PH12012502091A1 - Process for preparing 5-biphenyl-4-amino-2-methyl pentanoic acid - Google Patents

Process for preparing 5-biphenyl-4-amino-2-methyl pentanoic acid

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Publication number
PH12012502091A1
PH12012502091A1 PH1/2012/502091A PH12012502091A PH12012502091A1 PH 12012502091 A1 PH12012502091 A1 PH 12012502091A1 PH 12012502091 A PH12012502091 A PH 12012502091A PH 12012502091 A1 PH12012502091 A1 PH 12012502091A1
Authority
PH
Philippines
Prior art keywords
amino
biphenyl
preparing
pentanoic acid
preparation
Prior art date
Application number
PH1/2012/502091A
Other languages
English (en)
Inventor
Riss Bernhard
Wietfeld Bernhard
Hook David
Sedelmeier Gottfried
Ciszewski Lech
Murlidhar Waykole Liladhar
Banziger Markus
Napp Matthias
Hawker Steven
Ruch Thomas
Original Assignee
Novartis Ag
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Filing date
Publication date
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Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PH12012502091A1 publication Critical patent/PH12012502091A1/en

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    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D207/277—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D207/28—2-Pyrrolidone-5- carboxylic acids; Functional derivatives thereof, e.g. esters, nitriles
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    • C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
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    • C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
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BRPI0806700A8 (pt) 2019-01-22
AR064842A1 (es) 2009-04-29
AU2008204546B2 (en) 2012-03-15
US20150166468A1 (en) 2015-06-18
TN2009000296A1 (en) 2010-12-31
HK1139122A1 (zh) 2010-09-10
BRPI0806700A2 (pt) 2011-09-13
PL2121578T3 (pl) 2017-02-28
MX2009007474A (es) 2009-10-08
AU2012203155B2 (en) 2014-03-20
CL2008000077A1 (es) 2008-08-18
MA31284B1 (fr) 2010-04-01
HRP20161484T1 (hr) 2016-12-16
JP2010515698A (ja) 2010-05-13
CA2674291A1 (en) 2008-07-17
WO2008083967A3 (en) 2008-08-28
CO6251311A2 (es) 2011-02-21
HUE030695T2 (en) 2017-05-29
US8993785B2 (en) 2015-03-31

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