CR20110275A - 3-aminociclopentancarboxamidas como moduladores del receptor quimiocina - Google Patents

3-aminociclopentancarboxamidas como moduladores del receptor quimiocina

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Publication number
CR20110275A
CR20110275A CR20110275A CR20110275A CR20110275A CR 20110275 A CR20110275 A CR 20110275A CR 20110275 A CR20110275 A CR 20110275A CR 20110275 A CR20110275 A CR 20110275A CR 20110275 A CR20110275 A CR 20110275A
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CR
Costa Rica
Prior art keywords
chemiokin
aminociclopentancarboxamids
receptor modulators
compound
formula
Prior art date
Application number
CR20110275A
Other languages
English (en)
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Donald Joseph Rogier Jr
John Isidro Trujillo
Steve Ronald Turner
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CR20110275A publication Critical patent/CR20110275A/es

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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Abstract

Se provee un compuesto de la Fórmula, o una sal éste farmacéuticamente aceptable, en donde varios sustituyentes se definen en la presente.
CR20110275A 2008-11-26 2011-05-26 3-aminociclopentancarboxamidas como moduladores del receptor quimiocina CR20110275A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26

Publications (1)

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CR20110275A true CR20110275A (es) 2011-07-01

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Family Applications (1)

Application Number Title Priority Date Filing Date
CR20110275A CR20110275A (es) 2008-11-26 2011-05-26 3-aminociclopentancarboxamidas como moduladores del receptor quimiocina

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EP (1) EP2370442B9 (es)
JP (1) JP5108153B2 (es)
KR (1) KR101374412B1 (es)
CN (1) CN102227429B (es)
AP (1) AP3113A (es)
AU (1) AU2009321221B2 (es)
BR (1) BRPI0920936A2 (es)
CA (1) CA2743030C (es)
CL (1) CL2011001223A1 (es)
CO (1) CO6361921A2 (es)
CR (1) CR20110275A (es)
CU (1) CU24022B1 (es)
CY (1) CY1114020T1 (es)
DK (1) DK2370442T5 (es)
DO (1) DOP2011000154A (es)
EA (1) EA020470B1 (es)
EC (1) ECSP11011081A (es)
ES (1) ES2415430T3 (es)
GE (1) GEP20146064B (es)
HK (1) HK1161261A1 (es)
HR (1) HRP20130409T2 (es)
IL (1) IL212732A (es)
MA (1) MA32834B1 (es)
ME (1) ME01144B (es)
MX (1) MX2011005526A (es)
MY (1) MY152557A (es)
NI (1) NI201100102A (es)
NZ (1) NZ592919A (es)
PE (1) PE20110831A1 (es)
PL (1) PL2370442T3 (es)
PT (1) PT2370442E (es)
RS (2) RS52810B8 (es)
SI (1) SI2370442T1 (es)
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TN (1) TN2011000254A1 (es)
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PL2370442T3 (pl) * 2008-11-26 2013-08-30 Pfizer 3-Aminocyklopentanokarboksamidy jako modulatory receptora chemokiny
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1ｒ,2ｒ,3ｒ)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
EP3125920B1 (en) 2014-04-04 2020-12-23 Del Mar Pharmaceuticals Dianhydrogalactitol, diacetyldianhydrogalactitol or dibromodulcitol to treat non-small-cell carcinoma of the lung and ovarian cancer
JP2016029038A (ja) * 2014-07-17 2016-03-03 参天製薬株式会社 加齢黄斑変性の予防または治療剤
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EA020470B1 (ru) 2014-11-28
GEP20146064B (en) 2014-03-25
HRP20130409T1 (en) 2013-06-30
MA32834B1 (fr) 2011-11-01
CU20110121A7 (es) 2013-05-31
WO2010061329A1 (en) 2010-06-03
IL212732A (en) 2016-06-30
RS52810B (en) 2013-10-31
BRPI0920936A2 (pt) 2020-08-11
ME01144B (me) 2013-03-20
RS52810B8 (sr) 2019-08-30
ES2415430T3 (es) 2013-07-25
DOP2011000154A (es) 2011-07-31
EP2370442B9 (en) 2013-09-04
CO6361921A2 (es) 2012-01-20
SI2370442T1 (sl) 2013-06-28
EA201170721A1 (ru) 2011-12-30
JP5108153B2 (ja) 2012-12-26
NI201100102A (es) 2011-09-27
US8293903B2 (en) 2012-10-23
HK1161261A1 (en) 2012-08-24
AU2009321221B2 (en) 2013-04-04
EP2370442B1 (en) 2013-04-24
MX2011005526A (es) 2011-06-06
ZA201104069B (en) 2012-02-29
JP2012509931A (ja) 2012-04-26
CU24022B1 (es) 2014-07-30
US20110144129A1 (en) 2011-06-16
CA2743030C (en) 2013-10-22
CN102227429A (zh) 2011-10-26
ECSP11011081A (es) 2011-12-30
PT2370442E (pt) 2013-06-27
CA2743030A1 (en) 2010-06-03
AP3113A (en) 2015-01-31
KR101374412B1 (ko) 2014-03-17
RS52810B9 (sr) 2019-06-28
US20130197008A1 (en) 2013-08-01
SV2011003923A (es) 2011-07-28
AU2009321221A1 (en) 2010-06-03
HRP20130409T2 (hr) 2013-11-22
CY1114020T1 (el) 2016-07-27
ES2415430T9 (es) 2013-11-25
PL2370442T3 (pl) 2013-08-30
US8946413B2 (en) 2015-02-03
AP2011005732A0 (en) 2011-06-30
DK2370442T5 (da) 2013-09-23
MY152557A (en) 2014-10-31
TN2011000254A1 (fr) 2012-12-17
CN102227429B (zh) 2014-05-28
EP2370442A1 (en) 2011-10-05
CL2011001223A1 (es) 2011-09-02
KR20110075036A (ko) 2011-07-05
DK2370442T3 (da) 2013-06-17
PE20110831A1 (es) 2011-11-20
UA99978C2 (en) 2012-10-25
IL212732A0 (en) 2011-07-31
NZ592919A (en) 2013-05-31

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