AP3113A - 3-Aminocyclopentanecarboxamides as chemokine receptor modulators - Google Patents

3-Aminocyclopentanecarboxamides as chemokine receptor modulators

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Publication number
AP3113A
AP3113A AP2011005732A AP2011005732A AP3113A AP 3113 A AP3113 A AP 3113A AP 2011005732 A AP2011005732 A AP 2011005732A AP 2011005732 A AP2011005732 A AP 2011005732A AP 3113 A AP3113 A AP 3113A
Authority
AP
ARIPO
Prior art keywords
aminocyclopentanecarboxamides
chemokine receptor
receptor modulators
modulators
chemokine
Prior art date
Application number
AP2011005732A
Other languages
English (en)
Other versions
AP2011005732A0 (en
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of AP2011005732A0 publication Critical patent/AP2011005732A0/xx
Application granted granted Critical
Publication of AP3113A publication Critical patent/AP3113A/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Otolaryngology (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Nutrition Science (AREA)
  • Virology (AREA)
AP2011005732A 2008-11-26 2009-11-20 3-Aminocyclopentanecarboxamides as chemokine receptor modulators AP3113A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26
PCT/IB2009/055232 WO2010061329A1 (en) 2008-11-26 2009-11-20 3-aminocyclopentanecarboxamides as chemokine receptor modulators

Publications (2)

Publication Number Publication Date
AP2011005732A0 AP2011005732A0 (en) 2011-06-30
AP3113A true AP3113A (en) 2015-01-31

Family

ID=41693100

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2011005732A AP3113A (en) 2008-11-26 2009-11-20 3-Aminocyclopentanecarboxamides as chemokine receptor modulators

Country Status (39)

Country Link
US (2) US8293903B2 (es)
EP (1) EP2370442B9 (es)
JP (1) JP5108153B2 (es)
KR (1) KR101374412B1 (es)
CN (1) CN102227429B (es)
AP (1) AP3113A (es)
AU (1) AU2009321221B2 (es)
BR (1) BRPI0920936A2 (es)
CA (1) CA2743030C (es)
CL (1) CL2011001223A1 (es)
CO (1) CO6361921A2 (es)
CR (1) CR20110275A (es)
CU (1) CU24022B1 (es)
CY (1) CY1114020T1 (es)
DK (1) DK2370442T5 (es)
DO (1) DOP2011000154A (es)
EA (1) EA020470B1 (es)
EC (1) ECSP11011081A (es)
ES (1) ES2415430T3 (es)
GE (1) GEP20146064B (es)
HK (1) HK1161261A1 (es)
HR (1) HRP20130409T2 (es)
IL (1) IL212732A (es)
MA (1) MA32834B1 (es)
ME (1) ME01144B (es)
MX (1) MX2011005526A (es)
MY (1) MY152557A (es)
NI (1) NI201100102A (es)
NZ (1) NZ592919A (es)
PE (1) PE20110831A1 (es)
PL (1) PL2370442T3 (es)
PT (1) PT2370442E (es)
RS (2) RS52810B8 (es)
SI (1) SI2370442T1 (es)
SV (1) SV2011003923A (es)
TN (1) TN2011000254A1 (es)
UA (1) UA99978C2 (es)
WO (1) WO2010061329A1 (es)
ZA (1) ZA201104069B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GEP20146064B (en) * 2008-11-26 2014-03-25 Pfizer 3-minocyclopentanecarboxamides as chemokine receptor modulators
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1ｒ,2ｒ,3ｒ)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
KR102456088B1 (ko) 2014-04-04 2022-10-19 델 마 파마슈티컬스 폐의 비소세포 암종 및 난소암을 치료하기 위한 디안하이드로갈락티톨 및 이의 유사체 또는 유도체
WO2016010131A1 (ja) * 2014-07-17 2016-01-21 参天製薬株式会社 加齢黄斑変性の予防または治療剤
JOP20190040A1 (ar) * 2016-09-14 2019-03-10 Novartis Ag توليفة من ناهضات fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲（江蘇）醫藥有限公司 環戊烷化合物
JP7412034B1 (ja) 2022-11-02 2024-01-12 鈴木製機株式会社 搬送システム

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US20060020133A1 (en) * 2004-06-28 2006-01-26 Chu-Biao Xue 3-aminocyclopentanecarboxamides as modulators of chemokine receptors

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PL2370442T3 (pl) 2013-08-30
MY152557A (en) 2014-10-31
KR20110075036A (ko) 2011-07-05
WO2010061329A1 (en) 2010-06-03
EA201170721A1 (ru) 2011-12-30
US8293903B2 (en) 2012-10-23
SI2370442T1 (sl) 2013-06-28
PT2370442E (pt) 2013-06-27
AU2009321221A1 (en) 2010-06-03
CN102227429A (zh) 2011-10-26
EA020470B1 (ru) 2014-11-28
EP2370442A1 (en) 2011-10-05
RS52810B8 (sr) 2019-08-30
US20130197008A1 (en) 2013-08-01
ZA201104069B (en) 2012-02-29
UA99978C2 (en) 2012-10-25
CU20110121A7 (es) 2013-05-31
CN102227429B (zh) 2014-05-28
SV2011003923A (es) 2011-07-28
EP2370442B1 (en) 2013-04-24
HRP20130409T2 (hr) 2013-11-22
PE20110831A1 (es) 2011-11-20
DK2370442T5 (da) 2013-09-23
RS52810B9 (sr) 2019-06-28
JP2012509931A (ja) 2012-04-26
RS52810B (en) 2013-10-31
ES2415430T3 (es) 2013-07-25
IL212732A0 (en) 2011-07-31
CO6361921A2 (es) 2012-01-20
CR20110275A (es) 2011-07-01
IL212732A (en) 2016-06-30
JP5108153B2 (ja) 2012-12-26
KR101374412B1 (ko) 2014-03-17
NZ592919A (en) 2013-05-31
CA2743030C (en) 2013-10-22
DK2370442T3 (da) 2013-06-17
BRPI0920936A2 (pt) 2020-08-11
ECSP11011081A (es) 2011-12-30
CL2011001223A1 (es) 2011-09-02
MX2011005526A (es) 2011-06-06
US8946413B2 (en) 2015-02-03
ME01144B (me) 2013-03-20
ES2415430T9 (es) 2013-11-25
CU24022B1 (es) 2014-07-30
CA2743030A1 (en) 2010-06-03
GEP20146064B (en) 2014-03-25
HK1161261A1 (en) 2012-08-24
HRP20130409T1 (en) 2013-06-30
AP2011005732A0 (en) 2011-06-30
EP2370442B9 (en) 2013-09-04
NI201100102A (es) 2011-09-27
CY1114020T1 (el) 2016-07-27
TN2011000254A1 (fr) 2012-12-17
DOP2011000154A (es) 2011-07-31
AU2009321221B2 (en) 2013-04-04
US20110144129A1 (en) 2011-06-16
MA32834B1 (fr) 2011-11-01

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