TN2011000254A1 - 3-aminocyclopentanecarboxamides servant de modulateurs de recepteurs de chimiokines - Google Patents

3-aminocyclopentanecarboxamides servant de modulateurs de recepteurs de chimiokines

Info

Publication number
TN2011000254A1
TN2011000254A1 TN2011000254A TN2011000254A TN2011000254A1 TN 2011000254 A1 TN2011000254 A1 TN 2011000254A1 TN 2011000254 A TN2011000254 A TN 2011000254A TN 2011000254 A TN2011000254 A TN 2011000254A TN 2011000254 A1 TN2011000254 A1 TN 2011000254A1
Authority
TN
Tunisia
Prior art keywords
aminocyclopentanecarboxamides
modulators
chemokine receptors
compound
formula
Prior art date
Application number
TN2011000254A
Other languages
English (en)
French (fr)
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Jr Donald Joseph Rogier
John Isidro Trujillo
Steve Ronald Turner
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of TN2011000254A1 publication Critical patent/TN2011000254A1/fr

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Hematology (AREA)
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  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Vascular Medicine (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Nutrition Science (AREA)
  • Virology (AREA)
TN2011000254A 2008-11-26 2011-05-18 3-aminocyclopentanecarboxamides servant de modulateurs de recepteurs de chimiokines TN2011000254A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26
PCT/IB2009/055232 WO2010061329A1 (en) 2008-11-26 2009-11-20 3-aminocyclopentanecarboxamides as chemokine receptor modulators

Publications (1)

Publication Number Publication Date
TN2011000254A1 true TN2011000254A1 (fr) 2012-12-17

Family

ID=41693100

Family Applications (1)

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TN2011000254A TN2011000254A1 (fr) 2008-11-26 2011-05-18 3-aminocyclopentanecarboxamides servant de modulateurs de recepteurs de chimiokines

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US (2) US8293903B2 (enExample)
EP (1) EP2370442B9 (enExample)
JP (1) JP5108153B2 (enExample)
KR (1) KR101374412B1 (enExample)
CN (1) CN102227429B (enExample)
AP (1) AP3113A (enExample)
AU (1) AU2009321221B2 (enExample)
BR (1) BRPI0920936A2 (enExample)
CA (1) CA2743030C (enExample)
CL (1) CL2011001223A1 (enExample)
CO (1) CO6361921A2 (enExample)
CR (1) CR20110275A (enExample)
CU (1) CU24022B1 (enExample)
CY (1) CY1114020T1 (enExample)
DK (1) DK2370442T5 (enExample)
DO (1) DOP2011000154A (enExample)
EA (1) EA020470B1 (enExample)
EC (1) ECSP11011081A (enExample)
ES (1) ES2415430T3 (enExample)
GE (1) GEP20146064B (enExample)
HR (1) HRP20130409T2 (enExample)
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PT (1) PT2370442E (enExample)
RS (2) RS52810B9 (enExample)
SI (1) SI2370442T1 (enExample)
SV (1) SV2011003923A (enExample)
TN (1) TN2011000254A1 (enExample)
UA (1) UA99978C2 (enExample)
WO (1) WO2010061329A1 (enExample)
ZA (1) ZA201104069B (enExample)

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TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲（江蘇）醫藥有限公司 環戊烷化合物

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MX2011005526A (es) 2011-06-06
EP2370442A1 (en) 2011-10-05
US20110144129A1 (en) 2011-06-16
CN102227429B (zh) 2014-05-28
RS52810B (sr) 2013-10-31
EP2370442B9 (en) 2013-09-04
AP2011005732A0 (en) 2011-06-30
DK2370442T5 (da) 2013-09-23
PL2370442T3 (pl) 2013-08-30
IL212732A0 (en) 2011-07-31
AP3113A (en) 2015-01-31
US8946413B2 (en) 2015-02-03
CU20110121A7 (es) 2013-05-31
AU2009321221B2 (en) 2013-04-04
HRP20130409T1 (en) 2013-06-30
US20130197008A1 (en) 2013-08-01
EP2370442B1 (en) 2013-04-24
HRP20130409T2 (hr) 2013-11-22
RS52810B8 (sr) 2019-08-30
JP5108153B2 (ja) 2012-12-26
SI2370442T1 (sl) 2013-06-28
UA99978C2 (en) 2012-10-25
US8293903B2 (en) 2012-10-23
RS52810B9 (sr) 2019-06-28
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