PT2776038T - Inibidores de acc e utilizações dos mesmos - Google Patents

Inibidores de acc e utilizações dos mesmos

Info

Publication number
PT2776038T
PT2776038T PT128483617T PT12848361T PT2776038T PT 2776038 T PT2776038 T PT 2776038T PT 128483617 T PT128483617 T PT 128483617T PT 12848361 T PT12848361 T PT 12848361T PT 2776038 T PT2776038 T PT 2776038T
Authority
PT
Portugal
Prior art keywords
acc inhibitors
acc
inhibitors
Prior art date
Application number
PT128483617T
Other languages
English (en)
Portuguese (pt)
Inventor
C Harriman Geraldine
E Masse Craig
Harwood James
Bhat Sathesh
robert greenwood Jeremy
Original Assignee
Gilead Apollo Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Apollo Llc filed Critical Gilead Apollo Llc
Publication of PT2776038T publication Critical patent/PT2776038T/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
PT128483617T 2011-11-11 2012-11-09 Inibidores de acc e utilizações dos mesmos PT2776038T (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201161559023P 2011-11-11 2011-11-11
US201261615092P 2012-03-23 2012-03-23
US201261651878P 2012-05-25 2012-05-25
US201261675513P 2012-07-25 2012-07-25

Publications (1)

Publication Number Publication Date
PT2776038T true PT2776038T (pt) 2018-04-18

Family

ID=48281206

Family Applications (2)

Application Number Title Priority Date Filing Date
PT128483617T PT2776038T (pt) 2011-11-11 2012-11-09 Inibidores de acc e utilizações dos mesmos
PT172094559T PT3329919T (pt) 2011-11-11 2012-11-09 Inibidores de acc e suas utilizações

Family Applications After (1)

Application Number Title Priority Date Filing Date
PT172094559T PT3329919T (pt) 2011-11-11 2012-11-09 Inibidores de acc e suas utilizações

Country Status (26)

Country Link
US (5) US8969557B2 (enExample)
EP (3) EP3628320B1 (enExample)
JP (4) JP6114297B2 (enExample)
KR (3) KR102172902B1 (enExample)
CN (3) CN104105485B (enExample)
AU (3) AU2012335088B2 (enExample)
BR (2) BR112014011351B1 (enExample)
CA (1) CA2855372C (enExample)
CL (1) CL2014001241A1 (enExample)
CY (2) CY1120224T1 (enExample)
DK (2) DK2776038T3 (enExample)
EA (2) EA030264B1 (enExample)
ES (3) ES2767956T3 (enExample)
HR (2) HRP20180534T1 (enExample)
HU (2) HUE037444T2 (enExample)
LT (2) LT3329919T (enExample)
MX (3) MX344490B (enExample)
PL (3) PL3628320T3 (enExample)
PT (2) PT2776038T (enExample)
RS (1) RS57157B1 (enExample)
SI (2) SI3329919T1 (enExample)
SM (1) SMT201800191T1 (enExample)
TW (4) TWI655193B (enExample)
UA (2) UA123760C2 (enExample)
WO (1) WO2013071169A1 (enExample)
ZA (3) ZA201403633B (enExample)

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US10472374B2 (en) 2019-11-12
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ES2767956T3 (es) 2020-06-19
MX344490B (es) 2016-12-16
TW201720831A (zh) 2017-06-16
PL2776038T3 (pl) 2018-06-29
JP2014533281A (ja) 2014-12-11
KR102033806B1 (ko) 2019-10-17
KR20190041027A (ko) 2019-04-19
JP6756014B2 (ja) 2020-09-16
WO2013071169A1 (en) 2013-05-16
ES2912574T3 (es) 2022-05-26
AU2012335088B2 (en) 2017-08-24
NZ738735A (en) 2019-08-30
SMT201800191T1 (it) 2018-05-02
TW201930310A (zh) 2019-08-01
KR20140106554A (ko) 2014-09-03
TWI701253B (zh) 2020-08-11
CN104105485B (zh) 2017-04-12
ZA201704173B (en) 2021-08-25
BR112014011351A2 (pt) 2017-06-06
US20190016732A1 (en) 2019-01-17
UA114901C2 (uk) 2017-08-28
HUE037444T2 (hu) 2018-09-28
AU2019253834B2 (en) 2021-04-29
JP2017114910A (ja) 2017-06-29
TW201831492A (zh) 2018-09-01
MX390746B (es) 2025-03-21
CN106905346B (zh) 2019-05-28
DK3329919T3 (da) 2019-12-09
EA201692104A1 (ru) 2017-08-31
CN109970760B (zh) 2022-04-26
KR102060290B1 (ko) 2019-12-27
BR122019026836B1 (pt) 2021-02-23
US20200102323A1 (en) 2020-04-02
AU2017265088A1 (en) 2017-12-14
EP3329919B1 (en) 2019-11-06
EA201490826A1 (ru) 2015-01-30
EP3329919A1 (en) 2018-06-06
PL3628320T3 (pl) 2022-07-25
PL3329919T3 (pl) 2020-05-18
HRP20180534T1 (hr) 2018-05-04
AU2012335088A1 (en) 2014-05-29
RS57157B1 (sr) 2018-07-31
TW201350489A (zh) 2013-12-16
TWI612050B (zh) 2018-01-21
NZ723933A (en) 2018-03-23
KR102172902B1 (ko) 2020-11-02
CY1122657T1 (el) 2021-03-12
JP6114297B2 (ja) 2017-04-12
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TWI655193B (zh) 2019-04-01
EP3329919A8 (en) 2020-10-07
CN106905346A (zh) 2017-06-30
US8969557B2 (en) 2015-03-03
LT2776038T (lt) 2018-04-25
EP2776038A4 (en) 2015-04-01
SI2776038T1 (en) 2018-06-29
CL2014001241A1 (es) 2014-11-28
JP6543358B2 (ja) 2019-07-10
AU2019253834A1 (en) 2019-11-14
CA2855372C (en) 2022-03-22
EP3628320A1 (en) 2020-04-01
EP3628320B1 (en) 2022-03-16
EA030264B1 (ru) 2018-07-31
EA033598B1 (ru) 2019-11-07
ZA201704192B (en) 2021-10-27
US20130123231A1 (en) 2013-05-16
US9453026B2 (en) 2016-09-27
HRP20192202T1 (hr) 2020-03-06
BR112014011351B1 (pt) 2021-02-17
ES2665580T3 (es) 2018-04-26
NZ624819A (en) 2016-10-28
CN104105485A (zh) 2014-10-15
PT3329919T (pt) 2020-01-20
UA123760C2 (uk) 2021-06-02
JP6276442B2 (ja) 2018-02-07
AU2017265088B2 (en) 2019-08-08
ZA201403633B (en) 2021-10-27
LT3329919T (lt) 2020-02-10
MX2020000331A (es) 2022-03-16
JP2019147847A (ja) 2019-09-05
CA2855372A1 (en) 2013-05-16
MX2014005693A (es) 2014-11-26
US20150203510A1 (en) 2015-07-23
JP2018052989A (ja) 2018-04-05
US20160297834A1 (en) 2016-10-13
TWI582095B (zh) 2017-05-11
HUE047049T2 (hu) 2020-04-28
SI3329919T1 (sl) 2020-02-28
US9944655B2 (en) 2018-04-17
EP2776038A1 (en) 2014-09-17

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