RS51026B - Derivati 3-(4-amidopirol-2-ilmetiliden)-2-indolinona kao inhibitori protein kinaze - Google Patents

Derivati 3-(4-amidopirol-2-ilmetiliden)-2-indolinona kao inhibitori protein kinaze

Info

Publication number
RS51026B
RS51026B YUP-717/03A YUP71703A RS51026B RS 51026 B RS51026 B RS 51026B YU P71703 A YUP71703 A YU P71703A RS 51026 B RS51026 B RS 51026B
Authority
RS
Serbia
Prior art keywords
group
alkyl
hydrogen
hydroxy
substituted
Prior art date
Application number
YUP-717/03A
Other languages
English (en)
Serbian (sr)
Inventor
Congxin Liang
Li Sun
Peng Cho Tang
Chung Chen Wei
Michael A. Mauragis
Tomas Vojkovsky
Qingwu Jin
Paul Mattew Herrinton
Huiping Guan
Original Assignee
Sugen Inc.
Pharmacia & Upjohn Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sugen Inc., Pharmacia & Upjohn Company filed Critical Sugen Inc.
Publication of YU71703A publication Critical patent/YU71703A/sh
Publication of RS51026B publication Critical patent/RS51026B/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
YUP-717/03A 2001-02-15 2002-02-15 Derivati 3-(4-amidopirol-2-ilmetiliden)-2-indolinona kao inhibitori protein kinaze RS51026B (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26868301P 2001-02-15 2001-02-15
US31236101P 2001-08-15 2001-08-15

Publications (2)

Publication Number Publication Date
YU71703A YU71703A (sh) 2006-05-25
RS51026B true RS51026B (sr) 2010-10-31

Family

ID=26953263

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-717/03A RS51026B (sr) 2001-02-15 2002-02-15 Derivati 3-(4-amidopirol-2-ilmetiliden)-2-indolinona kao inhibitori protein kinaze

Country Status (40)

Country Link
US (4) US6653308B2 (enExample)
EP (1) EP1370554B1 (enExample)
JP (1) JP3677501B2 (enExample)
KR (1) KR100884858B1 (enExample)
CN (1) CN100338059C (enExample)
AP (1) AP1718A (enExample)
AR (1) AR042586A1 (enExample)
AT (1) ATE307128T1 (enExample)
AU (1) AU2002247133B2 (enExample)
BG (1) BG108098A (enExample)
BR (1) BR0207494A (enExample)
CA (1) CA2438314C (enExample)
CR (1) CR7056A (enExample)
CZ (1) CZ20032414A3 (enExample)
DE (1) DE60206736T2 (enExample)
DK (1) DK1370554T3 (enExample)
EA (1) EA007186B1 (enExample)
EE (1) EE200300385A (enExample)
ES (1) ES2251580T3 (enExample)
GE (1) GEP20053600B (enExample)
HR (1) HRP20030657B1 (enExample)
HU (1) HUP0303146A3 (enExample)
IL (2) IL157418A0 (enExample)
IS (1) IS2411B (enExample)
MA (1) MA26997A1 (enExample)
MX (1) MXPA03007367A (enExample)
MY (1) MY126235A (enExample)
NO (1) NO326604B1 (enExample)
NZ (1) NZ527572A (enExample)
OA (1) OA12834A (enExample)
PE (1) PE20021006A1 (enExample)
PL (1) PL364176A1 (enExample)
RS (1) RS51026B (enExample)
SI (1) SI1370554T1 (enExample)
SK (1) SK11332003A3 (enExample)
TN (1) TNSN03055A1 (enExample)
TW (1) TWI324155B (enExample)
UA (1) UA75635C2 (enExample)
WO (1) WO2002066463A1 (enExample)
ZA (2) ZA200306335B (enExample)

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