NI201100102A - 3 - aminociclopentancarboxamida como moduladores del receptor de quimioquinas. - Google Patents

3 - aminociclopentancarboxamida como moduladores del receptor de quimioquinas.

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Publication number
NI201100102A
NI201100102A NI201100102A NI201100102A NI201100102A NI 201100102 A NI201100102 A NI 201100102A NI 201100102 A NI201100102 A NI 201100102A NI 201100102 A NI201100102 A NI 201100102A NI 201100102 A NI201100102 A NI 201100102A
Authority
NI
Nicaragua
Prior art keywords
aminociclopentancarboxamide
receptor modulators
chemokines receptor
chemokines
compound
Prior art date
Application number
NI201100102A
Other languages
English (en)
Spanish (es)
Inventor
Venkateswaran Devraj Rajesh
Joseph Rogier Donald Jr
Huang Wei
Owen Hughes Robert
Isidro Trujillo John
Ronald Turner Steve
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NI201100102A publication Critical patent/NI201100102A/es

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
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  • Hematology (AREA)
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  • Hospice & Palliative Care (AREA)
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NI201100102A 2008-11-26 2011-05-24 3 - aminociclopentancarboxamida como moduladores del receptor de quimioquinas. NI201100102A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26

Publications (1)

Publication Number Publication Date
NI201100102A true NI201100102A (es) 2011-09-27

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NI201100102A NI201100102A (es) 2008-11-26 2011-05-24 3 - aminociclopentancarboxamida como moduladores del receptor de quimioquinas.

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EP (1) EP2370442B9 (enExample)
JP (1) JP5108153B2 (enExample)
KR (1) KR101374412B1 (enExample)
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PL2370442T3 (pl) * 2008-11-26 2013-08-30 Pfizer 3-Aminocyklopentanokarboksamidy jako modulatory receptora chemokiny
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1r,2r,3r)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
KR102359214B1 (ko) 2014-04-04 2022-02-07 델 마 파마슈티컬스 폐의 비소세포 암종 및 난소암을 치료하기 위한 디안하이드로갈락티톨 및 이의 유사체 또는 유도체
JP2016029038A (ja) * 2014-07-17 2016-03-03 参天製薬株式会社 加齢黄斑変性の予防または治療剤
PE20190972A1 (es) * 2016-09-14 2019-07-09 Novartis Ag Combinacion de agonistas de fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲(江蘇)醫藥有限公司 環戊烷化合物

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IL212732A (en) 2016-06-30
GEP20146064B (en) 2014-03-25
SI2370442T1 (sl) 2013-06-28
BRPI0920936A2 (pt) 2020-08-11
CN102227429B (zh) 2014-05-28
HK1161261A1 (en) 2012-08-24
EA020470B1 (ru) 2014-11-28
IL212732A0 (en) 2011-07-31
JP5108153B2 (ja) 2012-12-26
CU24022B1 (es) 2014-07-30
CY1114020T1 (el) 2016-07-27
MY152557A (en) 2014-10-31
HRP20130409T1 (en) 2013-06-30
EP2370442A1 (en) 2011-10-05
CO6361921A2 (es) 2012-01-20
US20130197008A1 (en) 2013-08-01
PL2370442T3 (pl) 2013-08-30
EP2370442B9 (en) 2013-09-04
US20110144129A1 (en) 2011-06-16
NZ592919A (en) 2013-05-31
HRP20130409T2 (hr) 2013-11-22
ECSP11011081A (es) 2011-12-30
AU2009321221A1 (en) 2010-06-03
RS52810B9 (sr) 2019-06-28
DK2370442T5 (da) 2013-09-23
CA2743030A1 (en) 2010-06-03
KR20110075036A (ko) 2011-07-05
AP3113A (en) 2015-01-31
MX2011005526A (es) 2011-06-06
SV2011003923A (es) 2011-07-28
AU2009321221B2 (en) 2013-04-04
ES2415430T3 (es) 2013-07-25
JP2012509931A (ja) 2012-04-26
MA32834B1 (fr) 2011-11-01
DK2370442T3 (da) 2013-06-17
ES2415430T9 (es) 2013-11-25
UA99978C2 (en) 2012-10-25
US8946413B2 (en) 2015-02-03
CL2011001223A1 (es) 2011-09-02
CN102227429A (zh) 2011-10-26
ME01144B (me) 2013-03-20
WO2010061329A1 (en) 2010-06-03
ZA201104069B (en) 2012-02-29
RS52810B8 (sr) 2019-08-30
DOP2011000154A (es) 2011-07-31
EA201170721A1 (ru) 2011-12-30
US8293903B2 (en) 2012-10-23
PE20110831A1 (es) 2011-11-20
KR101374412B1 (ko) 2014-03-17
AP2011005732A0 (en) 2011-06-30
PT2370442E (pt) 2013-06-27
CU20110121A7 (es) 2013-05-31
EP2370442B1 (en) 2013-04-24
CR20110275A (es) 2011-07-01
RS52810B (sr) 2013-10-31
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CA2743030C (en) 2013-10-22

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