DOP2011000154A - 3-aminociclopentancarboxamidas - Google Patents

3-aminociclopentancarboxamidas

Info

Publication number
DOP2011000154A
DOP2011000154A DO2011000154A DO2011000154A DOP2011000154A DO P2011000154 A DOP2011000154 A DO P2011000154A DO 2011000154 A DO2011000154 A DO 2011000154A DO 2011000154 A DO2011000154 A DO 2011000154A DO P2011000154 A DOP2011000154 A DO P2011000154A
Authority
DO
Dominican Republic
Prior art keywords
aminociclopentancarboxamidas
compound
formula
pharmaceutically acceptable
acceptable salt
Prior art date
Application number
DO2011000154A
Other languages
English (en)
Spanish (es)
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Donald Joseph Rogier Jr
John Isidro Trujillo
Steve Ronald Turner
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DOP2011000154A publication Critical patent/DOP2011000154A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
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  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Otolaryngology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Psychiatry (AREA)
  • Nutrition Science (AREA)
  • Virology (AREA)
DO2011000154A 2008-11-26 2011-05-25 3-aminociclopentancarboxamidas DOP2011000154A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26

Publications (1)

Publication Number Publication Date
DOP2011000154A true DOP2011000154A (es) 2011-07-31

Family

ID=41693100

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2011000154A DOP2011000154A (es) 2008-11-26 2011-05-25 3-aminociclopentancarboxamidas

Country Status (38)

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US (2) US8293903B2 (enExample)
EP (1) EP2370442B9 (enExample)
JP (1) JP5108153B2 (enExample)
KR (1) KR101374412B1 (enExample)
CN (1) CN102227429B (enExample)
AP (1) AP3113A (enExample)
AU (1) AU2009321221B2 (enExample)
BR (1) BRPI0920936A2 (enExample)
CA (1) CA2743030C (enExample)
CL (1) CL2011001223A1 (enExample)
CO (1) CO6361921A2 (enExample)
CR (1) CR20110275A (enExample)
CU (1) CU24022B1 (enExample)
CY (1) CY1114020T1 (enExample)
DK (1) DK2370442T5 (enExample)
DO (1) DOP2011000154A (enExample)
EA (1) EA020470B1 (enExample)
EC (1) ECSP11011081A (enExample)
ES (1) ES2415430T3 (enExample)
GE (1) GEP20146064B (enExample)
HR (1) HRP20130409T2 (enExample)
IL (1) IL212732A (enExample)
MA (1) MA32834B1 (enExample)
ME (1) ME01144B (enExample)
MX (1) MX2011005526A (enExample)
MY (1) MY152557A (enExample)
NI (1) NI201100102A (enExample)
NZ (1) NZ592919A (enExample)
PE (1) PE20110831A1 (enExample)
PL (1) PL2370442T3 (enExample)
PT (1) PT2370442E (enExample)
RS (2) RS52810B9 (enExample)
SI (1) SI2370442T1 (enExample)
SV (1) SV2011003923A (enExample)
TN (1) TN2011000254A1 (enExample)
UA (1) UA99978C2 (enExample)
WO (1) WO2010061329A1 (enExample)
ZA (1) ZA201104069B (enExample)

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BRPI0920936A2 (pt) * 2008-11-26 2020-08-11 Pfizer Inc 3-aminociclopentanocarboxamidas como moduladores de receptores de quimiocinas
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1ｒ,2ｒ,3ｒ)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
KR102456088B1 (ko) 2014-04-04 2022-10-19 델 마 파마슈티컬스 폐의 비소세포 암종 및 난소암을 치료하기 위한 디안하이드로갈락티톨 및 이의 유사체 또는 유도체
TW201605451A (zh) * 2014-07-17 2016-02-16 參天製藥股份有限公司 老年性黃斑部病變之預防或治療劑
JOP20190040A1 (ar) * 2016-09-14 2019-03-10 Novartis Ag توليفة من ناهضات fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲（江蘇）醫藥有限公司 環戊烷化合物

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KR101374412B1 (ko) 2014-03-17
CA2743030C (en) 2013-10-22
HRP20130409T2 (hr) 2013-11-22
PT2370442E (pt) 2013-06-27
CL2011001223A1 (es) 2011-09-02
AP3113A (en) 2015-01-31
BRPI0920936A2 (pt) 2020-08-11
DK2370442T5 (da) 2013-09-23
NZ592919A (en) 2013-05-31
SI2370442T1 (sl) 2013-06-28
EA201170721A1 (ru) 2011-12-30
AU2009321221B2 (en) 2013-04-04
CR20110275A (es) 2011-07-01
NI201100102A (es) 2011-09-27
RS52810B (sr) 2013-10-31
TN2011000254A1 (fr) 2012-12-17
CU20110121A7 (es) 2013-05-31
CO6361921A2 (es) 2012-01-20
WO2010061329A1 (en) 2010-06-03
CA2743030A1 (en) 2010-06-03
AU2009321221A1 (en) 2010-06-03
EP2370442B9 (en) 2013-09-04
MY152557A (en) 2014-10-31
ES2415430T9 (es) 2013-11-25
MA32834B1 (fr) 2011-11-01
GEP20146064B (en) 2014-03-25
RS52810B8 (sr) 2019-08-30
US20110144129A1 (en) 2011-06-16
DK2370442T3 (da) 2013-06-17
KR20110075036A (ko) 2011-07-05
JP2012509931A (ja) 2012-04-26
JP5108153B2 (ja) 2012-12-26
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US20130197008A1 (en) 2013-08-01
PL2370442T3 (pl) 2013-08-30
PE20110831A1 (es) 2011-11-20
IL212732A (en) 2016-06-30
ECSP11011081A (es) 2011-12-30
EA020470B1 (ru) 2014-11-28
ME01144B (me) 2013-03-20
UA99978C2 (en) 2012-10-25
US8946413B2 (en) 2015-02-03
EP2370442B1 (en) 2013-04-24
IL212732A0 (en) 2011-07-31
EP2370442A1 (en) 2011-10-05
CU24022B1 (es) 2014-07-30
CN102227429A (zh) 2011-10-26
CN102227429B (zh) 2014-05-28
ZA201104069B (en) 2012-02-29
CY1114020T1 (el) 2016-07-27
RS52810B9 (sr) 2019-06-28
US8293903B2 (en) 2012-10-23
HRP20130409T1 (en) 2013-06-30
HK1161261A1 (en) 2012-08-24
AP2011005732A0 (en) 2011-06-30
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SV2011003923A (es) 2011-07-28

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