SK17562001A3 - Použitie derivátov kyseliny (-)-(3-trihalogénmetylfenoxy)-(4- halogénfenyl)octovej na liečbu inzulínovej odolnosti, diabetu typu 2, hyperlipidémie a hyperurikémie - Google Patents

Použitie derivátov kyseliny (-)-(3-trihalogénmetylfenoxy)-(4- halogénfenyl)octovej na liečbu inzulínovej odolnosti, diabetu typu 2, hyperlipidémie a hyperurikémie Download PDF

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Publication number
SK17562001A3
SK17562001A3 SK1756-2001A SK17562001A SK17562001A3 SK 17562001 A3 SK17562001 A3 SK 17562001A3 SK 17562001 A SK17562001 A SK 17562001A SK 17562001 A3 SK17562001 A3 SK 17562001A3
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SK
Slovakia
Prior art keywords
compound
alkylamino
lower alkoxy
halofenate
alkoxy
Prior art date
Application number
SK1756-2001A
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English (en)
Slovak (sk)
Inventor
Kenneth L. Luskey
Jian Luo
Original Assignee
Metabolex, Inc.
Diatex, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23270381&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK17562001(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Metabolex, Inc., Diatex, Inc. filed Critical Metabolex, Inc.
Publication of SK17562001A3 publication Critical patent/SK17562001A3/sk

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/075—Ethers or acetals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A—HUMAN NECESSITIES
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    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/455—Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
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    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
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    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SK1756-2001A 1999-06-04 2000-06-02 Použitie derivátov kyseliny (-)-(3-trihalogénmetylfenoxy)-(4- halogénfenyl)octovej na liečbu inzulínovej odolnosti, diabetu typu 2, hyperlipidémie a hyperurikémie SK17562001A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/325,997 US6262118B1 (en) 1999-06-04 1999-06-04 Use of (-) (3-trihalomethylphenoxy) (4-halophenyl) acetic acid derivatives for treatment of insulin resistance, type 2 diabetes and hyperlipidemia
PCT/US2000/015235 WO2000074666A2 (en) 1999-06-04 2000-06-02 Use of (-) (3-trihalomethylphenoxy) (4-halophenyl) acetic acid derivatives for treatment of insulin resistance, type 2 diabetes, hyperlipidaemia and hyperuricaemia

Publications (1)

Publication Number Publication Date
SK17562001A3 true SK17562001A3 (sk) 2002-10-08

Family

ID=23270381

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1756-2001A SK17562001A3 (sk) 1999-06-04 2000-06-02 Použitie derivátov kyseliny (-)-(3-trihalogénmetylfenoxy)-(4- halogénfenyl)octovej na liečbu inzulínovej odolnosti, diabetu typu 2, hyperlipidémie a hyperurikémie

Country Status (32)

Country Link
US (6) US6262118B1 (zh)
EP (2) EP1183020B1 (zh)
JP (2) JP4685300B2 (zh)
KR (2) KR100721219B1 (zh)
CN (2) CN100379412C (zh)
AR (1) AR042574A1 (zh)
AT (2) ATE336235T1 (zh)
AU (1) AU775909C (zh)
BR (1) BR0011342A (zh)
CA (2) CA2751187C (zh)
CL (1) CL2011001971A1 (zh)
CO (1) CO5170453A1 (zh)
CY (1) CY1112861T1 (zh)
CZ (1) CZ20014341A3 (zh)
DE (1) DE60030109T2 (zh)
DK (2) DK1183020T3 (zh)
ES (2) ES2269151T3 (zh)
HK (2) HK1045111B (zh)
HU (1) HUP0201611A3 (zh)
IL (3) IL146914A0 (zh)
MX (1) MXPA01012435A (zh)
NO (1) NO20015909L (zh)
NZ (2) NZ515902A (zh)
PE (1) PE20010220A1 (zh)
PT (2) PT1183020E (zh)
RU (2) RU2281762C2 (zh)
SA (1) SA00210535B1 (zh)
SK (1) SK17562001A3 (zh)
TW (1) TWI264303B (zh)
UA (1) UA74147C2 (zh)
WO (1) WO2000074666A2 (zh)
ZA (3) ZA200300889B (zh)

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