NZ611485A - Modulators of atp-binding cassette transporters - Google Patents
Modulators of atp-binding cassette transportersInfo
- Publication number
- NZ611485A NZ611485A NZ61148507A NZ61148507A NZ611485A NZ 611485 A NZ611485 A NZ 611485A NZ 61148507 A NZ61148507 A NZ 61148507A NZ 61148507 A NZ61148507 A NZ 61148507A NZ 611485 A NZ611485 A NZ 611485A
- Authority
- NZ
- New Zealand
- Prior art keywords
- atp
- modulators
- binding cassette
- cassette transporters
- formula
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
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- Health & Medical Sciences (AREA)
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- Organic Chemistry (AREA)
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- Engineering & Computer Science (AREA)
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- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
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- Diabetes (AREA)
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- Hematology (AREA)
- Neurology (AREA)
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- Epidemiology (AREA)
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- Physics & Mathematics (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US79045906P | 2006-04-07 | 2006-04-07 | |
NZ596889A NZ596889A (en) | 2006-04-07 | 2007-04-09 | Use of amide indole derivatives as modulators of ATP-binding cassette transporters |
Publications (1)
Publication Number | Publication Date |
---|---|
NZ611485A true NZ611485A (en) | 2014-09-26 |
Family
ID=38477342
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NZ61148507A NZ611485A (en) | 2006-04-07 | 2007-04-09 | Modulators of atp-binding cassette transporters |
NZ596889A NZ596889A (en) | 2006-04-07 | 2007-04-09 | Use of amide indole derivatives as modulators of ATP-binding cassette transporters |
NZ571803A NZ571803A (en) | 2006-04-07 | 2007-04-09 | Amide indole derivatives as modulators of ATP-binding cassette transporters |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NZ596889A NZ596889A (en) | 2006-04-07 | 2007-04-09 | Use of amide indole derivatives as modulators of ATP-binding cassette transporters |
NZ571803A NZ571803A (en) | 2006-04-07 | 2007-04-09 | Amide indole derivatives as modulators of ATP-binding cassette transporters |
Country Status (22)
Families Citing this family (112)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20100074949A1 (en) | 2008-08-13 | 2010-03-25 | William Rowe | Pharmaceutical composition and administration thereof |
MXPA06002567A (es) | 2003-09-06 | 2006-09-04 | Vertex Pharma | Moduladores de transportadores con casete de union de atp. |
RU2006120549A (ru) * | 2003-11-14 | 2007-12-27 | Вертекс Фармасьютикалз Инкорпорейтед (Us) | Тиазолы и оксазолы, применяемые в качестве модуляторов транспортеров арт-связывающей кассеты |
CN1938279B (zh) * | 2004-01-30 | 2011-09-14 | 沃泰克斯药物股份有限公司 | Atp-结合弹夹转运蛋白调控剂 |
US7977322B2 (en) | 2004-08-20 | 2011-07-12 | Vertex Pharmaceuticals Incorporated | Modulators of ATP-binding cassette transporters |
CN101006076B (zh) | 2004-06-24 | 2010-09-29 | 沃泰克斯药物股份有限公司 | Atp-结合弹夹转运蛋白的调控剂 |
NZ566208A (en) | 2005-08-11 | 2010-09-30 | Vertex Pharma | 2-Thiazolamide derivatives as modulators of cystic fibrosis transmembrane conductance regulators |
EP2774925B1 (en) | 2005-11-08 | 2016-12-28 | Vertex Pharmaceuticals Incorporated | Heterocyclic modulators of ATP-binding cassette transporters |
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