EA020470B1 - 3-аминоциклопентанкарбоксамиды в качестве модуляторов рецептора хемокина - Google Patents

3-аминоциклопентанкарбоксамиды в качестве модуляторов рецептора хемокина Download PDF

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Publication number
EA020470B1
EA020470B1 EA201170721A EA201170721A EA020470B1 EA 020470 B1 EA020470 B1 EA 020470B1 EA 201170721 A EA201170721 A EA 201170721A EA 201170721 A EA201170721 A EA 201170721A EA 020470 B1 EA020470 B1 EA 020470B1
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EA
Eurasian Patent Office
Prior art keywords
amino
trifluoromethyl
diazabicyclo
carbonyl
anhydro
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EA201170721A
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English (en)
Russian (ru)
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EA201170721A1 (ru
Inventor
Раджеш Венкатесваран Деврадж
Вей Хуанг
Роберт Оуэн Хьюгес
Дональд Джозеф Роджиер Дж.
Джон Исидро Труджилло
Стив Рональд Тёрнер
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Пфайзер Инк.
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Publication of EA201170721A1 publication Critical patent/EA201170721A1/ru
Publication of EA020470B1 publication Critical patent/EA020470B1/ru

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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EA201170721A 2008-11-26 2009-11-20 3-аминоциклопентанкарбоксамиды в качестве модуляторов рецептора хемокина EA020470B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26
PCT/IB2009/055232 WO2010061329A1 (en) 2008-11-26 2009-11-20 3-aminocyclopentanecarboxamides as chemokine receptor modulators

Publications (2)

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EA201170721A1 EA201170721A1 (ru) 2011-12-30
EA020470B1 true EA020470B1 (ru) 2014-11-28

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EA201170721A EA020470B1 (ru) 2008-11-26 2009-11-20 3-аминоциклопентанкарбоксамиды в качестве модуляторов рецептора хемокина

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AP3113A (en) * 2008-11-26 2015-01-31 Pfizer 3-Aminocyclopentanecarboxamides as chemokine receptor modulators
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1ｒ,2ｒ,3ｒ)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
WO2015154064A2 (en) 2014-04-04 2015-10-08 Del Mar Pharmaceuticals Use of dianhydrogalactitol and analogs or derivatives thereof to treat non-small-cell carcinoma of the lung and ovarian cancer
TW201605451A (zh) * 2014-07-17 2016-02-16 參天製藥股份有限公司 老年性黃斑部病變之預防或治療劑
JOP20190040A1 (ar) * 2016-09-14 2019-03-10 Novartis Ag توليفة من ناهضات fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲（江蘇）醫藥有限公司 環戊烷化合物

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JP2012509931A (ja) 2012-04-26
MX2011005526A (es) 2011-06-06
EP2370442A1 (en) 2011-10-05
US20110144129A1 (en) 2011-06-16
CN102227429B (zh) 2014-05-28
RS52810B (sr) 2013-10-31
EP2370442B9 (en) 2013-09-04
AP2011005732A0 (en) 2011-06-30
DK2370442T5 (da) 2013-09-23
PL2370442T3 (pl) 2013-08-30
IL212732A0 (en) 2011-07-31
AP3113A (en) 2015-01-31
US8946413B2 (en) 2015-02-03
CU20110121A7 (es) 2013-05-31
TN2011000254A1 (fr) 2012-12-17
AU2009321221B2 (en) 2013-04-04
HRP20130409T1 (en) 2013-06-30
US20130197008A1 (en) 2013-08-01
EP2370442B1 (en) 2013-04-24
HRP20130409T2 (hr) 2013-11-22
RS52810B8 (sr) 2019-08-30
JP5108153B2 (ja) 2012-12-26
SI2370442T1 (sl) 2013-06-28
UA99978C2 (en) 2012-10-25
US8293903B2 (en) 2012-10-23
RS52810B9 (sr) 2019-06-28
CA2743030C (en) 2013-10-22
KR101374412B1 (ko) 2014-03-17
NZ592919A (en) 2013-05-31
EA201170721A1 (ru) 2011-12-30
ES2415430T3 (es) 2013-07-25
ECSP11011081A (es) 2011-12-30
KR20110075036A (ko) 2011-07-05
PT2370442E (pt) 2013-06-27
CY1114020T1 (el) 2016-07-27
HK1161261A1 (en) 2012-08-24
CN102227429A (zh) 2011-10-26
ZA201104069B (en) 2012-02-29
IL212732A (en) 2016-06-30
WO2010061329A1 (en) 2010-06-03
GEP20146064B (en) 2014-03-25
DOP2011000154A (es) 2011-07-31
DK2370442T3 (da) 2013-06-17
SV2011003923A (es) 2011-07-28
MY152557A (en) 2014-10-31
MA32834B1 (fr) 2011-11-01
CL2011001223A1 (es) 2011-09-02
BRPI0920936A2 (pt) 2020-08-11
ME01144B (me) 2013-03-20
CA2743030A1 (en) 2010-06-03
NI201100102A (es) 2011-09-27
CU24022B1 (es) 2014-07-30
CR20110275A (es) 2011-07-01
CO6361921A2 (es) 2012-01-20
ES2415430T9 (es) 2013-11-25
PE20110831A1 (es) 2011-11-20
AU2009321221A1 (en) 2010-06-03

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