RS52810B9 - 3-aminociklopentankarboksamidi kao modulatori hemokinskih receptora - Google Patents

3-aminociklopentankarboksamidi kao modulatori hemokinskih receptora

Info

Publication number
RS52810B9
RS52810B9 RS20130260A RSP20130260A RS52810B9 RS 52810 B9 RS52810 B9 RS 52810B9 RS 20130260 A RS20130260 A RS 20130260A RS P20130260 A RSP20130260 A RS P20130260A RS 52810 B9 RS52810 B9 RS 52810B9
Authority
RS
Serbia
Prior art keywords
amino
trifluoromethyl
carbonyl
diazabicyclo
dideoxy
Prior art date
Application number
RS20130260A
Other languages
English (en)
Serbian (sr)
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Jr Donald Joseph Rogier
John Isidro Trujillo
Steve Ronald Turner
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of RS52810B publication Critical patent/RS52810B/sr
Publication of RS52810B9 publication Critical patent/RS52810B9/sr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P11/06Antiasthmatics
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    • A61P13/12Drugs for disorders of the urinary system of the kidneys
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
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    • AHUMAN NECESSITIES
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Otolaryngology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Virology (AREA)
  • Emergency Medicine (AREA)
RS20130260A 2008-11-26 2009-11-20 3-aminociklopentankarboksamidi kao modulatori hemokinskih receptora RS52810B9 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26
PCT/IB2009/055232 WO2010061329A1 (en) 2008-11-26 2009-11-20 3-aminocyclopentanecarboxamides as chemokine receptor modulators
EP09774939.4A EP2370442B9 (en) 2008-11-26 2009-11-20 3-Aminocyclopentanecarboxamides as chemokine receptor modulators

Publications (2)

Publication Number Publication Date
RS52810B RS52810B (sr) 2013-10-31
RS52810B9 true RS52810B9 (sr) 2019-06-28

Family

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Family Applications (2)

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RS20130260A RS52810B9 (sr) 2008-11-26 2009-11-20 3-aminociklopentankarboksamidi kao modulatori hemokinskih receptora
RS20130260D RS52810B8 (sr) 2008-11-26 2009-11-20 3-aminociklopentankarboksamidi kao modulatori hemokinskih receptora

Family Applications After (1)

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RS20130260D RS52810B8 (sr) 2008-11-26 2009-11-20 3-aminociklopentankarboksamidi kao modulatori hemokinskih receptora

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EP (1) EP2370442B9 (enExample)
JP (1) JP5108153B2 (enExample)
KR (1) KR101374412B1 (enExample)
CN (1) CN102227429B (enExample)
AP (1) AP3113A (enExample)
AU (1) AU2009321221B2 (enExample)
BR (1) BRPI0920936A2 (enExample)
CA (1) CA2743030C (enExample)
CL (1) CL2011001223A1 (enExample)
CO (1) CO6361921A2 (enExample)
CR (1) CR20110275A (enExample)
CU (1) CU24022B1 (enExample)
CY (1) CY1114020T1 (enExample)
DK (1) DK2370442T5 (enExample)
DO (1) DOP2011000154A (enExample)
EA (1) EA020470B1 (enExample)
EC (1) ECSP11011081A (enExample)
ES (1) ES2415430T3 (enExample)
GE (1) GEP20146064B (enExample)
HR (1) HRP20130409T2 (enExample)
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ME (1) ME01144B (enExample)
MX (1) MX2011005526A (enExample)
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NZ (1) NZ592919A (enExample)
PE (1) PE20110831A1 (enExample)
PL (1) PL2370442T3 (enExample)
PT (1) PT2370442E (enExample)
RS (2) RS52810B9 (enExample)
SI (1) SI2370442T1 (enExample)
SV (1) SV2011003923A (enExample)
TN (1) TN2011000254A1 (enExample)
UA (1) UA99978C2 (enExample)
WO (1) WO2010061329A1 (enExample)
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ME01144B (me) * 2008-11-26 2013-03-20 Pfizer 3-aminociklopentankarboksamidi kao modulatori hemokin receptora
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1r,2r,3r)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
CA2946538A1 (en) 2014-04-04 2015-10-08 Del Mar Pharmaceuticals Use of dianhydrogalactitol and analogs or derivatives thereof to treat non-small-cell carcinoma of the lung and ovarian cancer
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JOP20190040A1 (ar) * 2016-09-14 2019-03-10 Novartis Ag توليفة من ناهضات fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲(江蘇)醫藥有限公司 環戊烷化合物

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IL212732A0 (en) 2011-07-31
ECSP11011081A (es) 2011-12-30
BRPI0920936A2 (pt) 2020-08-11
AU2009321221A1 (en) 2010-06-03
US20110144129A1 (en) 2011-06-16
UA99978C2 (en) 2012-10-25
ES2415430T3 (es) 2013-07-25
RS52810B8 (sr) 2019-08-30
CR20110275A (es) 2011-07-01
IL212732A (en) 2016-06-30
HK1161261A1 (en) 2012-08-24
RS52810B (sr) 2013-10-31
DK2370442T3 (da) 2013-06-17
CY1114020T1 (el) 2016-07-27
US20130197008A1 (en) 2013-08-01
ME01144B (me) 2013-03-20
JP2012509931A (ja) 2012-04-26
TN2011000254A1 (fr) 2012-12-17
PT2370442E (pt) 2013-06-27
CA2743030A1 (en) 2010-06-03
JP5108153B2 (ja) 2012-12-26
MA32834B1 (fr) 2011-11-01
AP2011005732A0 (en) 2011-06-30
CU24022B1 (es) 2014-07-30
DK2370442T5 (da) 2013-09-23
NI201100102A (es) 2011-09-27
EP2370442B1 (en) 2013-04-24
AU2009321221B2 (en) 2013-04-04
GEP20146064B (en) 2014-03-25
PE20110831A1 (es) 2011-11-20
CU20110121A7 (es) 2013-05-31
ZA201104069B (en) 2012-02-29
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EP2370442B9 (en) 2013-09-04
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KR20110075036A (ko) 2011-07-05
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WO2010061329A1 (en) 2010-06-03
EA020470B1 (ru) 2014-11-28
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EP2370442A1 (en) 2011-10-05
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CN102227429A (zh) 2011-10-26
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DOP2011000154A (es) 2011-07-31
PL2370442T3 (pl) 2013-08-30
SI2370442T1 (sl) 2013-06-28
EA201170721A1 (ru) 2011-12-30
HRP20130409T2 (hr) 2013-11-22
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AP3113A (en) 2015-01-31
KR101374412B1 (ko) 2014-03-17

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