1) | BR112014017021A8 (pt) |
CA (1) | CA2863259A1 (pt) |
HK (1) | HK1209632A1 (pt) |
TW (2) | TW201728592A (pt) |
WO (1) | WO2013106535A1 (pt) |
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2013
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AU2017228639A1 (en) | 2017-10-26 |
BR112014017021A8 (pt) | 2017-07-04 |
CA2863259A1 (en) | 2013-07-18 |
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CN104582705A (zh) | 2015-04-29 |
EP2802330A4 (en) | 2015-10-21 |
EP2802330A1 (en) | 2014-11-19 |
TW201333014A (zh) | 2013-08-16 |
HK1209632A1 (en) | 2016-04-08 |
WO2013106535A1 (en) | 2013-07-18 |
US20130231328A1 (en) | 2013-09-05 |
TW201728592A (zh) | 2017-08-16 |
JP2015503618A (ja) | 2015-02-02 |
US9212190B2 (en) | 2015-12-15 |
WO2013106535A9 (en) | 2014-09-04 |
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