ZA201403633B - Acc inhibitors and uses thereof - Google Patents

Acc inhibitors and uses thereof

Info

Publication number
ZA201403633B
ZA201403633B ZA2014/03633A ZA201403633A ZA201403633B ZA 201403633 B ZA201403633 B ZA 201403633B ZA 2014/03633 A ZA2014/03633 A ZA 2014/03633A ZA 201403633 A ZA201403633 A ZA 201403633A ZA 201403633 B ZA201403633 B ZA 201403633B
Authority
ZA
South Africa
Prior art keywords
acc inhibitors
acc
inhibitors
Prior art date
Application number
ZA2014/03633A
Other languages
English (en)
Inventor
Geraldine C Harriman
James Harwood
Jeremy Robert Greenwood
Craig E Masse
Sathesh Bhat
Original Assignee
Nimbus Apollo Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nimbus Apollo Inc filed Critical Nimbus Apollo Inc
Publication of ZA201403633B publication Critical patent/ZA201403633B/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
ZA2014/03633A 2011-11-11 2014-05-19 Acc inhibitors and uses thereof ZA201403633B (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161559023P 2011-11-11 2011-11-11
US201261615092P 2012-03-23 2012-03-23
US201261651878P 2012-05-25 2012-05-25
US201261675513P 2012-07-25 2012-07-25
PCT/US2012/064528 WO2013071169A1 (en) 2011-11-11 2012-11-09 Acc inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
ZA201403633B true ZA201403633B (en) 2021-10-27

Family

ID=48281206

Family Applications (3)

Application Number Title Priority Date Filing Date
ZA2014/03633A ZA201403633B (en) 2011-11-11 2014-05-19 Acc inhibitors and uses thereof
ZA2017/04173A ZA201704173B (en) 2011-11-11 2017-06-19 Acc inhibitors and uses thereof
ZA2017/04192A ZA201704192B (en) 2011-11-11 2017-06-19 Acc inhibitors and uses thereof

Family Applications After (2)

Application Number Title Priority Date Filing Date
ZA2017/04173A ZA201704173B (en) 2011-11-11 2017-06-19 Acc inhibitors and uses thereof
ZA2017/04192A ZA201704192B (en) 2011-11-11 2017-06-19 Acc inhibitors and uses thereof

Country Status (26)

Country Link
US (5) US8969557B2 (enExample)
EP (3) EP3329919B1 (enExample)
JP (4) JP6114297B2 (enExample)
KR (3) KR102033806B1 (enExample)
CN (3) CN106905346B (enExample)
AU (3) AU2012335088B2 (enExample)
BR (2) BR112014011351B1 (enExample)
CA (1) CA2855372C (enExample)
CL (1) CL2014001241A1 (enExample)
CY (2) CY1120224T1 (enExample)
DK (2) DK3329919T3 (enExample)
EA (2) EA030264B1 (enExample)
ES (3) ES2767956T3 (enExample)
HR (2) HRP20180534T1 (enExample)
HU (2) HUE037444T2 (enExample)
LT (2) LT2776038T (enExample)
MX (3) MX370976B (enExample)
PL (3) PL3329919T3 (enExample)
PT (2) PT3329919T (enExample)
RS (1) RS57157B1 (enExample)
SI (2) SI3329919T1 (enExample)
SM (1) SMT201800191T1 (enExample)
TW (4) TWI701253B (enExample)
UA (2) UA123760C2 (enExample)
WO (1) WO2013071169A1 (enExample)
ZA (3) ZA201403633B (enExample)

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MX2020000331A (es) 2022-03-16
CA2855372C (en) 2022-03-22
RS57157B1 (sr) 2018-07-31
PT3329919T (pt) 2020-01-20
UA123760C2 (uk) 2021-06-02
JP2014533281A (ja) 2014-12-11
EP3329919B1 (en) 2019-11-06
US20200102323A1 (en) 2020-04-02
AU2017265088A1 (en) 2017-12-14
BR112014011351A2 (pt) 2017-06-06
PL2776038T3 (pl) 2018-06-29
US9944655B2 (en) 2018-04-17
NZ738735A (en) 2019-08-30
KR102033806B1 (ko) 2019-10-17
KR20140106554A (ko) 2014-09-03
EA030264B1 (ru) 2018-07-31
TWI612050B (zh) 2018-01-21
CN104105485A (zh) 2014-10-15
DK2776038T3 (en) 2018-04-23
MX2014005693A (es) 2014-11-26
JP2019147847A (ja) 2019-09-05
MX344490B (es) 2016-12-16
NZ624819A (en) 2016-10-28
EP2776038B1 (en) 2018-01-10
ES2767956T3 (es) 2020-06-19
EP2776038A4 (en) 2015-04-01
TW201350489A (zh) 2013-12-16
CA2855372A1 (en) 2013-05-16
TWI582095B (zh) 2017-05-11
DK3329919T3 (da) 2019-12-09
EA201692104A1 (ru) 2017-08-31
ES2912574T3 (es) 2022-05-26
WO2013071169A1 (en) 2013-05-16
NZ723933A (en) 2018-03-23
CN109970760A (zh) 2019-07-05
TWI701253B (zh) 2020-08-11
US8969557B2 (en) 2015-03-03
US20160297834A1 (en) 2016-10-13
HUE037444T2 (hu) 2018-09-28
KR102060290B1 (ko) 2019-12-27
AU2019253834A1 (en) 2019-11-14
JP6276442B2 (ja) 2018-02-07
US20150203510A1 (en) 2015-07-23
CN106905346B (zh) 2019-05-28
CY1122657T1 (el) 2021-03-12
SI3329919T1 (sl) 2020-02-28
KR20190041027A (ko) 2019-04-19
EP3628320A1 (en) 2020-04-01
AU2012335088A1 (en) 2014-05-29
US20130123231A1 (en) 2013-05-16
TWI655193B (zh) 2019-04-01
JP6756014B2 (ja) 2020-09-16
CN106905346A (zh) 2017-06-30
JP2017114910A (ja) 2017-06-29
US20190016732A1 (en) 2019-01-17
TW201930310A (zh) 2019-08-01
CN104105485B (zh) 2017-04-12
EP2776038A1 (en) 2014-09-17
CY1120224T1 (el) 2018-12-12
EP3329919A1 (en) 2018-06-06
MX370976B (es) 2020-01-10
CN109970760B (zh) 2022-04-26
UA114901C2 (uk) 2017-08-28
AU2019253834B2 (en) 2021-04-29
SI2776038T1 (en) 2018-06-29
CL2014001241A1 (es) 2014-11-28
ZA201704192B (en) 2021-10-27
KR20190143473A (ko) 2019-12-30
EA033598B1 (ru) 2019-11-07
HRP20180534T1 (hr) 2018-05-04
EP3329919A8 (en) 2020-10-07
AU2012335088B2 (en) 2017-08-24
BR112014011351B1 (pt) 2021-02-17
SMT201800191T1 (it) 2018-05-02
AU2017265088B2 (en) 2019-08-08
JP6543358B2 (ja) 2019-07-10
JP2018052989A (ja) 2018-04-05
US9453026B2 (en) 2016-09-27
KR102172902B1 (ko) 2020-11-02
TW201831492A (zh) 2018-09-01
MX390746B (es) 2025-03-21

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