CR20110275A - 3-aminociclopentancarboxamidas como moduladores del receptor quimiocina - Google Patents

3-aminociclopentancarboxamidas como moduladores del receptor quimiocina

Info

Publication number
CR20110275A
CR20110275A CR20110275A CR20110275A CR20110275A CR 20110275 A CR20110275 A CR 20110275A CR 20110275 A CR20110275 A CR 20110275A CR 20110275 A CR20110275 A CR 20110275A CR 20110275 A CR20110275 A CR 20110275A
Authority
CR
Costa Rica
Prior art keywords
chemiokin
aminociclopentancarboxamids
receptor modulators
compound
formula
Prior art date
Application number
CR20110275A
Other languages
English (en)
Spanish (es)
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Donald Joseph Rogier Jr
John Isidro Trujillo
Steve Ronald Turner
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CR20110275A publication Critical patent/CR20110275A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P11/00—Drugs for disorders of the respiratory system
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    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Immunology (AREA)
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CR20110275A 2008-11-26 2011-05-26 3-aminociclopentancarboxamidas como moduladores del receptor quimiocina CR20110275A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26

Publications (1)

Publication Number Publication Date
CR20110275A true CR20110275A (es) 2011-07-01

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EP (1) EP2370442B9 (enExample)
JP (1) JP5108153B2 (enExample)
KR (1) KR101374412B1 (enExample)
CN (1) CN102227429B (enExample)
AP (1) AP3113A (enExample)
AU (1) AU2009321221B2 (enExample)
BR (1) BRPI0920936A2 (enExample)
CA (1) CA2743030C (enExample)
CL (1) CL2011001223A1 (enExample)
CO (1) CO6361921A2 (enExample)
CR (1) CR20110275A (enExample)
CU (1) CU24022B1 (enExample)
CY (1) CY1114020T1 (enExample)
DK (1) DK2370442T5 (enExample)
DO (1) DOP2011000154A (enExample)
EA (1) EA020470B1 (enExample)
EC (1) ECSP11011081A (enExample)
ES (1) ES2415430T3 (enExample)
GE (1) GEP20146064B (enExample)
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PT2370442E (pt) * 2008-11-26 2013-06-27 Pfizer 3-aminociclopentanocarboxamidas como moduladores de receptor de quimiocina
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1ｒ,2ｒ,3ｒ)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
CA2946538A1 (en) 2014-04-04 2015-10-08 Del Mar Pharmaceuticals Use of dianhydrogalactitol and analogs or derivatives thereof to treat non-small-cell carcinoma of the lung and ovarian cancer
JP2016029038A (ja) * 2014-07-17 2016-03-03 参天製薬株式会社 加齢黄斑変性の予防または治療剤
JOP20190040A1 (ar) * 2016-09-14 2019-03-10 Novartis Ag توليفة من ناهضات fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲（江蘇）醫藥有限公司 環戊烷化合物

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EP2370442B9 (en) 2013-09-04
SI2370442T1 (sl) 2013-06-28
EA201170721A1 (ru) 2011-12-30
CN102227429B (zh) 2014-05-28
US8293903B2 (en) 2012-10-23
JP5108153B2 (ja) 2012-12-26
TN2011000254A1 (fr) 2012-12-17
CA2743030A1 (en) 2010-06-03
CL2011001223A1 (es) 2011-09-02
US20110144129A1 (en) 2011-06-16
AP3113A (en) 2015-01-31
IL212732A (en) 2016-06-30
MA32834B1 (fr) 2011-11-01
EA020470B1 (ru) 2014-11-28
ES2415430T3 (es) 2013-07-25
US8946413B2 (en) 2015-02-03
BRPI0920936A2 (pt) 2020-08-11
CU20110121A7 (es) 2013-05-31
ZA201104069B (en) 2012-02-29
PE20110831A1 (es) 2011-11-20
AP2011005732A0 (en) 2011-06-30
HRP20130409T1 (en) 2013-06-30
AU2009321221A1 (en) 2010-06-03
RS52810B9 (sr) 2019-06-28
NZ592919A (en) 2013-05-31
CA2743030C (en) 2013-10-22
CO6361921A2 (es) 2012-01-20
SV2011003923A (es) 2011-07-28
WO2010061329A1 (en) 2010-06-03
US20130197008A1 (en) 2013-08-01
KR20110075036A (ko) 2011-07-05
CY1114020T1 (el) 2016-07-27
GEP20146064B (en) 2014-03-25
DOP2011000154A (es) 2011-07-31
PL2370442T3 (pl) 2013-08-30
NI201100102A (es) 2011-09-27
MY152557A (en) 2014-10-31
ECSP11011081A (es) 2011-12-30
IL212732A0 (en) 2011-07-31
AU2009321221B2 (en) 2013-04-04
RS52810B8 (sr) 2019-08-30
EP2370442A1 (en) 2011-10-05
EP2370442B1 (en) 2013-04-24
DK2370442T5 (da) 2013-09-23
CU24022B1 (es) 2014-07-30
CN102227429A (zh) 2011-10-26
UA99978C2 (en) 2012-10-25
DK2370442T3 (da) 2013-06-17
JP2012509931A (ja) 2012-04-26
PT2370442E (pt) 2013-06-27
MX2011005526A (es) 2011-06-06
ME01144B (me) 2013-03-20
ES2415430T9 (es) 2013-11-25
KR101374412B1 (ko) 2014-03-17
RS52810B (sr) 2013-10-31
HK1161261A1 (en) 2012-08-24
HRP20130409T2 (hr) 2013-11-22

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