CU24022B1 - 3-aminociclopentancarboxamidas - Google Patents

3-aminociclopentancarboxamidas

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Publication number
CU24022B1
CU24022B1 CU2011000121A CU20110121A CU24022B1 CU 24022 B1 CU24022 B1 CU 24022B1 CU 2011000121 A CU2011000121 A CU 2011000121A CU 20110121 A CU20110121 A CU 20110121A CU 24022 B1 CU24022 B1 CU 24022B1
Authority
CU
Cuba
Prior art keywords
aminociclopentancarboxamidas
hept
diazabicyclo
cyclopentyl
carbonyl
Prior art date
Application number
CU2011000121A
Other languages
English (en)
Other versions
CU20110121A7 (es
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Jr Donald Joseph Rogier
John Isidro Trujillo
Steve Ronald Turner
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CU20110121A7 publication Critical patent/CU20110121A7/es
Publication of CU24022B1 publication Critical patent/CU24022B1/es

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Veterinary Medicine (AREA)
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  • Neurology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
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  • Otolaryngology (AREA)
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Abstract

La invención se refiere a derivados de (2,5-diazabiciclo(2.2.1)hept-2-il)carbonil)ciclopentil)amino útiles como moduladores del receptor de quimiocina.
CU2011000121A 2008-11-26 2011-05-26 3-aminociclopentancarboxamidas CU24022B1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26
PCT/IB2009/055232 WO2010061329A1 (en) 2008-11-26 2009-11-20 3-aminocyclopentanecarboxamides as chemokine receptor modulators

Publications (2)

Publication Number Publication Date
CU20110121A7 CU20110121A7 (es) 2013-05-31
CU24022B1 true CU24022B1 (es) 2014-07-30

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ID=41693100

Family Applications (1)

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CU2011000121A CU24022B1 (es) 2008-11-26 2011-05-26 3-aminociclopentancarboxamidas

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US (2) US8293903B2 (es)
EP (1) EP2370442B9 (es)
JP (1) JP5108153B2 (es)
KR (1) KR101374412B1 (es)
CN (1) CN102227429B (es)
AP (1) AP3113A (es)
AU (1) AU2009321221B2 (es)
BR (1) BRPI0920936A2 (es)
CA (1) CA2743030C (es)
CL (1) CL2011001223A1 (es)
CO (1) CO6361921A2 (es)
CR (1) CR20110275A (es)
CU (1) CU24022B1 (es)
CY (1) CY1114020T1 (es)
DK (1) DK2370442T5 (es)
DO (1) DOP2011000154A (es)
EA (1) EA020470B1 (es)
EC (1) ECSP11011081A (es)
ES (1) ES2415430T3 (es)
GE (1) GEP20146064B (es)
HK (1) HK1161261A1 (es)
HR (1) HRP20130409T2 (es)
IL (1) IL212732A (es)
MA (1) MA32834B1 (es)
ME (1) ME01144B (es)
MX (1) MX2011005526A (es)
MY (1) MY152557A (es)
NI (1) NI201100102A (es)
NZ (1) NZ592919A (es)
PE (1) PE20110831A1 (es)
PL (1) PL2370442T3 (es)
PT (1) PT2370442E (es)
RS (2) RS52810B8 (es)
SI (1) SI2370442T1 (es)
SV (1) SV2011003923A (es)
TN (1) TN2011000254A1 (es)
UA (1) UA99978C2 (es)
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DK2370442T5 (da) * 2008-11-26 2013-09-23 Pfizer 3-aminocyclopentancarboxamider som chemokinreceptor modulatorer
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1r,2r,3r)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
KR102456088B1 (ko) 2014-04-04 2022-10-19 델 마 파마슈티컬스 폐의 비소세포 암종 및 난소암을 치료하기 위한 디안하이드로갈락티톨 및 이의 유사체 또는 유도체
TW201605451A (zh) * 2014-07-17 2016-02-16 參天製藥股份有限公司 老年性黃斑部病變之預防或治療劑
JOP20190040A1 (ar) * 2016-09-14 2019-03-10 Novartis Ag توليفة من ناهضات fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲(江蘇)醫藥有限公司 環戊烷化合物
JP7412034B1 (ja) 2022-11-02 2024-01-12 鈴木製機株式会社 搬送システム

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BRPI0920936A2 (pt) 2020-08-11
US8293903B2 (en) 2012-10-23
SV2011003923A (es) 2011-07-28
US20130197008A1 (en) 2013-08-01
HK1161261A1 (en) 2012-08-24
EP2370442B1 (en) 2013-04-24
MY152557A (en) 2014-10-31
EP2370442A1 (en) 2011-10-05
DOP2011000154A (es) 2011-07-31
ECSP11011081A (es) 2011-12-30
ES2415430T9 (es) 2013-11-25
JP5108153B2 (ja) 2012-12-26
WO2010061329A1 (en) 2010-06-03
KR20110075036A (ko) 2011-07-05
EA020470B1 (ru) 2014-11-28
EA201170721A1 (ru) 2011-12-30
CU20110121A7 (es) 2013-05-31
US20110144129A1 (en) 2011-06-16
PL2370442T3 (pl) 2013-08-30
CA2743030A1 (en) 2010-06-03
TN2011000254A1 (fr) 2012-12-17
CN102227429B (zh) 2014-05-28
CY1114020T1 (el) 2016-07-27
CL2011001223A1 (es) 2011-09-02
AP2011005732A0 (en) 2011-06-30
MX2011005526A (es) 2011-06-06
AP3113A (en) 2015-01-31
HRP20130409T2 (hr) 2013-11-22
GEP20146064B (en) 2014-03-25
IL212732A (en) 2016-06-30
ZA201104069B (en) 2012-02-29
IL212732A0 (en) 2011-07-31
NZ592919A (en) 2013-05-31
NI201100102A (es) 2011-09-27
AU2009321221A1 (en) 2010-06-03
DK2370442T3 (da) 2013-06-17
HRP20130409T1 (en) 2013-06-30
US8946413B2 (en) 2015-02-03
AU2009321221B2 (en) 2013-04-04
ES2415430T3 (es) 2013-07-25
RS52810B (en) 2013-10-31
CO6361921A2 (es) 2012-01-20
CR20110275A (es) 2011-07-01
CA2743030C (en) 2013-10-22
KR101374412B1 (ko) 2014-03-17
JP2012509931A (ja) 2012-04-26
RS52810B8 (sr) 2019-08-30
CN102227429A (zh) 2011-10-26
PE20110831A1 (es) 2011-11-20
SI2370442T1 (sl) 2013-06-28
UA99978C2 (en) 2012-10-25
MA32834B1 (fr) 2011-11-01
ME01144B (me) 2013-03-20
RS52810B9 (sr) 2019-06-28
DK2370442T5 (da) 2013-09-23
PT2370442E (pt) 2013-06-27
EP2370442B9 (en) 2013-09-04

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